KE3694A - Aromatic heterocyclic esters of steroids,their preparation and pharmaceutical compositions containing them - Google Patents

Aromatic heterocyclic esters of steroids,their preparation and pharmaceutical compositions containing them

Info

Publication number
KE3694A
KE3694A KE3694A KE369487A KE3694A KE 3694 A KE3694 A KE 3694A KE 3694 A KE3694 A KE 3694A KE 369487 A KE369487 A KE 369487A KE 3694 A KE3694 A KE 3694A
Authority
KE
Kenya
Prior art keywords
aromatic heterocyclic
steroids
preparation
pharmaceutical compositions
compositions containing
Prior art date
Application number
KE3694A
Other languages
English (en)
Inventor
Elliot L Shapiro
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of KE3694A publication Critical patent/KE3694A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyridine Compounds (AREA)
KE3694A 1981-02-02 1987-02-19 Aromatic heterocyclic esters of steroids,their preparation and pharmaceutical compositions containing them KE3694A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23076381A 1981-02-02 1981-02-02
EP82100490A EP0057401B1 (fr) 1981-02-02 1982-01-25 Esters aromatiques hétérocycliques de stéroides, leur préparation et compositions pharmaceutiques les contenant

Publications (1)

Publication Number Publication Date
KE3694A true KE3694A (en) 1987-03-13

Family

ID=22866476

Family Applications (1)

Application Number Title Priority Date Filing Date
KE3694A KE3694A (en) 1981-02-02 1987-02-19 Aromatic heterocyclic esters of steroids,their preparation and pharmaceutical compositions containing them

Country Status (25)

Country Link
US (1) US4472393A (fr)
EP (1) EP0057401B1 (fr)
JP (1) JPS57146800A (fr)
KR (1) KR890000761B1 (fr)
AT (1) ATE8790T1 (fr)
AU (1) AU549102B2 (fr)
BG (1) BG60799B2 (fr)
CA (1) CA1177822A (fr)
CY (1) CY1359A (fr)
DE (1) DE3260474D1 (fr)
DK (1) DK162770C (fr)
FI (1) FI78111C (fr)
HK (1) HK68487A (fr)
HU (1) HU188769B (fr)
IE (1) IE52576B1 (fr)
IL (1) IL64885A (fr)
KE (1) KE3694A (fr)
MX (1) MX9203403A (fr)
NL (1) NL930095I2 (fr)
NO (2) NO157020C (fr)
NZ (1) NZ199600A (fr)
OA (1) OA07116A (fr)
PH (1) PH19733A (fr)
PT (1) PT74357B (fr)
ZA (1) ZA82566B (fr)

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US4221787A (en) * 1978-03-28 1980-09-09 Interx Research Corporation Esteramide prodrugs of anti-inflammatory corticosteroids

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AU549102B2 (en) 1986-01-16
NZ199600A (en) 1984-09-28
NO157020C (no) 1988-01-06
OA07116A (fr) 1984-03-31
NO157020B (no) 1987-09-28
EP0057401A1 (fr) 1982-08-11
KR890000761B1 (ko) 1989-04-05
NL930095I2 (nl) 1994-12-01
NO1994018I1 (no) 1994-10-07
PT74357B (en) 1984-05-30
IE52576B1 (en) 1987-12-23
CA1177822A (fr) 1984-11-13
FI820280L (fi) 1982-08-03
ZA82566B (en) 1982-12-29
JPS6360036B2 (fr) 1988-11-22
FI78111B (fi) 1989-02-28
IL64885A0 (en) 1982-03-31
IL64885A (en) 1985-05-31
JPS57146800A (en) 1982-09-10
MX9203403A (es) 1992-07-01
DE3260474D1 (en) 1984-09-06
AU7991882A (en) 1982-08-12
DK39082A (da) 1982-08-03
PH19733A (en) 1986-06-17
PT74357A (en) 1982-02-01
US4472393A (en) 1984-09-18
DK162770C (da) 1992-04-27
ATE8790T1 (de) 1984-08-15
CY1359A (en) 1987-08-07
DK162770B (da) 1991-12-09
NO820263L (no) 1982-08-03
FI78111C (fi) 1989-06-12
IE820207L (en) 1982-08-02
HU188769B (en) 1986-05-28
KR830009138A (ko) 1983-12-17
HK68487A (en) 1987-10-02
NL930095I1 (nl) 1993-10-01
EP0057401B1 (fr) 1984-08-01
BG60799B2 (bg) 1996-03-29

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