ZA200403684B - Macrolides. - Google Patents

Macrolides.

Info

Publication number
ZA200403684B
ZA200403684B ZA200403684A ZA200403684A ZA200403684B ZA 200403684 B ZA200403684 B ZA 200403684B ZA 200403684 A ZA200403684 A ZA 200403684A ZA 200403684 A ZA200403684 A ZA 200403684A ZA 200403684 B ZA200403684 B ZA 200403684B
Authority
ZA
South Africa
Prior art keywords
macrolides
Prior art date
Application number
ZA200403684A
Other languages
English (en)
Inventor
Sulejman Alihodzic
Andrea Berdik
Stefano Biondi
Federica Damiani
Miljenko Dumic
Antun Hutinec
Sergio Luciuro
Zorica Marusic-Istuk
Alfredo Paio
Anna Quaglia
Vlado Stimac
Daniele Andreotti
Ilaria Bientinesi
Manuela Ciraco
Marko Djerek
Vesna Erakovic
Gorjana Lazarevski
Natasa Marsic
Stjepan Mutak
Drazen Pavlovic
Wolfgang Schoenfeld
Jessica Tibasco
Original Assignee
Glaxo Group Ltd
Pliva Istrazivacki Inst D O O
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd, Pliva Istrazivacki Inst D O O filed Critical Glaxo Group Ltd
Publication of ZA200403684B publication Critical patent/ZA200403684B/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Steroid Compounds (AREA)
ZA200403684A 2001-11-14 2004-05-13 Macrolides. ZA200403684B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0127349.9A GB0127349D0 (en) 2001-11-14 2001-11-14 Macrolides

Publications (1)

Publication Number Publication Date
ZA200403684B true ZA200403684B (en) 2005-09-13

Family

ID=9925777

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200403684A ZA200403684B (en) 2001-11-14 2004-05-13 Macrolides.

Country Status (20)

Country Link
US (1) US7202221B2 (zh)
EP (1) EP1453846B1 (zh)
JP (1) JP2005515978A (zh)
CN (1) CN1307194C (zh)
AR (1) AR037371A1 (zh)
AT (1) ATE362479T1 (zh)
BR (1) BR0214132A (zh)
CA (1) CA2466975A1 (zh)
DE (1) DE60220180T2 (zh)
EA (1) EA007433B1 (zh)
ES (1) ES2287332T3 (zh)
GB (1) GB0127349D0 (zh)
HR (1) HRP20040433A2 (zh)
HU (1) HUP0402225A3 (zh)
IL (1) IL161710A0 (zh)
PL (1) PL371472A1 (zh)
RS (1) RS41904A (zh)
UA (1) UA77210C2 (zh)
WO (1) WO2003042228A1 (zh)
ZA (1) ZA200403684B (zh)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6995143B2 (en) * 2002-02-28 2006-02-07 Basilea Pharmaceutica Ag Macrolides with antibacterial activity
US7135573B2 (en) 2002-05-13 2006-11-14 Enanta Pharmaceuticals, Inc. Processes for the preparation of O-(6-Pyrazol-1-yl-pyridin-3-ylmethyl)-hydroxylamine
US7910558B2 (en) 2002-05-13 2011-03-22 Enanta Pharmaceuticals, Inc. Bridged macrocyclic compounds and processes for the preparation thereof
US6764998B1 (en) 2003-06-18 2004-07-20 Enanta Pharmaceuticals, Inc. 6,11-4C-bicyclic 9a-azalide derivatives
WO2005070918A1 (en) 2002-05-13 2005-08-04 Enanta Pharmaceuticals, Inc. Process for the preparation of t-11 bicyclic erythromycin derivatives
CA2484308A1 (en) * 2002-05-14 2003-11-27 The Regents Of The University Of California Substituted quinolone carboxylic acids, their derivatives, site of action, and uses thereof
AR043050A1 (es) 2002-09-26 2005-07-13 Rib X Pharmaceuticals Inc Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos
GB0225384D0 (en) * 2002-10-31 2002-12-11 Glaxo Group Ltd Novel compounds
US6645941B1 (en) 2003-03-26 2003-11-11 Enanta Pharmaceuticals, Inc. 6,11-3C-bicyclic 9a-azalide derivatives
SI1628989T1 (sl) * 2003-05-13 2007-06-30 Glaxo Group Ltd Nove cikliäśne spojine s 14 in 15 obroäśnimi äśleni
GB0310980D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310984D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310979D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
GB0310986D0 (en) * 2003-05-13 2003-06-18 Glaxo Group Ltd Novel compounds
US7276487B2 (en) 2003-09-23 2007-10-02 Enanta Pharmaceuticals, Inc. 9a, 11-3C-bicyclic 9a-azalide derivatives
US7265094B2 (en) 2004-01-09 2007-09-04 Enanta Pharmaceuticals, Inc. 9N-substituted 6-11 bicyclic erythromycin derivatives
EP2716647A3 (en) 2004-02-27 2014-08-20 Rib-X Pharmaceuticals, Inc. Macrocyclic compounds and methods of making and using the same
US20080255060A1 (en) * 2004-05-06 2008-10-16 Sulejman Alihodzic Ester Linked Macrolides Useful For The Treatment of Microbial Infections
WO2005108413A1 (en) * 2004-05-06 2005-11-17 Glaxosmithkline Istrazivacki Centar Zagreb D.O.O Carbamate linked macrolides useful for the treatment of microbial infections
WO2006047167A2 (en) * 2004-10-21 2006-05-04 Janssen Pharmaceutica, N.V. 9 alkyl and 9 alkylidenyl 6-0 alkyl-11, 12 carbamate ketolide antimicrobials
GB0424959D0 (en) 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
GB0424958D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
GB0424951D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
GB0424961D0 (en) * 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
AU2007283556B2 (en) 2006-08-09 2011-10-06 Basilea Pharmaceutica Ag New macrolides useful against inflammatory and allergic disseases
JP2010501541A (ja) 2006-08-24 2010-01-21 ウォックハート リサーチ センター 抗菌活性を有する新規マクロライド及びケトライド
US8410065B2 (en) 2008-02-08 2013-04-02 Basilea Pharmaceutica Ag Macrolides and their use
ES2561332T3 (es) 2009-05-27 2016-02-25 Wockhardt Limited Compuestos cetólidos que tienen actividad antimicrobiana
WO2012076989A1 (en) 2010-12-09 2012-06-14 Wockhardt Limited Ketolide compounds
CN103380141A (zh) * 2011-01-31 2013-10-30 明治制果药业株式会社 新大环内酯衍生物
EP2681222B1 (en) 2011-03-01 2018-02-28 Wockhardt Limited Process for preparation of ketolide intermediates

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0126344A2 (en) 1983-05-20 1984-11-28 Abbott Laboratories Tripeptide esters of therapeutic agents
US4742049A (en) 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
IL93936A (en) 1989-03-28 1994-06-24 Abbott Lab History of 9-dioxo-21,9-epoxy - erythromycin, method of preparation History of 11-oxo and 11-hydroxy, and pharmaceutical preparations containing them
CA2064634C (en) * 1991-04-04 1998-08-04 James V. Heck 9-deoxo-8a-aza-8a-homoerythromycin a derivatives modified at the 4"- and8a-positions
BR9708929A (pt) 1996-05-07 1999-08-03 Abbott Lab Composto composição farmacêutica e processos para controlar uma infecção bacteriana em um mamífero e para preparar compostos de macrólidos
EP0895999A1 (en) * 1997-08-06 1999-02-10 Pfizer Products Inc. C-4" substituted macrolide antibiotics
US6262030B1 (en) 1998-11-03 2001-07-17 Pfizer Inc. Erythromycin derivatives
WO2000071557A1 (en) 1999-05-24 2000-11-30 Pfizer Products Inc. 13-methyl-erythromycin derivatives
DE60025370T2 (de) 1999-08-24 2006-09-21 Abbott Laboratories, Abbott Park 9a-azalide mit antibakterieller wirkung
ES2254389T3 (es) 2000-02-24 2006-06-16 Abbott Laboratories Agentes anti-infecciosos utiles contra cepas bacterianas resistntes a multiples farmacos.
US6946446B2 (en) 2000-02-24 2005-09-20 Abbott Laboratories Anti-infective agents useful against multidrug-resistant strains of bacteria
JP2002173498A (ja) 2000-09-27 2002-06-21 Hokuriku Seiyaku Co Ltd エリスロマイシン誘導体
GB0025688D0 (en) * 2000-10-19 2000-12-06 Glaxo Group Ltd Macrolides

Also Published As

Publication number Publication date
EA007433B1 (ru) 2006-10-27
DE60220180D1 (de) 2007-06-28
CA2466975A1 (en) 2003-05-22
US7202221B2 (en) 2007-04-10
US20050080025A1 (en) 2005-04-14
EP1453846B1 (en) 2007-05-16
EP1453846A1 (en) 2004-09-08
HRP20040433A2 (en) 2005-04-30
EA200400536A1 (ru) 2004-12-30
RS41904A (en) 2006-10-27
JP2005515978A (ja) 2005-06-02
BR0214132A (pt) 2004-09-14
ATE362479T1 (de) 2007-06-15
IL161710A0 (en) 2004-09-27
UA77210C2 (en) 2006-11-15
HUP0402225A3 (en) 2006-01-30
CN1307194C (zh) 2007-03-28
CN1612888A (zh) 2005-05-04
WO2003042228A1 (en) 2003-05-22
AR037371A1 (es) 2004-11-03
ES2287332T3 (es) 2007-12-16
GB0127349D0 (en) 2002-01-02
HUP0402225A2 (hu) 2005-02-28
PL371472A1 (en) 2005-06-13
DE60220180T2 (de) 2008-01-17

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