ZA878128B - Benzo(5,6)cycloheptapyridines,compositions and methods of use - Google Patents

Benzo(5,6)cycloheptapyridines,compositions and methods of use

Info

Publication number
ZA878128B
ZA878128B ZA878128A ZA878128A ZA878128B ZA 878128 B ZA878128 B ZA 878128B ZA 878128 A ZA878128 A ZA 878128A ZA 878128 A ZA878128 A ZA 878128A ZA 878128 B ZA878128 B ZA 878128B
Authority
ZA
South Africa
Prior art keywords
benzo
methods
cycloheptapyridines
compositions
cyclohepta
Prior art date
Application number
ZA878128A
Other languages
English (en)
Inventor
J. Piwinski John
K. Ganguly Ashit
J. Green Michael
J. Villani Frank
Wong Jesse
Original Assignee
Schering Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corporation filed Critical Schering Corporation
Publication of ZA878128B publication Critical patent/ZA878128B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/16—Ring systems of three rings containing carbocyclic rings other than six-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Cosmetics (AREA)
  • Hydrogenated Pyridines (AREA)
ZA878128A 1986-10-31 1987-10-29 Benzo(5,6)cycloheptapyridines,compositions and methods of use ZA878128B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/925,342 US4826853A (en) 1986-10-31 1986-10-31 6,11-Dihydro-11-(N-substituted-4-piperidylidene)-5H-benzo(5,6)cyclohepta(1,2-B)pyridines and compositions and methods of use

Publications (1)

Publication Number Publication Date
ZA878128B true ZA878128B (en) 1988-04-29

Family

ID=25451584

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA878128A ZA878128B (en) 1986-10-31 1987-10-29 Benzo(5,6)cycloheptapyridines,compositions and methods of use

Country Status (22)

Country Link
US (1) US4826853A (sv)
EP (3) EP0685476A1 (sv)
JP (1) JPH0678316B2 (sv)
KR (1) KR930002489B1 (sv)
AT (1) ATE116310T1 (sv)
AU (1) AU604285B2 (sv)
CA (2) CA1305147C (sv)
CS (1) CS414391A3 (sv)
DE (1) DE3750929T2 (sv)
DK (1) DK73193D0 (sv)
ES (1) ES2068179T3 (sv)
FI (1) FI96768C (sv)
HK (1) HK186396A (sv)
IE (1) IE65174B1 (sv)
IL (1) IL84310A0 (sv)
MY (1) MY102986A (sv)
NZ (1) NZ222347A (sv)
OA (1) OA09546A (sv)
PH (1) PH26184A (sv)
SG (1) SG44597A1 (sv)
WO (1) WO1988003138A1 (sv)
ZA (1) ZA878128B (sv)

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CN110818684B (zh) * 2019-10-08 2023-04-07 深圳市南山区人民医院 一种抗金黄色葡萄球菌毒力和生物被膜形成的抑制剂Lo-SH及其用途
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CN115385892A (zh) * 2021-10-28 2022-11-25 天津市昕晨投资发展有限公司 地氯雷他定衍生物、其制备方法及其用途
CN115141229B (zh) * 2022-07-21 2023-12-12 华创合成制药股份有限公司 抗组胺类化合物及其制备方法和用途

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US4804666A (en) * 1985-08-14 1989-02-14 Schering Corporation Antiallergic 6,11-dihydro-11-(4-piperidylidene)-5H-benzo(5,6)cyclohepta(1,2-B)pyridines

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DK73193A (da) 1993-06-21
US4826853A (en) 1989-05-02
CA1321589C (en) 1993-08-24
CA1305147C (en) 1992-07-14
HK186396A (en) 1996-10-11
IE65174B1 (en) 1995-10-04
DE3750929T2 (de) 1995-06-01
WO1988003138A1 (en) 1988-05-05
AU8336287A (en) 1988-05-25
CS414391A3 (en) 1992-09-16
SG44597A1 (en) 1997-12-19
FI96768C (sv) 1996-08-26
EP0270818A1 (en) 1988-06-15
JPH0678316B2 (ja) 1994-10-05
DE3750929D1 (de) 1995-02-09
DK73193D0 (da) 1993-06-21
IL84310A0 (en) 1988-03-31
KR930002489B1 (ko) 1993-04-02
PH26184A (en) 1992-03-18
ES2068179T3 (es) 1995-04-16
ATE116310T1 (de) 1995-01-15
IE872913L (en) 1988-04-30
KR880701716A (ko) 1988-11-04
JPH02500910A (ja) 1990-03-29
OA09546A (en) 1993-01-31
FI891806A0 (sv) 1989-04-17
EP0270818B1 (en) 1994-12-28
FI96768B (sv) 1996-05-15
NZ222347A (en) 1990-03-27
FI891806A (sv) 1989-04-17
EP0685476A1 (en) 1995-12-06
EP0330673A1 (en) 1989-09-06
AU604285B2 (en) 1990-12-13
MY102986A (en) 1993-03-31

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