ZA200508863B - Template-fixed -hairpin peptidomimetics with CXCR4 antagonizing activity - Google Patents
Template-fixed -hairpin peptidomimetics with CXCR4 antagonizing activity Download PDFInfo
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- ZA200508863B ZA200508863B ZA200508863A ZA200508863A ZA200508863B ZA 200508863 B ZA200508863 B ZA 200508863B ZA 200508863 A ZA200508863 A ZA 200508863A ZA 200508863 A ZA200508863 A ZA 200508863A ZA 200508863 B ZA200508863 B ZA 200508863B
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- alkenyl
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Classifications
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- Biophysics (AREA)
- Biochemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Immunology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Analytical Chemistry (AREA)
- Epidemiology (AREA)
- Virology (AREA)
- Gastroenterology & Hepatology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pain & Pain Management (AREA)
- Tropical Medicine & Parasitology (AREA)
- AIDS & HIV (AREA)
- Rheumatology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cosmetics (AREA)
- Detergent Compositions (AREA)
- Treatment Of Liquids With Adsorbents In General (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/EP2003/004640 WO2004096839A1 (en) | 2003-05-02 | 2003-05-02 | Template-fixed beta-hairpin peptidomimetics with cxcr4 antagonizing activity |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200508863B true ZA200508863B (en) | 2007-03-28 |
Family
ID=33395700
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200508863A ZA200508863B (en) | 2003-05-02 | 2005-11-01 | Template-fixed -hairpin peptidomimetics with CXCR4 antagonizing activity |
Country Status (17)
| Country | Link |
|---|---|
| US (3) | US7786078B2 (no) |
| EP (3) | EP1622931B1 (no) |
| JP (3) | JP4846564B2 (no) |
| KR (5) | KR20130059463A (no) |
| CN (1) | CN1802385B (no) |
| AU (2) | AU2003232253A1 (no) |
| BR (3) | BRPI0409928B8 (no) |
| CA (3) | CA2524253C (no) |
| EA (1) | EA010163B1 (no) |
| ES (3) | ES2550856T3 (no) |
| HK (1) | HK1094210A1 (no) |
| IL (3) | IL171530A (no) |
| MX (1) | MXPA05011550A (no) |
| NO (2) | NO333793B1 (no) |
| NZ (1) | NZ543806A (no) |
| WO (2) | WO2004096839A1 (no) |
| ZA (1) | ZA200508863B (no) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN105111280B (zh) * | 2005-02-17 | 2020-01-24 | 波利弗尔有限公司 | 具有蛋白酶抑制活性的模板固定的β-发夹肽模拟物 |
| EP1856140B1 (en) * | 2005-02-17 | 2013-12-25 | Polyphor Ltd. | Template-fixed beta-hairpin peptidomimetics with protease inhibitory activity |
| WO2006117011A1 (en) * | 2005-05-02 | 2006-11-09 | Polyphor Ltd. | Dye conjugates of template-fixed peptidomimetics |
| ES2427989T3 (es) | 2005-10-28 | 2013-11-05 | Ono Pharmaceutical Co., Ltd. | Compuesto que contiene un grupo básico y uso del mismo |
| PL1961744T3 (pl) | 2005-11-18 | 2013-09-30 | Ono Pharmaceutical Co | Związek zawierający grupę zasadową oraz jego zastosowanie |
| WO2007079597A1 (en) * | 2006-01-16 | 2007-07-19 | Polyphor Ltd. | Template - fixed peptidomimetics with antimicrobial activity |
| AU2007345497B2 (en) * | 2007-01-29 | 2013-01-17 | Polyphor Ltd. | Template-fixed peptidomimetics |
| PL2132221T3 (pl) | 2007-02-28 | 2011-04-29 | Polyphor Ltd | Przyłączone do matrycy peptydomimetyki |
| WO2009074807A2 (en) | 2007-12-12 | 2009-06-18 | Imperial Innovations Limited | Methods |
| US20110230426A1 (en) * | 2008-08-08 | 2011-09-22 | Polyphor Ag | Template-fixed peptidomimetics |
| US8883720B2 (en) | 2008-11-26 | 2014-11-11 | Polyphor Ag | Template-fixed beta-hairpin peptidomimetics with CXCR4 antagonizing activity |
| WO2010127704A1 (en) * | 2009-05-07 | 2010-11-11 | Polyphor Ag | Beta-hairpin peptidomimetics having cxcr4 antagonizing activity |
| SG195055A1 (en) | 2011-06-07 | 2013-12-30 | Polyphor Ag | Beta - hairpin peptidomimetics as cxc4 antagonists |
| AR087363A1 (es) * | 2011-07-29 | 2014-03-19 | Pf Medicament | Uso del anticuerpo i-3859 para la deteccion y diagnostico de los canceres |
| WO2013050346A1 (en) | 2011-10-07 | 2013-04-11 | Polyphor Ag | Template -fixed peptidomimetics as inhibitors of fpr1 |
| ES2647076T3 (es) * | 2012-06-06 | 2017-12-19 | Polyphor Ag | Peptidomiméticos de horquilla beta |
| AU2013301576B2 (en) * | 2012-08-08 | 2017-10-19 | Polyphor Ag | Combinations with a backbone-cyclized peptide |
| US10544527B2 (en) * | 2015-03-24 | 2020-01-28 | Toray Industries, Inc. | Fabric and clothing having flame retardancy and high visibility |
| WO2017066454A2 (en) | 2015-10-14 | 2017-04-20 | X-Therma, Inc. | Compositions and methods for reducing ice crystal formation |
| EP3630153A2 (en) * | 2017-05-22 | 2020-04-08 | National Hellenic Research Foundation | Macrocyclic modulators of disease associated protein misfolding and aggregation |
| WO2023227771A1 (en) | 2022-05-27 | 2023-11-30 | Fundación Privada Instituto De Salud Global Barcelona | Cyclic peptides with antibacterial activity against multidrug resistant (mdr) pathogens |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE177114T1 (de) | 1993-10-14 | 1999-03-15 | Seikagaku Kogyo Co Ltd | Polypeptide und daraus hergestellte, gegen hiv wirksame substanzen |
| EP1214336A1 (en) * | 1999-08-30 | 2002-06-19 | Universität Zürich | Synthesis of template-fixed beta-hairpin loop mimetics |
| US7253146B2 (en) * | 2001-02-23 | 2007-08-07 | Polyphor Ltd | Template-fixed peptidomimetics with antimicrobial activity |
| CN101157924A (zh) * | 2001-12-11 | 2008-04-09 | 人体基因组科学有限公司 | 嗜中性白细胞因子α |
| AU2002342618C1 (en) * | 2002-08-20 | 2008-10-30 | Polyphor Ltd. | Template-fixed peptidomimetics with antibacterial activity |
| ATE393774T1 (de) * | 2002-10-02 | 2008-05-15 | Polyphor Ltd | Matrizenfixierte peptidomimetika mit antimikrobieller wirkung |
-
2003
- 2003-05-02 WO PCT/EP2003/004640 patent/WO2004096839A1/en active Application Filing
- 2003-05-02 AU AU2003232253A patent/AU2003232253A1/en not_active Abandoned
-
2004
- 2004-04-29 KR KR1020137011887A patent/KR20130059463A/ko not_active Application Discontinuation
- 2004-04-29 MX MXPA05011550A patent/MXPA05011550A/es active IP Right Grant
- 2004-04-29 EP EP04730251.8A patent/EP1622931B1/en not_active Expired - Lifetime
- 2004-04-29 EA EA200501550A patent/EA010163B1/ru not_active IP Right Cessation
- 2004-04-29 KR KR1020117013433A patent/KR101330238B1/ko active IP Right Grant
- 2004-04-29 EP EP12185905.2A patent/EP2540735B1/en not_active Expired - Lifetime
- 2004-04-29 BR BRPI0409928A patent/BRPI0409928B8/pt active IP Right Grant
- 2004-04-29 JP JP2006505321A patent/JP4846564B2/ja not_active Expired - Lifetime
- 2004-04-29 CA CA2524253A patent/CA2524253C/en not_active Expired - Lifetime
- 2004-04-29 ES ES12185905.2T patent/ES2550856T3/es not_active Expired - Lifetime
- 2004-04-29 BR BR122019016210A patent/BR122019016210B8/pt active IP Right Grant
- 2004-04-29 KR KR1020117013434A patent/KR101330239B1/ko active IP Right Grant
- 2004-04-29 ES ES04730251.8T patent/ES2550241T3/es not_active Expired - Lifetime
- 2004-04-29 CN CN2004800158452A patent/CN1802385B/zh not_active Expired - Lifetime
- 2004-04-29 CA CA2847486A patent/CA2847486C/en not_active Expired - Lifetime
- 2004-04-29 AU AU2004234062A patent/AU2004234062B2/en not_active Expired
- 2004-04-29 WO PCT/EP2004/004535 patent/WO2004096840A1/en active Application Filing
- 2004-04-29 BR BR122019016211A patent/BR122019016211B8/pt active IP Right Grant
- 2004-04-29 NZ NZ543806A patent/NZ543806A/en unknown
- 2004-04-29 KR KR1020057020836A patent/KR101230453B1/ko active IP Right Grant
- 2004-04-29 KR KR1020137011885A patent/KR20130059462A/ko not_active Application Discontinuation
- 2004-04-29 US US10/555,088 patent/US7786078B2/en active Active
- 2004-04-29 CA CA2847490A patent/CA2847490C/en not_active Expired - Lifetime
- 2004-04-29 EP EP12185927.6A patent/EP2540736B1/en not_active Expired - Lifetime
- 2004-04-29 ES ES12185927.6T patent/ES2563094T3/es not_active Expired - Lifetime
-
2005
- 2005-10-23 IL IL171530A patent/IL171530A/en active IP Right Grant
- 2005-11-01 ZA ZA200508863A patent/ZA200508863B/en unknown
- 2005-11-25 NO NO20055585A patent/NO333793B1/no unknown
-
2006
- 2006-12-22 HK HK06114147.7A patent/HK1094210A1/xx not_active IP Right Cessation
-
2010
- 2010-07-01 US US12/828,998 patent/US8895695B2/en active Active
-
2011
- 2011-02-18 JP JP2011033325A patent/JP5307169B2/ja not_active Expired - Lifetime
-
2013
- 2013-05-17 JP JP2013104857A patent/JP5770781B2/ja not_active Expired - Lifetime
- 2013-08-08 NO NO20131086A patent/NO340835B1/no not_active IP Right Cessation
- 2013-08-13 IL IL227933A patent/IL227933B/en active IP Right Grant
- 2013-08-13 IL IL227932A patent/IL227932B/en active IP Right Grant
-
2014
- 2014-09-24 US US14/495,737 patent/US9518092B2/en not_active Expired - Lifetime
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