AP726A - Process and intermediates for preparing substituted chromanol derivatives. - Google Patents

Process and intermediates for preparing substituted chromanol derivatives. Download PDF

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Publication number
AP726A
AP726A APAP/P/1997/001083A AP9701083A AP726A AP 726 A AP726 A AP 726A AP 9701083 A AP9701083 A AP 9701083A AP 726 A AP726 A AP 726A
Authority
AP
ARIPO
Prior art keywords
compound
alkyl
formula
phenyl
enantiomer
Prior art date
Application number
APAP/P/1997/001083A
Other languages
English (en)
Other versions
AP9701083A0 (en
Inventor
Anthony D Piscopio
Joel M Hawkins
Stephane Caron
Sarah E Kelly
Jeffrey W Raggon
Michael J Castaldi
Robert W Dugger
Sally G Ruggeri
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of AP9701083A0 publication Critical patent/AP9701083A0/xx
Application granted granted Critical
Publication of AP726A publication Critical patent/AP726A/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00—Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40—Halogenated unsaturated alcohols
    • C07C33/50—Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22—Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
APAP/P/1997/001083A 1996-09-16 1997-09-11 Process and intermediates for preparing substituted chromanol derivatives. AP726A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2637296P 1996-09-16 1996-09-16

Publications (2)

Publication Number Publication Date
AP9701083A0 AP9701083A0 (en) 1997-10-31
AP726A true AP726A (en) 1999-01-29

Family

ID=21831429

Family Applications (1)

Application Number Title Priority Date Filing Date
APAP/P/1997/001083A AP726A (en) 1996-09-16 1997-09-11 Process and intermediates for preparing substituted chromanol derivatives.

Country Status (39)

Country Link
US (4) US6096906A (sk)
EP (1) EP0925292B1 (sk)
JP (1) JP3117730B2 (sk)
KR (1) KR100339164B1 (sk)
CN (1) CN1108298C (sk)
AP (1) AP726A (sk)
AT (1) ATE249452T1 (sk)
AU (1) AU713701B2 (sk)
BG (1) BG63542B1 (sk)
BR (1) BR9711482A (sk)
CA (1) CA2265043C (sk)
CO (1) CO4600635A1 (sk)
DE (1) DE69724801T2 (sk)
DK (1) DK0925292T3 (sk)
DZ (1) DZ2308A1 (sk)
EA (1) EA002204B1 (sk)
ES (1) ES2206738T3 (sk)
GT (3) GT199700104A (sk)
HN (1) HN1997000127A (sk)
HR (1) HRP970497B1 (sk)
ID (1) ID19613A (sk)
IL (1) IL128732A0 (sk)
IS (1) IS4980A (sk)
MA (1) MA24319A1 (sk)
NO (1) NO991254L (sk)
NZ (1) NZ334214A (sk)
OA (1) OA10995A (sk)
PA (1) PA8437901A1 (sk)
PE (1) PE109798A1 (sk)
PL (1) PL332351A1 (sk)
PT (1) PT925292E (sk)
SK (1) SK31399A3 (sk)
TN (1) TNSN97155A1 (sk)
TR (1) TR199900592T2 (sk)
TW (1) TW449579B (sk)
UA (1) UA58520C2 (sk)
WO (1) WO1998011085A1 (sk)
YU (1) YU13299A (sk)
ZA (1) ZA978291B (sk)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6436987B1 (en) * 2000-06-08 2002-08-20 Pfizer Inc. Crystalline forms of (3S-trans)-2-[3,4-dihydro-4-hydroxy-3-(phenylmethyl)-2H-1-benzopyran-7-yl]-4-(trifluoromethyl)-benzoic acid
CA2433516A1 (en) * 2001-01-30 2002-08-08 Keith Michael Devries Processes for preparing chromanylbenzoic acids
AU4239302A (en) * 2001-06-28 2003-01-02 Pfizer Products Inc. Benzoic acid substituted benzopyrans for the treatment of atherosclerosis
ES2551916T3 (es) * 2007-07-23 2015-11-24 The Board Of Trustees Of The University Of Illinois Sistema para controlar la reactividad de los ácidos borónicos
US8338601B2 (en) * 2008-09-26 2012-12-25 Board Of Trustees Of The University Of Illinois Slow release of organoboronic acids in cross-coupling reactions
US8350099B2 (en) 2009-09-02 2013-01-08 E I Du Pont De Nemours And Company Fluorovinyl ether functionalized aromatic diesters, derivatives thereof, and process for the preparation thereof
US8378061B2 (en) * 2009-09-02 2013-02-19 E.I. Du Pont De Nemours And Company Polyester films with improved oil repellency
US20110218319A1 (en) * 2009-09-02 2011-09-08 E. I. Du Pont De Nemours And Company Polyaramid films comprising fluorovinylether functionalized aromatic moieties
TW201113311A (en) * 2009-09-02 2011-04-16 Du Pont Polyaramid films comprising fluorovinylether functionalized aromatic moieties
AU2010289583A1 (en) * 2009-09-02 2012-03-15 E. I. Du Pont De Nemours And Company Polyesters comprising fluorovinylether functionalized aromatic moieties
WO2011028766A2 (en) * 2009-09-02 2011-03-10 E. I. Du Pont De Nemours And Company Fluorinated 4-oxo-chroman-carboxylates
WO2011103435A2 (en) 2010-02-18 2011-08-25 The Board Of Trustees Of The University Of Illinois Methods for forming protected organoboronic acids
US10500178B2 (en) 2015-03-13 2019-12-10 The Board Of Trustees Of The Leland Stanford Junior University LTB4 inhibition to prevent and treat human lymphedema

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996011925A1 (en) * 1994-10-13 1996-04-25 Pfizer Inc. Benzopyran and benzo-fused compounds, their preparation and their use as leukotriene b4' (ltb4) antagonists
WO1996011920A1 (en) * 1994-10-13 1996-04-25 Pfizer Inc. Benzopyran and benzo-fused compounds, their preparation and their use as leukotriene b4 (ltb4) antagonists
WO1996016955A1 (en) * 1994-11-30 1996-06-06 Pfizer Inc. Processes and intermediates for preparing cis(+)3-[4,-6-dihydroxychroman-3-ylmethyl]-4-methoxyaniline

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9119920D0 (en) * 1991-09-18 1991-10-30 Glaxo Group Ltd Chemical compounds
MX9300312A (es) * 1992-01-23 1993-07-31 Pfizer Antagonistas benzopiranicos y relacionado de ltb.
WO1993015066A1 (en) * 1992-01-23 1993-08-05 Pfizer Inc. Benzopyran and related ltb4 antagonists
BR9307277A (pt) * 1992-10-21 1999-05-11 Pfizer Derivados sulfonamida de compostos de anel cicloalquílico e heterocíclico substituído com hidróxi condensado com benzeno
JPH07507811A (ja) * 1992-10-21 1995-08-31 ファイザー・インク． 鏡像異性のシス−３−（４，６−ジヒドロキシクロマン−３−イル−メチル）安息香酸

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1996011925A1 (en) * 1994-10-13 1996-04-25 Pfizer Inc. Benzopyran and benzo-fused compounds, their preparation and their use as leukotriene b4' (ltb4) antagonists
WO1996011920A1 (en) * 1994-10-13 1996-04-25 Pfizer Inc. Benzopyran and benzo-fused compounds, their preparation and their use as leukotriene b4 (ltb4) antagonists
WO1996016955A1 (en) * 1994-11-30 1996-06-06 Pfizer Inc. Processes and intermediates for preparing cis(+)3-[4,-6-dihydroxychroman-3-ylmethyl]-4-methoxyaniline

Also Published As

Publication number Publication date
DZ2308A1 (fr) 2002-12-28
DE69724801T2 (de) 2004-06-17
DK0925292T3 (da) 2004-01-12
CO4600635A1 (es) 1998-05-08
US20020099227A1 (en) 2002-07-25
EA002204B1 (ru) 2002-02-28
JP3117730B2 (ja) 2000-12-18
ZA978291B (en) 1999-03-15
CA2265043C (en) 2003-01-14
NZ334214A (en) 2000-09-29
BR9711482A (pt) 1999-08-24
AU3781497A (en) 1998-04-02
JP2000502726A (ja) 2000-03-07
ES2206738T3 (es) 2004-05-16
BG63542B1 (bg) 2002-04-30
TR199900592T2 (xx) 1999-06-21
TW449579B (en) 2001-08-11
NO991254D0 (no) 1999-03-15
TNSN97155A1 (fr) 2005-03-15
PT925292E (pt) 2004-01-30
EA199900204A1 (ru) 1999-08-26
YU13299A (sh) 2001-03-07
US6444826B1 (en) 2002-09-03
ATE249452T1 (de) 2003-09-15
GT199700104AA (es) 1999-03-28
DE69724801D1 (de) 2003-10-16
SK31399A3 (en) 2000-05-16
MA24319A1 (fr) 1998-04-01
US20020042526A1 (en) 2002-04-11
PE109798A1 (es) 1999-01-13
UA58520C2 (uk) 2003-08-15
GT199700104BA (es) 1999-03-28
CN1230954A (zh) 1999-10-06
EP0925292A1 (en) 1999-06-30
WO1998011085A1 (en) 1998-03-19
EP0925292B1 (en) 2003-09-10
IL128732A0 (en) 2000-01-31
CA2265043A1 (en) 1998-03-19
IS4980A (is) 1999-02-16
US6096906A (en) 2000-08-01
HRP970497A2 (en) 1998-08-31
AP9701083A0 (en) 1997-10-31
GT199700104A (es) 1999-03-02
AU713701B2 (en) 1999-12-09
PL332351A1 (en) 1999-09-13
NO991254L (no) 1999-05-14
US6355825B1 (en) 2002-03-12
BG103231A (en) 1999-12-30
CN1108298C (zh) 2003-05-14
OA10995A (en) 2001-11-06
ID19613A (id) 1998-07-23
HRP970497B1 (en) 2002-06-30
US6288242B1 (en) 2001-09-11
KR20000036136A (ko) 2000-06-26
PA8437901A1 (es) 2000-05-24
KR100339164B1 (ko) 2002-06-01
HN1997000127A (es) 1997-12-20

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