ZA200610357B - Indoles useful in the treatment of inflammation - Google Patents
Indoles useful in the treatment of inflammation Download PDFInfo
- Publication number
- ZA200610357B ZA200610357B ZA200610357A ZA200610357A ZA200610357B ZA 200610357 B ZA200610357 B ZA 200610357B ZA 200610357 A ZA200610357 A ZA 200610357A ZA 200610357 A ZA200610357 A ZA 200610357A ZA 200610357 B ZA200610357 B ZA 200610357B
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- ZA
- South Africa
- Prior art keywords
- compound
- optionally substituted
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- alkyl
- halo
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- 125000001791 phenazinyl group Chemical group C1(=CC=CC2=NC3=CC=CC=C3N=C12)* 0.000 description 1
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- 238000003419 tautomerization reaction Methods 0.000 description 1
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Classifications
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| CN102186845B (zh) | 2008-10-17 | 2016-09-07 | 阿卡制药有限公司 | S1p受体调节剂以及它们的用途 |
| EP2344446A4 (en) | 2008-10-17 | 2012-04-04 | Akaal Pharma Pty Ltd | S1P RECEPTOR MODULATORS |
| US20120029016A1 (en) | 2008-12-30 | 2012-02-02 | Biolipox Ab | Indoles Useful in the Treatment of Inflammation |
| WO2010127152A2 (en) * | 2009-04-29 | 2010-11-04 | Irm Llc | Compounds and compositions as microsomal prostaglandin e synthase-1 inhibitors |
| US8889730B2 (en) | 2012-04-10 | 2014-11-18 | Pfizer Inc. | Indole and indazole compounds that activate AMPK |
| CA2905242C (en) | 2013-03-15 | 2016-11-29 | Pfizer Inc. | Indole compounds that activate ampk |
| CN108929203A (zh) * | 2018-08-14 | 2018-12-04 | 重庆市化工研究院 | 一种芳香族乙烯基醚及其合成方法和应用 |
| WO2021040393A1 (ko) * | 2019-08-26 | 2021-03-04 | 국제약품 주식회사 | 인돌 카복사미드 유도체 및 그를 포함하는 약제학적 조성물 |
| CN113233980B (zh) * | 2021-04-02 | 2022-04-05 | 台州学院 | 一种β-氯代酸酯及α,β-不饱和酸酯类化合物的合成方法 |
| CN118121595B (zh) * | 2024-05-06 | 2024-08-16 | 广州市朝利良生物科技有限公司 | 化合物eh-p005j在制备促伤口愈合药物中的用途 |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
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-
2005
- 2005-06-17 KR KR1020077001307A patent/KR20070028553A/ko not_active Withdrawn
- 2005-06-17 BR BRPI0512252-0A patent/BRPI0512252A/pt not_active IP Right Cessation
- 2005-06-17 AT AT05751812T patent/ATE405549T1/de not_active IP Right Cessation
- 2005-06-17 EP EP05751812A patent/EP1778632B1/en not_active Expired - Lifetime
- 2005-06-17 AU AU2005254782A patent/AU2005254782A1/en not_active Abandoned
- 2005-06-17 MX MXPA06014535A patent/MXPA06014535A/es unknown
- 2005-06-17 US US11/629,624 patent/US7705023B2/en not_active Expired - Fee Related
- 2005-06-17 CN CNA2005800277808A patent/CN101006053A/zh active Pending
- 2005-06-17 ZA ZA200610357A patent/ZA200610357B/en unknown
- 2005-06-17 ES ES05751812T patent/ES2315877T3/es not_active Expired - Lifetime
- 2005-06-17 WO PCT/GB2005/002391 patent/WO2005123673A1/en not_active Ceased
- 2005-06-17 RU RU2007101705/04A patent/RU2007101705A/ru not_active Application Discontinuation
- 2005-06-17 DE DE602005009209T patent/DE602005009209D1/de not_active Expired - Lifetime
- 2005-06-17 CA CA002570363A patent/CA2570363A1/en not_active Abandoned
- 2005-06-17 JP JP2007516043A patent/JP2008502669A/ja not_active Withdrawn
-
2006
- 2006-11-30 IL IL179728A patent/IL179728A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA06014535A (es) | 2007-06-05 |
| KR20070028553A (ko) | 2007-03-12 |
| RU2007101705A (ru) | 2008-07-27 |
| EP1778632A1 (en) | 2007-05-02 |
| BRPI0512252A (pt) | 2008-02-19 |
| EP1778632B1 (en) | 2008-08-20 |
| ATE405549T1 (de) | 2008-09-15 |
| WO2005123673A1 (en) | 2005-12-29 |
| CA2570363A1 (en) | 2005-12-29 |
| JP2008502669A (ja) | 2008-01-31 |
| ES2315877T3 (es) | 2009-04-01 |
| US20070287715A1 (en) | 2007-12-13 |
| DE602005009209D1 (de) | 2008-10-02 |
| IL179728A0 (en) | 2007-05-15 |
| AU2005254782A1 (en) | 2005-12-29 |
| US7705023B2 (en) | 2010-04-27 |
| CN101006053A (zh) | 2007-07-25 |
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