ZA82566B - Aromatic heterocyclic esters of steroids,their preparation and pharmaceutical compositions containing them - Google Patents

Aromatic heterocyclic esters of steroids,their preparation and pharmaceutical compositions containing them

Info

Publication number
ZA82566B
ZA82566B ZA82566A ZA82566A ZA82566B ZA 82566 B ZA82566 B ZA 82566B ZA 82566 A ZA82566 A ZA 82566A ZA 82566 A ZA82566 A ZA 82566A ZA 82566 B ZA82566 B ZA 82566B
Authority
ZA
South Africa
Prior art keywords
aromatic heterocyclic
steroids
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
ZA82566A
Other languages
English (en)
Inventor
Elliot L Shapiro
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of ZA82566B publication Critical patent/ZA82566B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J33/00Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/002Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J17/00Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J43/00Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyridine Compounds (AREA)
ZA82566A 1981-02-02 1982-01-28 Aromatic heterocyclic esters of steroids,their preparation and pharmaceutical compositions containing them ZA82566B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23076381A 1981-02-02 1981-02-02

Publications (1)

Publication Number Publication Date
ZA82566B true ZA82566B (en) 1982-12-29

Family

ID=22866476

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA82566A ZA82566B (en) 1981-02-02 1982-01-28 Aromatic heterocyclic esters of steroids,their preparation and pharmaceutical compositions containing them

Country Status (25)

Country Link
US (1) US4472393A (fr)
EP (1) EP0057401B1 (fr)
JP (1) JPS57146800A (fr)
KR (1) KR890000761B1 (fr)
AT (1) ATE8790T1 (fr)
AU (1) AU549102B2 (fr)
BG (1) BG60799B2 (fr)
CA (1) CA1177822A (fr)
CY (1) CY1359A (fr)
DE (1) DE3260474D1 (fr)
DK (1) DK162770C (fr)
FI (1) FI78111C (fr)
HK (1) HK68487A (fr)
HU (1) HU188769B (fr)
IE (1) IE52576B1 (fr)
IL (1) IL64885A (fr)
KE (1) KE3694A (fr)
MX (1) MX9203403A (fr)
NL (1) NL930095I2 (fr)
NO (2) NO157020C (fr)
NZ (1) NZ199600A (fr)
OA (1) OA07116A (fr)
PH (1) PH19733A (fr)
PT (1) PT74357B (fr)
ZA (1) ZA82566B (fr)

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US4221787A (en) * 1978-03-28 1980-09-09 Interx Research Corporation Esteramide prodrugs of anti-inflammatory corticosteroids

Also Published As

Publication number Publication date
IE820207L (en) 1982-08-02
NL930095I2 (nl) 1994-12-01
NO157020B (no) 1987-09-28
PT74357A (en) 1982-02-01
JPS57146800A (en) 1982-09-10
HK68487A (en) 1987-10-02
ATE8790T1 (de) 1984-08-15
DE3260474D1 (en) 1984-09-06
HU188769B (en) 1986-05-28
NO820263L (no) 1982-08-03
CA1177822A (fr) 1984-11-13
PT74357B (en) 1984-05-30
EP0057401B1 (fr) 1984-08-01
DK162770B (da) 1991-12-09
EP0057401A1 (fr) 1982-08-11
IL64885A (en) 1985-05-31
AU549102B2 (en) 1986-01-16
NL930095I1 (nl) 1993-10-01
NO1994018I1 (no) 1994-10-07
BG60799B2 (bg) 1996-03-29
KR890000761B1 (ko) 1989-04-05
FI78111C (fi) 1989-06-12
OA07116A (fr) 1984-03-31
CY1359A (en) 1987-08-07
PH19733A (en) 1986-06-17
FI820280L (fi) 1982-08-03
AU7991882A (en) 1982-08-12
NO157020C (no) 1988-01-06
MX9203403A (es) 1992-07-01
FI78111B (fi) 1989-02-28
US4472393A (en) 1984-09-18
KR830009138A (ko) 1983-12-17
DK162770C (da) 1992-04-27
KE3694A (en) 1987-03-13
NZ199600A (en) 1984-09-28
IE52576B1 (en) 1987-12-23
JPS6360036B2 (fr) 1988-11-22
DK39082A (da) 1982-08-03
IL64885A0 (en) 1982-03-31

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