CS414391A3 - Benzo(5,6)cycloheptapyridines, preparations and methods of use - Google Patents

Benzo(5,6)cycloheptapyridines, preparations and methods of use Download PDF

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Publication number
CS414391A3
CS414391A3 CS914143A CS414391A CS414391A3 CS 414391 A3 CS414391 A3 CS 414391A3 CS 914143 A CS914143 A CS 914143A CS 414391 A CS414391 A CS 414391A CS 414391 A3 CS414391 A3 CS 414391A3
Authority
CS
Czechoslovakia
Prior art keywords
benzo
pyridine
cyclohepta
dihydro
formula
Prior art date
Application number
CS914143A
Other languages
Czech (cs)
English (en)
Inventor
John J Piwinski
Ashit K Ganguly
Frank J Villani
Jesse Wong
Michael J Green
Charles A Magatti
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of CS414391A3 publication Critical patent/CS414391A3/cs

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/16—Ring systems of three rings containing carbocyclic rings other than six-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Cosmetics (AREA)
CS914143A 1986-10-31 1991-12-30 Benzo(5,6)cycloheptapyridines, preparations and methods of use CS414391A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/925,342 US4826853A (en) 1986-10-31 1986-10-31 6,11-Dihydro-11-(N-substituted-4-piperidylidene)-5H-benzo(5,6)cyclohepta(1,2-B)pyridines and compositions and methods of use

Publications (1)

Publication Number Publication Date
CS414391A3 true CS414391A3 (en) 1992-09-16

Family

ID=25451584

Family Applications (1)

Application Number Title Priority Date Filing Date
CS914143A CS414391A3 (en) 1986-10-31 1991-12-30 Benzo(5,6)cycloheptapyridines, preparations and methods of use

Country Status (22)

Country Link
US (1) US4826853A (sv)
EP (3) EP0270818B1 (sv)
JP (1) JPH0678316B2 (sv)
KR (1) KR930002489B1 (sv)
AT (1) ATE116310T1 (sv)
AU (1) AU604285B2 (sv)
CA (2) CA1305147C (sv)
CS (1) CS414391A3 (sv)
DE (1) DE3750929T2 (sv)
DK (1) DK73193A (sv)
ES (1) ES2068179T3 (sv)
FI (1) FI96768C (sv)
HK (1) HK186396A (sv)
IE (1) IE65174B1 (sv)
IL (1) IL84310A0 (sv)
MY (1) MY102986A (sv)
NZ (1) NZ222347A (sv)
OA (1) OA09546A (sv)
PH (1) PH26184A (sv)
SG (1) SG44597A1 (sv)
WO (1) WO1988003138A1 (sv)
ZA (1) ZA878128B (sv)

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FI96768B (sv) 1996-05-15
IL84310A0 (en) 1988-03-31
FI891806A0 (sv) 1989-04-17
DE3750929D1 (de) 1995-02-09
JPH0678316B2 (ja) 1994-10-05
PH26184A (en) 1992-03-18
MY102986A (en) 1993-03-31
EP0330673A1 (en) 1989-09-06
EP0270818A1 (en) 1988-06-15
DE3750929T2 (de) 1995-06-01
ES2068179T3 (es) 1995-04-16
SG44597A1 (en) 1997-12-19
EP0270818B1 (en) 1994-12-28
DK73193D0 (da) 1993-06-21
AU604285B2 (en) 1990-12-13
KR880701716A (ko) 1988-11-04
EP0685476A1 (en) 1995-12-06
US4826853A (en) 1989-05-02
IE872913L (en) 1988-04-30
ATE116310T1 (de) 1995-01-15
FI96768C (sv) 1996-08-26
CA1321589C (en) 1993-08-24
IE65174B1 (en) 1995-10-04
KR930002489B1 (ko) 1993-04-02
NZ222347A (en) 1990-03-27
OA09546A (en) 1993-01-31
AU8336287A (en) 1988-05-25
JPH02500910A (ja) 1990-03-29
HK186396A (en) 1996-10-11
DK73193A (da) 1993-06-21
CA1305147C (en) 1992-07-14
WO1988003138A1 (en) 1988-05-05
FI891806A (sv) 1989-04-17
ZA878128B (en) 1988-04-29

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