AR095035A1 - Uso de un agonista del receptor 2 del péptido formilo para la preparación de una composición farmacéutica para el tratamiento de inflamación y enfermedades dérmicas - Google Patents
Uso de un agonista del receptor 2 del péptido formilo para la preparación de una composición farmacéutica para el tratamiento de inflamación y enfermedades dérmicasInfo
- Publication number
- AR095035A1 AR095035A1 ARP140100733A ARP140100733A AR095035A1 AR 095035 A1 AR095035 A1 AR 095035A1 AR P140100733 A ARP140100733 A AR P140100733A AR P140100733 A ARP140100733 A AR P140100733A AR 095035 A1 AR095035 A1 AR 095035A1
- Authority
- AR
- Argentina
- Prior art keywords
- dermal
- treatment
- halogen
- healing
- pharmaceutical composition
- Prior art date
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- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/196—Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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- Dermatology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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| MX376348B (es) | 2011-10-26 | 2025-03-07 | Allergan Inc | Derivados de amida de aminoacidos sustituidos con n-urea como moduladores de receptor de tipo peptido receptor de formilo-1 (fprl-1). |
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| MA37618B1 (fr) | 2012-05-16 | 2017-08-31 | Actelion Pharmaceuticals Ltd | Dérivés pontés fluorés de spiro[2.4]heptane en tant qu'agonistes de récepteur alx |
| EP2850058B1 (en) | 2012-05-16 | 2016-07-13 | Actelion Pharmaceuticals Ltd. | 1-(p-tolyl)cyclopropyl substituted bridged spiro[2.4]heptane derivatives as alx receptor agonists |
| CN103665043B (zh) | 2012-08-30 | 2017-11-10 | 江苏豪森药业集团有限公司 | 一种替诺福韦前药及其在医药上的应用 |
| KR20210024691A (ko) * | 2013-03-06 | 2021-03-05 | 알러간, 인코포레이티드 | 피부 질환 치료용 포르밀 펩티드 수용체 2의 항진제의 용도 |
| AR096686A1 (es) | 2013-06-25 | 2016-01-27 | Actelion Pharmaceuticals Ltd | Derivados de espiro[2.4]heptano puenteados sustituidos con difluoroetil-oxazol como agonistas del receptor de alx |
| EP3022174B1 (en) * | 2013-07-16 | 2018-09-05 | Allergan, Inc. | Derivatives of n-urea substituted amino acids as formyl peptide receptor modulators |
| BR112016001106A8 (pt) | 2013-07-18 | 2017-12-26 | Actelion Pharmaceuticals Ltd | Derivados de espiro [2,4] heptano interligados piperazina substituídos como agonistas do receptor de alx |
| AR097279A1 (es) | 2013-08-09 | 2016-03-02 | Actelion Pharmaceuticals Ltd | Derivados de benzimidazolil-metil urea como agonistas del receptor de alx |
| WO2015116566A1 (en) * | 2014-01-29 | 2015-08-06 | Allergan, Inc. | 2,5-dioxoimidazolidin-1-yl-3-urea derivatives as formyl peptide modulators |
| US9663457B2 (en) | 2014-04-09 | 2017-05-30 | Allergan, Inc. | Carbamoyl hydrazine derivatives as formyl peptide modulators |
| EP3145916B1 (en) | 2014-05-21 | 2020-02-12 | Allergan, Inc. | Imidazole derivatives as formyl peptide receptor modulators |
| BR112018011046A2 (pt) * | 2015-12-10 | 2018-11-21 | Bristol-Myers Squibb Company | agonistas receptores de piperidinona formil peptí-deo 2 e de formil peptídeo 1 |
| CA3017967A1 (en) | 2016-03-28 | 2017-10-05 | Allergan, Inc. | Phenyl urea derivatives as n-formyl peptide receptor modulators |
| JP2019515901A (ja) * | 2016-04-12 | 2019-06-13 | アラーガン、インコーポレイテッドAllergan,Incorporated | N−ホルミルペプチド受容体モジュレータとしてのフェニル尿素誘導体 |
| MX2019003867A (es) | 2016-10-06 | 2019-08-05 | Daiichi Sankyo Co Ltd | Derivado de urea. |
| GB2561540A (en) * | 2017-03-13 | 2018-10-24 | Nodthera Ltd | Chemical compounds |
| ES2799098B2 (es) * | 2019-06-10 | 2021-12-10 | Univ Madrid Carlos Iii | Aptameros agonistas del receptor fpr2 y usos de los mismos |
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| DE10005275A1 (de) * | 2000-02-07 | 2001-08-09 | Bayer Ag | Neuartige Glycokonjugate |
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| KR20210024691A (ko) * | 2013-03-06 | 2021-03-05 | 알러간, 인코포레이티드 | 피부 질환 치료용 포르밀 펩티드 수용체 2의 항진제의 용도 |
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2014
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- 2014-03-04 WO PCT/US2014/020273 patent/WO2014138046A1/en not_active Ceased
- 2014-03-04 CA CA3114477A patent/CA3114477A1/en not_active Abandoned
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- 2014-03-04 JP JP2015561540A patent/JP6196328B2/ja not_active Expired - Fee Related
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- 2014-03-04 KR KR1020157024039A patent/KR102223384B1/ko not_active Expired - Fee Related
- 2014-03-04 AU AU2014226001A patent/AU2014226001B2/en not_active Ceased
- 2014-03-04 CA CA2899804A patent/CA2899804A1/en not_active Abandoned
- 2014-03-04 HK HK16107753.4A patent/HK1219661A1/zh unknown
- 2014-03-04 CN CN201480011861.8A patent/CN105007908B/zh not_active Expired - Fee Related
- 2014-03-04 CN CN201711029910.2A patent/CN107714683A/zh active Pending
- 2014-03-04 RU RU2015134778A patent/RU2696487C2/ru active
- 2014-03-04 BR BR112015021392-8A patent/BR112015021392B1/pt not_active IP Right Cessation
- 2014-03-04 BR BR122017004256A patent/BR122017004256A2/pt not_active Application Discontinuation
- 2014-03-04 EP EP14713302.9A patent/EP2964214A1/en not_active Withdrawn
- 2014-03-06 TW TW103107759A patent/TW201446241A/zh unknown
- 2014-03-06 AR ARP140100733A patent/AR095035A1/es unknown
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2017
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2021
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