FI891806A0 - Förfarande för framställning av farmakologiskt värdefullt benso/5,6/cykloheptapyridin - Google Patents

Förfarande för framställning av farmakologiskt värdefullt benso/5,6/cykloheptapyridin

Info

Publication number
FI891806A0
FI891806A0 FI891806A FI891806A FI891806A0 FI 891806 A0 FI891806 A0 FI 891806A0 FI 891806 A FI891806 A FI 891806A FI 891806 A FI891806 A FI 891806A FI 891806 A0 FI891806 A0 FI 891806A0
Authority
FI
Finland
Prior art keywords
benzo
cycloheptapyridine
method produces
pharmacologically valuable
produces pharmacologically
Prior art date
Application number
FI891806A
Other languages
English (en)
Finnish (fi)
Other versions
FI96768C (sv
FI96768B (sv
FI891806A (sv
Inventor
John J Piwinski
Ashit K Ganguly
Michael J Green
Frank J Villani
Jesse Wong
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of FI891806A0 publication Critical patent/FI891806A0/sv
Publication of FI891806A publication Critical patent/FI891806A/sv
Application granted granted Critical
Publication of FI96768B publication Critical patent/FI96768B/sv
Publication of FI96768C publication Critical patent/FI96768C/sv

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/04—Ortho- or peri-condensed ring systems
    • C07D221/06—Ring systems of three rings
    • C07D221/16—Ring systems of three rings containing carbocyclic rings other than six-membered
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Cosmetics (AREA)
FI891806A 1986-10-31 1989-04-17 Förfarande för framställning av farmakologiskt värdefullt benso/5,6/cykloheptapyridin FI96768C (sv)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US06/925,342 US4826853A (en) 1986-10-31 1986-10-31 6,11-Dihydro-11-(N-substituted-4-piperidylidene)-5H-benzo(5,6)cyclohepta(1,2-B)pyridines and compositions and methods of use
US92534286 1986-10-31
PCT/US1987/002777 WO1988003138A1 (en) 1986-10-31 1987-10-29 Benzo[5,6]cycloheptapyridines, compositions and methods of use
US8702777 1987-10-29

Publications (4)

Publication Number Publication Date
FI891806A0 true FI891806A0 (sv) 1989-04-17
FI891806A FI891806A (sv) 1989-04-17
FI96768B FI96768B (sv) 1996-05-15
FI96768C FI96768C (sv) 1996-08-26

Family

ID=25451584

Family Applications (1)

Application Number Title Priority Date Filing Date
FI891806A FI96768C (sv) 1986-10-31 1989-04-17 Förfarande för framställning av farmakologiskt värdefullt benso/5,6/cykloheptapyridin

Country Status (22)

Country Link
US (1) US4826853A (sv)
EP (3) EP0270818B1 (sv)
JP (1) JPH0678316B2 (sv)
KR (1) KR930002489B1 (sv)
AT (1) ATE116310T1 (sv)
AU (1) AU604285B2 (sv)
CA (2) CA1305147C (sv)
CS (1) CS414391A3 (sv)
DE (1) DE3750929T2 (sv)
DK (1) DK73193D0 (sv)
ES (1) ES2068179T3 (sv)
FI (1) FI96768C (sv)
HK (1) HK186396A (sv)
IE (1) IE65174B1 (sv)
IL (1) IL84310A0 (sv)
MY (1) MY102986A (sv)
NZ (1) NZ222347A (sv)
OA (1) OA09546A (sv)
PH (1) PH26184A (sv)
SG (1) SG44597A1 (sv)
WO (1) WO1988003138A1 (sv)
ZA (1) ZA878128B (sv)

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CN110818685A (zh) * 2019-10-08 2020-02-21 深圳市南山区人民医院 一种抗金黄色葡萄球菌毒力和生物被膜形成的抑制剂Lo-异己基及其用途
CN110845473B (zh) * 2019-10-08 2023-04-07 深圳市南山区人民医院 一种抗金黄色葡萄球菌毒力和生物被膜形成的抑制剂Lo-乙酸乙酯及其用途
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CN115385892A (zh) * 2021-10-28 2022-11-25 天津市昕晨投资发展有限公司 地氯雷他定衍生物、其制备方法及其用途
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EP0330673A1 (en) 1989-09-06
IE872913L (en) 1988-04-30
IL84310A0 (en) 1988-03-31
CA1305147C (en) 1992-07-14
IE65174B1 (en) 1995-10-04
JPH02500910A (ja) 1990-03-29
SG44597A1 (en) 1997-12-19
ES2068179T3 (es) 1995-04-16
AU604285B2 (en) 1990-12-13
CA1321589C (en) 1993-08-24
NZ222347A (en) 1990-03-27
ATE116310T1 (de) 1995-01-15
EP0270818A1 (en) 1988-06-15
DK73193A (da) 1993-06-21
JPH0678316B2 (ja) 1994-10-05
MY102986A (en) 1993-03-31
FI96768C (sv) 1996-08-26
CS414391A3 (en) 1992-09-16
WO1988003138A1 (en) 1988-05-05
FI96768B (sv) 1996-05-15
EP0270818B1 (en) 1994-12-28
PH26184A (en) 1992-03-18
EP0685476A1 (en) 1995-12-06
ZA878128B (en) 1988-04-29
AU8336287A (en) 1988-05-25
OA09546A (en) 1993-01-31
DE3750929T2 (de) 1995-06-01
FI891806A (sv) 1989-04-17
HK186396A (en) 1996-10-11
US4826853A (en) 1989-05-02
KR880701716A (ko) 1988-11-04
DK73193D0 (da) 1993-06-21
KR930002489B1 (ko) 1993-04-02
DE3750929D1 (de) 1995-02-09

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