AR087742A1 - Compuestos de hexahidropirano[3,4-d][1,3]tiazin-2-amina - Google Patents

Compuestos de hexahidropirano[3,4-d][1,3]tiazin-2-amina

Info

Publication number
AR087742A1
AR087742A1 ARP120103210A ARP120103210A AR087742A1 AR 087742 A1 AR087742 A1 AR 087742A1 AR P120103210 A ARP120103210 A AR P120103210A AR P120103210 A ARP120103210 A AR P120103210A AR 087742 A1 AR087742 A1 AR 087742A1
Authority
AR
Argentina
Prior art keywords
alkyl
hydrogen
r5ar5b
cycloalkyl
optionally substituted
Prior art date
Application number
ARP120103210A
Other languages
English (en)
Spanish (es)
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of AR087742A1 publication Critical patent/AR087742A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
ARP120103210A 2011-08-31 2012-08-30 Compuestos de hexahidropirano[3,4-d][1,3]tiazin-2-amina AR087742A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201161529367P 2011-08-31 2011-08-31

Publications (1)

Publication Number Publication Date
AR087742A1 true AR087742A1 (es) 2014-04-16

Family

ID=47010661

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP120103210A AR087742A1 (es) 2011-08-31 2012-08-30 Compuestos de hexahidropirano[3,4-d][1,3]tiazin-2-amina

Country Status (8)

Country Link
US (2) US8933221B2 (enExample)
EP (1) EP2751116B1 (enExample)
JP (1) JP6043355B2 (enExample)
AR (1) AR087742A1 (enExample)
ES (1) ES2605565T3 (enExample)
TW (1) TW201326182A (enExample)
UY (1) UY34302A (enExample)
WO (1) WO2013030713A1 (enExample)

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JP2018531923A (ja) * 2015-09-24 2018-11-01 ファイザー・インク Ｎ−［２−（２−アミノ−６，６−二置換−４，４ａ，５，６−テトラヒドロピラノ［３，４−ｄ］［１，３］チアジン−８ａ（８Ｈ）−イル）−１，３−チアゾール−４−イル］アミド
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Also Published As

Publication number Publication date
US20150087637A1 (en) 2015-03-26
US9550795B2 (en) 2017-01-24
WO2013030713A1 (en) 2013-03-07
UY34302A (es) 2013-04-05
EP2751116B1 (en) 2016-10-12
JP2014525432A (ja) 2014-09-29
US20130053373A1 (en) 2013-02-28
EP2751116A1 (en) 2014-07-09
ES2605565T3 (es) 2017-03-15
TW201326182A (zh) 2013-07-01
JP6043355B2 (ja) 2016-12-14
US8933221B2 (en) 2015-01-13

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