AR064735A1 - Agonistas de gpcr y composicion farmaceutica en base al compuesto - Google Patents

Agonistas de gpcr y composicion farmaceutica en base al compuesto

Info

Publication number
AR064735A1
AR064735A1 ARP080100017A ARP080100017A AR064735A1 AR 064735 A1 AR064735 A1 AR 064735A1 AR P080100017 A ARP080100017 A AR P080100017A AR P080100017 A ARP080100017 A AR P080100017A AR 064735 A1 AR064735 A1 AR 064735A1
Authority
AR
Argentina
Prior art keywords
compound
pharmaceutical composition
composition based
gpcr agonists
alkyl
Prior art date
Application number
ARP080100017A
Other languages
English (en)
Spanish (es)
Original Assignee
Prosidion Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0700125A external-priority patent/GB0700125D0/en
Priority claimed from GB0708746A external-priority patent/GB0708746D0/en
Priority claimed from GB0719763A external-priority patent/GB0719763D0/en
Application filed by Prosidion Ltd filed Critical Prosidion Ltd
Publication of AR064735A1 publication Critical patent/AR064735A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
ARP080100017A 2007-01-04 2008-01-03 Agonistas de gpcr y composicion farmaceutica en base al compuesto AR064735A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0700125A GB0700125D0 (en) 2007-01-04 2007-01-04 GPCR agonists
GB0708746A GB0708746D0 (en) 2007-05-08 2007-05-08 GPCR agonists
GB0719763A GB0719763D0 (en) 2007-10-10 2007-10-10 GPCR agonists

Publications (1)

Publication Number Publication Date
AR064735A1 true AR064735A1 (es) 2009-04-22

Family

ID=39199058

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP080100017A AR064735A1 (es) 2007-01-04 2008-01-03 Agonistas de gpcr y composicion farmaceutica en base al compuesto

Country Status (20)

Country Link
US (1) US20100105732A1 (Direct)
EP (2) EP2114935B1 (Direct)
JP (1) JP2010514831A (Direct)
AR (1) AR064735A1 (Direct)
AT (1) ATE517103T1 (Direct)
BR (1) BRPI0806500A2 (Direct)
CA (1) CA2674455A1 (Direct)
CL (1) CL2008000018A1 (Direct)
CY (1) CY1112474T1 (Direct)
DK (1) DK2114935T3 (Direct)
EA (1) EA015130B1 (Direct)
HR (1) HRP20110750T1 (Direct)
PE (1) PE20081659A1 (Direct)
PL (1) PL2114935T3 (Direct)
PT (1) PT2114935E (Direct)
RS (1) RS51943B (Direct)
SA (1) SA08280757B1 (Direct)
SI (1) SI2114935T1 (Direct)
TW (1) TW200835482A (Direct)
WO (1) WO2008081207A1 (Direct)

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* Cited by examiner, † Cited by third party
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AU2006264649A1 (en) * 2005-06-30 2007-01-11 Prosidion Limited GPCR agonists
CL2008000017A1 (es) * 2007-01-04 2008-08-01 Prosidion Ltd Compuestos derivados de heterociclos de nitrogeno y oxigeno, agonistas de gpcr; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de la obesidad, diabetes, sindrome metabolico, hiperlipidemia, toleranci
JP2010539152A (ja) 2007-09-10 2010-12-16 プロシディオン・リミテッド 代謝障害の治療のための化合物
WO2009047264A1 (en) 2007-10-10 2009-04-16 Novartis Ag Spiropyrrolidines and their use against hcv and hiv infection
GB0812649D0 (en) * 2008-07-10 2008-08-20 Prosidion Ltd Compounds
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GB0904285D0 (en) 2009-03-12 2009-04-22 Prosidion Ltd Compounds for the treatment of metabolic disorders
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GB0904284D0 (en) 2009-03-12 2009-04-22 Prosidion Ltd Compounds for the treatment of metabolic disorders
JP2012530758A (ja) 2009-06-24 2012-12-06 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規化合物、医薬組成物及びそれに関する方法
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TW201209054A (en) 2010-05-28 2012-03-01 Prosidion Ltd Novel compounds
WO2011157827A1 (de) 2010-06-18 2011-12-22 Sanofi Azolopyridin-3-on-derivate als inhibitoren von lipasen und phospholipasen
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GB201114389D0 (en) 2011-08-22 2011-10-05 Prosidion Ltd Novel compounds
AR083904A1 (es) 2010-11-18 2013-04-10 Prosidion Ltd Derivados de 1,4-pirrolidinas disustituidos y 3-il-aminas y sus usos en el tratamiento de desordenes metabolicos
KR101913619B1 (ko) 2011-06-09 2018-12-28 리젠 파마슈티컬스 소시에떼 아노님 Gpr-119의 조절제로서의 신규한 화합물
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CL2008000017A1 (es) * 2007-01-04 2008-08-01 Prosidion Ltd Compuestos derivados de heterociclos de nitrogeno y oxigeno, agonistas de gpcr; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de la obesidad, diabetes, sindrome metabolico, hiperlipidemia, toleranci

Also Published As

Publication number Publication date
EP2114935A1 (en) 2009-11-11
HK1135705A1 (en) 2010-06-11
JP2010514831A (ja) 2010-05-06
RS51943B (sr) 2012-02-29
EA015130B1 (ru) 2011-06-30
PT2114935E (pt) 2011-10-17
ATE517103T1 (de) 2011-08-15
SA08280757B1 (ar) 2011-01-15
HRP20110750T1 (hr) 2011-11-30
EP2114935B1 (en) 2011-07-20
PE20081659A1 (es) 2008-10-24
TW200835482A (en) 2008-09-01
EA200900880A1 (ru) 2010-02-26
PL2114935T3 (pl) 2012-03-30
US20100105732A1 (en) 2010-04-29
CL2008000018A1 (es) 2008-08-01
DK2114935T3 (da) 2011-10-31
CA2674455A1 (en) 2008-07-10
SI2114935T1 (sl) 2011-11-30
EP2377864A1 (en) 2011-10-19
WO2008081207A1 (en) 2008-07-10
BRPI0806500A2 (pt) 2014-04-22
CY1112474T1 (el) 2015-12-09

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