ZA775361B - Uracil derivatives and process for the preparation thereof - Google Patents

Uracil derivatives and process for the preparation thereof

Info

Publication number
ZA775361B
ZA775361B ZA00775361A ZA775361A ZA775361B ZA 775361 B ZA775361 B ZA 775361B ZA 00775361 A ZA00775361 A ZA 00775361A ZA 775361 A ZA775361 A ZA 775361A ZA 775361 B ZA775361 B ZA 775361B
Authority
ZA
South Africa
Prior art keywords
preparation
uracil derivatives
uracil
derivatives
Prior art date
Application number
ZA00775361A
Other languages
English (en)
Inventor
Y Ike
H Tamura
S Ozaki
K Ishikawa
Original Assignee
Mitsui Toatsu Chemicals
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mitsui Toatsu Chemicals filed Critical Mitsui Toatsu Chemicals
Publication of ZA775361B publication Critical patent/ZA775361B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
    • C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/553—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms with halogen atoms or nitro radicals directly attached to ring carbon atoms, e.g. fluorouracil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ZA00775361A 1976-09-06 1977-09-06 Uracil derivatives and process for the preparation thereof ZA775361B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP10571476A JPS5331676A (en) 1976-09-06 1976-09-06 Uracil derivatives and their preparation

Publications (1)

Publication Number Publication Date
ZA775361B true ZA775361B (en) 1978-07-26

Family

ID=14414993

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA00775361A ZA775361B (en) 1976-09-06 1977-09-06 Uracil derivatives and process for the preparation thereof

Country Status (16)

Country Link
US (1) US4267326A (fr)
JP (1) JPS5331676A (fr)
AU (1) AU513153B2 (fr)
CH (1) CH634567A5 (fr)
DE (1) DE2739912A1 (fr)
DK (1) DK142413B (fr)
FI (1) FI62071C (fr)
FR (1) FR2363563A1 (fr)
GB (1) GB1543467A (fr)
HU (1) HU177482B (fr)
NL (1) NL7709808A (fr)
PH (1) PH14000A (fr)
PL (1) PL108914B1 (fr)
SE (1) SE438856B (fr)
SU (1) SU795468A3 (fr)
ZA (1) ZA775361B (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5379879A (en) * 1976-12-23 1978-07-14 Mitsui Toatsu Chem Inc 1,3-substituted-5-fluorouracils and process for their preparation
JPS54122281A (en) * 1978-03-13 1979-09-21 Mitsui Toatsu Chem Inc 5-fluorouracil derivative and its preparation
JPS5668674A (en) * 1979-11-08 1981-06-09 Shionogi & Co Ltd 5-fluorouracil derivative
JPS5724369A (en) * 1980-07-19 1982-02-08 Tokyo Kinzoku Kogyo Kk Pyrimidine derivative and its preparation
JPS5738774A (en) * 1980-08-19 1982-03-03 Chugai Pharmaceut Co Ltd Uracil derivative and its preparation
DE3480706D1 (de) * 1983-10-20 1990-01-18 Terumo Corp 5-fluoruracilabkoemmlinge sowie medizinische zusammensetzungen die diese enthalten.
DK197486A (da) * 1986-04-30 1987-10-31 Ferring Farma Lab 5-fluoruracilprodug
US6051576A (en) * 1994-01-28 2000-04-18 University Of Kentucky Research Foundation Means to achieve sustained release of synergistic drugs by conjugation
SI2445502T1 (sl) 2009-06-25 2017-10-30 Alkermes Pharma Ireland Limited Heterociklične spojine za zdravljenje neuroloških in psiholoških motenj
EP2445343B1 (fr) 2009-06-25 2021-08-04 Alkermes Pharma Ireland Limited Promédicaments de composés nh acides
EP2897592B1 (fr) 2012-09-19 2020-02-19 Alkermes Pharma Ireland Limited Compositions pharmaceutiques ayant une plus grande stabilité au stockage
RU2688233C2 (ru) 2014-03-20 2019-05-21 Алкермес Фарма Айэленд Лимитед Препараты арипипразола, имеющие повышенные скорости впрыска
CN112423754A (zh) 2018-03-05 2021-02-26 奥克梅斯制药爱尔兰有限公司 阿立哌唑的给药策略
CN109761915B (zh) * 2019-03-05 2021-12-21 沈阳药科大学 靶向mct1转运体的5-氟尿嘧啶成酯前药

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5324952B2 (fr) * 1973-11-28 1978-07-24
JPS603071B2 (ja) * 1975-02-17 1985-01-25 三井製薬工業株式会社 １−（α−アシロキシアルキル）−５−フルオロウラシル類の製造方法

Also Published As

Publication number Publication date
NL7709808A (nl) 1978-03-08
FR2363563B1 (fr) 1980-06-20
JPS5331676A (en) 1978-03-25
DK394477A (fr) 1978-03-07
PL200685A1 (pl) 1978-10-09
CH634567A5 (de) 1983-02-15
FI772594A (fi) 1978-03-07
JPS6114148B2 (fr) 1986-04-17
AU2857177A (en) 1979-03-15
US4267326A (en) 1981-05-12
AU513153B2 (en) 1980-11-20
DK142413C (fr) 1981-03-23
FI62071B (fi) 1982-07-30
PL108914B1 (en) 1980-05-31
FI62071C (fi) 1982-11-10
PH14000A (en) 1980-11-28
DE2739912A1 (de) 1978-03-09
FR2363563A1 (fr) 1978-03-31
SE438856B (sv) 1985-05-13
DK142413B (da) 1980-10-27
GB1543467A (en) 1979-04-04
SE7709942L (sv) 1978-03-07
SU795468A3 (ru) 1981-01-07
HU177482B (en) 1981-10-28

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