AR037371A1 - Compuesto macrolida, proceso para su preparacion, composicion farmaceutica que lo comprende y su uso para la preparacion de un medicamento - Google Patents
Compuesto macrolida, proceso para su preparacion, composicion farmaceutica que lo comprende y su uso para la preparacion de un medicamentoInfo
- Publication number
- AR037371A1 AR037371A1 ARP020104364A ARP020104364A AR037371A1 AR 037371 A1 AR037371 A1 AR 037371A1 AR P020104364 A ARP020104364 A AR P020104364A AR P020104364 A ARP020104364 A AR P020104364A AR 037371 A1 AR037371 A1 AR 037371A1
- Authority
- AR
- Argentina
- Prior art keywords
- hydrogen
- optionally substituted
- alkyl
- bicyclic heteroaryl
- hydroxy
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0127349.9A GB0127349D0 (en) | 2001-11-14 | 2001-11-14 | Macrolides |
Publications (1)
Publication Number | Publication Date |
---|---|
AR037371A1 true AR037371A1 (es) | 2004-11-03 |
Family
ID=9925777
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP020104364A AR037371A1 (es) | 2001-11-14 | 2002-11-13 | Compuesto macrolida, proceso para su preparacion, composicion farmaceutica que lo comprende y su uso para la preparacion de un medicamento |
Country Status (20)
Country | Link |
---|---|
US (1) | US7202221B2 (hu) |
EP (1) | EP1453846B1 (hu) |
JP (1) | JP2005515978A (hu) |
CN (1) | CN1307194C (hu) |
AR (1) | AR037371A1 (hu) |
AT (1) | ATE362479T1 (hu) |
BR (1) | BR0214132A (hu) |
CA (1) | CA2466975A1 (hu) |
DE (1) | DE60220180T2 (hu) |
EA (1) | EA007433B1 (hu) |
ES (1) | ES2287332T3 (hu) |
GB (1) | GB0127349D0 (hu) |
HR (1) | HRP20040433A2 (hu) |
HU (1) | HUP0402225A3 (hu) |
IL (1) | IL161710A0 (hu) |
PL (1) | PL371472A1 (hu) |
RS (1) | RS41904A (hu) |
UA (1) | UA77210C2 (hu) |
WO (1) | WO2003042228A1 (hu) |
ZA (1) | ZA200403684B (hu) |
Families Citing this family (31)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6995143B2 (en) * | 2002-02-28 | 2006-02-07 | Basilea Pharmaceutica Ag | Macrolides with antibacterial activity |
WO2005070918A1 (en) | 2002-05-13 | 2005-08-04 | Enanta Pharmaceuticals, Inc. | Process for the preparation of t-11 bicyclic erythromycin derivatives |
US6764998B1 (en) | 2003-06-18 | 2004-07-20 | Enanta Pharmaceuticals, Inc. | 6,11-4C-bicyclic 9a-azalide derivatives |
US7135573B2 (en) | 2002-05-13 | 2006-11-14 | Enanta Pharmaceuticals, Inc. | Processes for the preparation of O-(6-Pyrazol-1-yl-pyridin-3-ylmethyl)-hydroxylamine |
US7910558B2 (en) | 2002-05-13 | 2011-03-22 | Enanta Pharmaceuticals, Inc. | Bridged macrocyclic compounds and processes for the preparation thereof |
DK1503759T3 (da) * | 2002-05-14 | 2009-04-14 | Univ California | Substituerede quinoloncarboxylsyrer, deres derivater, virkningssted og anvendelser heraf |
US7091196B2 (en) | 2002-09-26 | 2006-08-15 | Rib-X Pharmaceuticals, Inc. | Bifunctional heterocyclic compounds and methods of making and using same |
GB0225384D0 (en) * | 2002-10-31 | 2002-12-11 | Glaxo Group Ltd | Novel compounds |
US6645941B1 (en) | 2003-03-26 | 2003-11-11 | Enanta Pharmaceuticals, Inc. | 6,11-3C-bicyclic 9a-azalide derivatives |
GB0310980D0 (en) * | 2003-05-13 | 2003-06-18 | Glaxo Group Ltd | Novel compounds |
US20070293472A1 (en) * | 2003-05-13 | 2007-12-20 | Glaxo Group Limited | Novel 14 and 15 Membered Ring Compounds |
GB0310986D0 (en) | 2003-05-13 | 2003-06-18 | Glaxo Group Ltd | Novel compounds |
GB0310979D0 (en) * | 2003-05-13 | 2003-06-18 | Glaxo Group Ltd | Novel compounds |
GB0310984D0 (en) * | 2003-05-13 | 2003-06-18 | Glaxo Group Ltd | Novel compounds |
US7276487B2 (en) | 2003-09-23 | 2007-10-02 | Enanta Pharmaceuticals, Inc. | 9a, 11-3C-bicyclic 9a-azalide derivatives |
WO2005070113A2 (en) | 2004-01-09 | 2005-08-04 | Enanta Pharmaceuticals, Inc. | 9n-substituted 6-11 bicyclic erythromycin derivatives |
EP1723159B1 (en) | 2004-02-27 | 2019-06-12 | Melinta Therapeutics, Inc. | Macrocyclic compounds and methods of making and using the same |
EP1756134A1 (en) * | 2004-05-06 | 2007-02-28 | GlaxoSmithKline istrazivacki centar Zagreb d.o.o. | Carbamate linked macrolides useful for the treatment of microbial infections |
WO2005108412A1 (en) * | 2004-05-06 | 2005-11-17 | Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. | Ester linked macrolides useful for the treatment of microbial infections |
WO2006047167A2 (en) * | 2004-10-21 | 2006-05-04 | Janssen Pharmaceutica, N.V. | 9 alkyl and 9 alkylidenyl 6-0 alkyl-11, 12 carbamate ketolide antimicrobials |
GB0424961D0 (en) * | 2004-11-11 | 2004-12-15 | Glaxo Group Ltd | Novel compounds |
GB0424951D0 (en) * | 2004-11-11 | 2004-12-15 | Glaxo Group Ltd | Novel compounds |
GB0424959D0 (en) * | 2004-11-11 | 2004-12-15 | Glaxo Group Ltd | Novel compounds |
GB0424958D0 (en) * | 2004-11-11 | 2004-12-15 | Glaxo Group Ltd | Novel compounds |
PL2049556T3 (pl) | 2006-08-09 | 2013-12-31 | Basilea Pharmaceutica Ag | Nowe makrolidy użyteczne przeciw chorobom zapalnym i alergicznym |
CN101541331A (zh) | 2006-08-24 | 2009-09-23 | 沃克哈特研究中心 | 具有抗微生物活性的新颖大环内酯和酮内酯 |
BRPI0908343A2 (pt) | 2008-02-08 | 2020-08-18 | Basilea Pharmaceutica Ag | macrolídeos e seu uso |
MX2011012614A (es) | 2009-05-27 | 2012-02-22 | Wockhardt Ltd | Compuestos de quetolida que tienen actividad antimicrobiana. |
RU2601550C2 (ru) | 2010-12-09 | 2016-11-10 | Вокхардт Лимитед | Кетолидные соединения |
KR20140004187A (ko) * | 2011-01-31 | 2014-01-10 | 메이지 세이카 파루마 가부시키가이샤 | 신규 마크로라이드 유도체 |
JP5718488B2 (ja) | 2011-03-01 | 2015-05-13 | ウォックハート リミテッド | ケトライド中間体の調製方法 |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0126344A2 (en) | 1983-05-20 | 1984-11-28 | Abbott Laboratories | Tripeptide esters of therapeutic agents |
US4742049A (en) * | 1986-06-04 | 1988-05-03 | Abbott Laboratories | Semisynthetic erythromycin antibiotics |
NZ233117A (en) | 1989-03-28 | 1991-05-28 | Abbott Lab | 9-deoxo-9,12-epoxy-erythromycin derivatives and pharmaceutical compositions |
CA2064634C (en) * | 1991-04-04 | 1998-08-04 | James V. Heck | 9-deoxo-8a-aza-8a-homoerythromycin a derivatives modified at the 4"- and8a-positions |
EP1007530B1 (en) | 1996-05-07 | 2005-11-16 | Abbott Laboratories | 6-o-substituted erythromycin compounds and method for making same |
EP0895999A1 (en) * | 1997-08-06 | 1999-02-10 | Pfizer Products Inc. | C-4" substituted macrolide antibiotics |
US6262030B1 (en) | 1998-11-03 | 2001-07-17 | Pfizer Inc. | Erythromycin derivatives |
HUP0201516A3 (en) | 1999-05-24 | 2003-03-28 | Pfizer Prod Inc | 13-methyl-erythromycin derivatives, process for their preparation and pharmaceutical compositions containing them |
AU6748500A (en) | 1999-08-24 | 2001-03-19 | Abbott Laboratories | 9a-azalides with antibacterial activity |
CA2398848C (en) | 2000-02-24 | 2007-09-25 | Abbott Laboratories | Anti-infective agents useful against multidrug-resistant strains of bacteria |
US6946446B2 (en) | 2000-02-24 | 2005-09-20 | Abbott Laboratories | Anti-infective agents useful against multidrug-resistant strains of bacteria |
JP2002173498A (ja) | 2000-09-27 | 2002-06-21 | Hokuriku Seiyaku Co Ltd | エリスロマイシン誘導体 |
GB0025688D0 (en) | 2000-10-19 | 2000-12-06 | Glaxo Group Ltd | Macrolides |
-
2001
- 2001-11-14 GB GBGB0127349.9A patent/GB0127349D0/en not_active Ceased
-
2002
- 2002-11-13 WO PCT/GB2002/005101 patent/WO2003042228A1/en active IP Right Grant
- 2002-11-13 CA CA002466975A patent/CA2466975A1/en not_active Abandoned
- 2002-11-13 EA EA200400536A patent/EA007433B1/ru not_active IP Right Cessation
- 2002-11-13 BR BR0214132-9A patent/BR0214132A/pt not_active IP Right Cessation
- 2002-11-13 PL PL02371472A patent/PL371472A1/xx not_active Application Discontinuation
- 2002-11-13 EP EP02779670A patent/EP1453846B1/en not_active Expired - Lifetime
- 2002-11-13 RS YU41904A patent/RS41904A/sr unknown
- 2002-11-13 JP JP2003544063A patent/JP2005515978A/ja active Pending
- 2002-11-13 DE DE60220180T patent/DE60220180T2/de not_active Expired - Fee Related
- 2002-11-13 ES ES02779670T patent/ES2287332T3/es not_active Expired - Lifetime
- 2002-11-13 HU HU0402225A patent/HUP0402225A3/hu unknown
- 2002-11-13 AR ARP020104364A patent/AR037371A1/es unknown
- 2002-11-13 US US10/495,413 patent/US7202221B2/en not_active Expired - Fee Related
- 2002-11-13 AT AT02779670T patent/ATE362479T1/de not_active IP Right Cessation
- 2002-11-13 CN CNB028270452A patent/CN1307194C/zh not_active Expired - Fee Related
- 2002-11-13 UA UA20040503313A patent/UA77210C2/uk unknown
- 2002-11-13 IL IL16171002A patent/IL161710A0/xx unknown
-
2004
- 2004-05-13 ZA ZA200403684A patent/ZA200403684B/xx unknown
- 2004-05-14 HR HR20040433A patent/HRP20040433A2/hr not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
PL371472A1 (en) | 2005-06-13 |
GB0127349D0 (en) | 2002-01-02 |
ATE362479T1 (de) | 2007-06-15 |
ES2287332T3 (es) | 2007-12-16 |
EA007433B1 (ru) | 2006-10-27 |
US20050080025A1 (en) | 2005-04-14 |
BR0214132A (pt) | 2004-09-14 |
EA200400536A1 (ru) | 2004-12-30 |
CN1612888A (zh) | 2005-05-04 |
DE60220180T2 (de) | 2008-01-17 |
RS41904A (en) | 2006-10-27 |
UA77210C2 (en) | 2006-11-15 |
IL161710A0 (en) | 2004-09-27 |
ZA200403684B (en) | 2005-09-13 |
CN1307194C (zh) | 2007-03-28 |
US7202221B2 (en) | 2007-04-10 |
CA2466975A1 (en) | 2003-05-22 |
DE60220180D1 (de) | 2007-06-28 |
HRP20040433A2 (en) | 2005-04-30 |
JP2005515978A (ja) | 2005-06-02 |
HUP0402225A2 (hu) | 2005-02-28 |
HUP0402225A3 (en) | 2006-01-30 |
EP1453846A1 (en) | 2004-09-08 |
EP1453846B1 (en) | 2007-05-16 |
WO2003042228A1 (en) | 2003-05-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |