AP2006003767A0 - Morpholine compounds - Google Patents

Morpholine compounds

Info

Publication number
AP2006003767A0
AP2006003767A0 AP2006003767A AP2006003767A AP2006003767A0 AP 2006003767 A0 AP2006003767 A0 AP 2006003767A0 AP 2006003767 A AP2006003767 A AP 2006003767A AP 2006003767 A AP2006003767 A AP 2006003767A AP 2006003767 A0 AP2006003767 A0 AP 2006003767A0
Authority
AP
ARIPO
Prior art keywords
morpholine compounds
morpholine
compounds
Prior art date
Application number
AP2006003767A
Other languages
English (en)
Inventor
Malcolm Christian Mackenny
Alan Stobie
Florian Wakenhut
Gavin Alistair Whitlock
Paul Vincent Fish
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32482498&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AP2006003767(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of AP2006003767A0 publication Critical patent/AP2006003767A0/xx

Links

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D265/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/281,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/301,4-Oxazines; Hydrogenated 1,4-oxazines not condensed with other rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Reproductive Health (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Psychology (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Immunology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
AP2006003767A 2004-04-30 2005-04-20 Morpholine compounds AP2006003767A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0409744.0A GB0409744D0 (en) 2004-04-30 2004-04-30 Novel compounds
PCT/IB2005/001154 WO2005105100A1 (fr) 2004-04-30 2005-04-20 Composes de morpholine

Publications (1)

Publication Number Publication Date
AP2006003767A0 true AP2006003767A0 (en) 2006-10-31

Family

ID=32482498

Family Applications (1)

Application Number Title Priority Date Filing Date
AP2006003767A AP2006003767A0 (en) 2004-04-30 2005-04-20 Morpholine compounds

Country Status (33)

Country Link
US (3) US20050250775A1 (fr)
EP (1) EP1744754A1 (fr)
JP (2) JP4181622B2 (fr)
KR (4) KR20090006888A (fr)
CN (1) CN1950089A (fr)
AP (1) AP2006003767A0 (fr)
AR (1) AR048934A1 (fr)
AU (1) AU2005237301A1 (fr)
BR (1) BRPI0510515A (fr)
CA (1) CA2564990C (fr)
CR (1) CR8717A (fr)
DO (1) DOP2005000064A (fr)
EA (1) EA200601802A1 (fr)
EC (1) ECSP066958A (fr)
GB (1) GB0409744D0 (fr)
GE (1) GEP20084549B (fr)
GT (1) GT200500098A (fr)
IL (1) IL178313A0 (fr)
MA (1) MA28554B1 (fr)
MX (1) MXPA06012640A (fr)
NI (1) NI200600257A (fr)
NL (1) NL1028927C2 (fr)
NO (1) NO20064282L (fr)
NZ (1) NZ550054A (fr)
PA (1) PA8631601A1 (fr)
PE (1) PE20060305A1 (fr)
SV (1) SV2005002099A (fr)
TN (1) TNSN06347A1 (fr)
TW (2) TW200914431A (fr)
UA (1) UA86970C2 (fr)
UY (1) UY28873A1 (fr)
WO (1) WO2005105100A1 (fr)
ZA (1) ZA200608661B (fr)

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BRPI0510453A (pt) * 2004-04-30 2007-10-30 Warner Lambert Co composto substituìdos com morfolina para o tratamento de distúrbios do sistema nervoso central
GB0409744D0 (en) * 2004-04-30 2004-06-09 Pfizer Ltd Novel compounds
JP2009516705A (ja) * 2005-11-18 2009-04-23 アストラゼネカ・アクチエボラーグ 塩の形態
US8389510B2 (en) * 2005-11-18 2013-03-05 Astrazeneca Ab Crystalline forms
WO2007062339A2 (fr) * 2005-11-18 2007-05-31 Astrazeneca Ab Formulations liquides
US20090215744A1 (en) * 2005-11-18 2009-08-27 Astrazeneca Ab Solid Formulations
CN101360502B (zh) * 2005-11-18 2012-03-14 阿斯利康公司 结晶形式
US8030332B2 (en) * 2006-02-01 2011-10-04 Merck Sharp & Dohme Corp. Potassium channel inhibitors
EP1892530A1 (fr) * 2006-08-25 2008-02-27 Boehringer Ingelheim Pharma GmbH & Co. KG Procédé de détermination de l'activité de transport d'une protéine de transport
KR101103118B1 (ko) * 2007-11-02 2012-01-04 동아제약주식회사 신규한 1,3-디히드로-5-이소벤조퓨란카르보니트릴 유도체 화합물 및 이를 함유하는 조루증 치료용 약학조성물
JP5405571B2 (ja) * 2008-07-24 2014-02-05 セラヴァンス, インコーポレーテッド 3−(フェノキシフェニルメチル)ピロリジン化合物
US8637577B2 (en) 2009-01-22 2014-01-28 Absorption Pharmaceuticals, LLC Desensitizing drug product
WO2010120910A1 (fr) * 2009-04-15 2010-10-21 Theravance, Inc. Composés 3-(phénoxypyrrolidin-3-yl-méthyle) hétéroaryle, 3-(phénylpyrrolidin-3-ylméthoxy) hétéroaryle, et 3-(hétéroarylpyrrolidin-3-ylméthoxy) hétéroaryle
CN102471258A (zh) * 2009-07-13 2012-05-23 施万制药 3-苯氧基甲基吡咯烷化合物
ES2495366T3 (es) 2009-07-21 2014-09-17 Theravance, Inc. Compuestos de 3-fenoximetilpirrolidina
AR077969A1 (es) 2009-08-31 2011-10-05 Abbott Healthcare Products Bv Derivados de (tio)morfolina comomoduladores de s1p
TW201206893A (en) 2010-07-09 2012-02-16 Abbott Healthcare Products Bv Bisaryl (thio) morpholine derivatives as S1P modulators
TWI522361B (zh) 2010-07-09 2016-02-21 艾伯維公司 作為s1p調節劑的稠合雜環衍生物
TWI543984B (zh) 2010-07-09 2016-08-01 艾伯維公司 作為s1p調節劑的螺-哌啶衍生物
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