NO820263L - Fremgangsmaate ved fremstilling av heterocycliske estere av steroider - Google Patents

Fremgangsmaate ved fremstilling av heterocycliske estere av steroider

Info

Publication number
NO820263L
NO820263L NO820263A NO820263A NO820263L NO 820263 L NO820263 L NO 820263L NO 820263 A NO820263 A NO 820263A NO 820263 A NO820263 A NO 820263A NO 820263 L NO820263 L NO 820263L
Authority
NO
Norway
Prior art keywords
steroids
procedure
preparation
heterocyclic esters
heterocyclic
Prior art date
Application number
NO820263A
Other languages
English (en)
Other versions
NO157020B (no
NO157020C (no
Inventor
Elliot L Shapiro
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Corp filed Critical Schering Corp
Publication of NO820263L publication Critical patent/NO820263L/no
Publication of NO157020B publication Critical patent/NO157020B/no
Publication of NO157020C publication Critical patent/NO157020C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J43/00—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J43/003—Normal steroids having a nitrogen-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pyridine Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
NO820263A 1981-02-02 1982-01-28 AnalogifremgangsmŸte ved fremstilling av terapeutisk aktive 3,20-dioxo-1,4-pregnadien-17alfa-ol-17-aromatiske heterocykliske carboxylater. NO157020C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23076381A 1981-02-02 1981-02-02

Publications (3)

Publication Number Publication Date
NO820263L true NO820263L (no) 1982-08-03
NO157020B NO157020B (no) 1987-09-28
NO157020C NO157020C (no) 1988-01-06

Family

ID=22866476

Family Applications (2)

Application Number Title Priority Date Filing Date
NO820263A NO157020C (no) 1981-02-02 1982-01-28 AnalogifremgangsmŸte ved fremstilling av terapeutisk aktive 3,20-dioxo-1,4-pregnadien-17alfa-ol-17-aromatiske heterocykliske carboxylater.
NO1994018C NO1994018I1 (no) 1981-02-02 1994-10-07 Mometasonfuroat

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO1994018C NO1994018I1 (no) 1981-02-02 1994-10-07 Mometasonfuroat

Country Status (25)

Country Link
US (1) US4472393A (no)
EP (1) EP0057401B1 (no)
JP (1) JPS57146800A (no)
KR (1) KR890000761B1 (no)
AT (1) ATE8790T1 (no)
AU (1) AU549102B2 (no)
BG (1) BG60799B2 (no)
CA (1) CA1177822A (no)
CY (1) CY1359A (no)
DE (1) DE3260474D1 (no)
DK (1) DK162770C (no)
FI (1) FI78111C (no)
HK (1) HK68487A (no)
HU (1) HU188769B (no)
IE (1) IE52576B1 (no)
IL (1) IL64885A (no)
KE (1) KE3694A (no)
MX (1) MX9203403A (no)
NL (1) NL930095I2 (no)
NO (2) NO157020C (no)
NZ (1) NZ199600A (no)
OA (1) OA07116A (no)
PH (1) PH19733A (no)
PT (1) PT74357B (no)
ZA (1) ZA82566B (no)

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GB1253831A (en) * 1968-01-19 1971-11-17 Glaxo Lab Ltd 9alpha,21-DIHALOPREGNANE COMPOUNDS
US3980778A (en) * 1973-10-25 1976-09-14 The Upjohn Company Anti-inflammatory steroid
NL7502252A (nl) * 1974-02-27 1975-08-29 Pierrel Spa Werkwijze voor het bereiden van een geneesmid- del met anti-inflammatoire werking, gevormd ge- neesmiddel verkregen volgens deze werkwijze alsmede werkwijze voor het bereiden van in het geneesmiddel gebruikte nieuwe steroiden.
GB1505701A (en) * 1975-06-14 1978-03-30 Pierrel Spa 2-chloro-6beta-fluoropregnanes
US4221787A (en) * 1978-03-28 1980-09-09 Interx Research Corporation Esteramide prodrugs of anti-inflammatory corticosteroids

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MX9203403A (es) 1992-07-01
JPS57146800A (en) 1982-09-10
DK39082A (da) 1982-08-03
PT74357B (en) 1984-05-30
DK162770B (da) 1991-12-09
HK68487A (en) 1987-10-02
IE52576B1 (en) 1987-12-23
PH19733A (en) 1986-06-17
CA1177822A (en) 1984-11-13
JPS6360036B2 (no) 1988-11-22
IL64885A0 (en) 1982-03-31
HU188769B (en) 1986-05-28
EP0057401B1 (en) 1984-08-01
NO157020B (no) 1987-09-28
PT74357A (en) 1982-02-01
DE3260474D1 (en) 1984-09-06
AU549102B2 (en) 1986-01-16
NZ199600A (en) 1984-09-28
OA07116A (fr) 1984-03-31
FI78111C (fi) 1989-06-12
KE3694A (en) 1987-03-13
IL64885A (en) 1985-05-31
KR890000761B1 (ko) 1989-04-05
NO1994018I1 (no) 1994-10-07
DK162770C (da) 1992-04-27
BG60799B2 (bg) 1996-03-29
IE820207L (en) 1982-08-02
ATE8790T1 (de) 1984-08-15
FI820280L (fi) 1982-08-03
US4472393A (en) 1984-09-18
NL930095I1 (nl) 1993-10-01
CY1359A (en) 1987-08-07
KR830009138A (ko) 1983-12-17
NO157020C (no) 1988-01-06
NL930095I2 (nl) 1994-12-01
ZA82566B (en) 1982-12-29
EP0057401A1 (en) 1982-08-11
AU7991882A (en) 1982-08-12
FI78111B (fi) 1989-02-28

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