ZA200308782B - Piperazine oxime derivatives having NK-1 receptor antagonistic activity. - Google Patents

Piperazine oxime derivatives having NK-1 receptor antagonistic activity. Download PDF

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Publication number
ZA200308782B
ZA200308782B ZA200308782A ZA200308782A ZA200308782B ZA 200308782 B ZA200308782 B ZA 200308782B ZA 200308782 A ZA200308782 A ZA 200308782A ZA 200308782 A ZA200308782 A ZA 200308782A ZA 200308782 B ZA200308782 B ZA 200308782B
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disorders
disorder
substance
disease
compound
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ZA200308782A
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Inventor
Jan H Van Maarseveen
Martinus Th M Tulp
Wouter I Iwema Bakker
Amoldus H J Herremans
Gustaaf J M Van Scharrenburg
Andrew C Mccreary
Hein K A C Coolen
Adrianus Van Den Hoogenband
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Solvay Pharmaceutical B V
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Publication of ZA200308782B publication Critical patent/ZA200308782B/en

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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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  • Diabetes (AREA)
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ZA200308782A 2001-07-09 2003-11-11 Piperazine oxime derivatives having NK-1 receptor antagonistic activity. ZA200308782B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP01202631 2001-07-09

Publications (1)

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ZA200308782B true ZA200308782B (en) 2005-02-11

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ZA200308782A ZA200308782B (en) 2001-07-09 2003-11-11 Piperazine oxime derivatives having NK-1 receptor antagonistic activity.

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US (1) US7094779B2 (ko)
EP (1) EP1406894B1 (ko)
JP (1) JP3765543B2 (ko)
KR (1) KR100900889B1 (ko)
CN (1) CN1223591C (ko)
AR (1) AR034722A1 (ko)
AT (1) ATE285407T1 (ko)
AU (1) AU2002333229B2 (ko)
BR (1) BR0210080A (ko)
CA (1) CA2446726A1 (ko)
DE (1) DE60202371T2 (ko)
DK (1) DK1406894T3 (ko)
ES (1) ES2230521T3 (ko)
HK (1) HK1067364A1 (ko)
HR (1) HRP20030912A2 (ko)
HU (1) HUP0401093A3 (ko)
IL (2) IL158728A0 (ko)
MX (1) MXPA04000230A (ko)
NO (1) NO20040065L (ko)
PL (1) PL366841A1 (ko)
PT (1) PT1406894E (ko)
RU (1) RU2273639C2 (ko)
SI (1) SI1406894T1 (ko)
UA (1) UA75425C2 (ko)
WO (1) WO2003006459A1 (ko)
ZA (1) ZA200308782B (ko)

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KR100616099B1 (ko) * 2004-09-20 2006-08-28 한국과학기술연구원 Ｔ-타입 칼슘채널 길항제로 유효한 신규 피페라지닐알킬이소옥사졸 유도체
AU2006272951A1 (en) 2005-05-17 2007-02-01 Plexxikon, Inc. Pyrrol (2,3-b) pyridine derivatives protein kinase inhibitors
AU2006261993B2 (en) 2005-06-22 2011-11-17 Plexxikon, Inc. Pyrrolo (2, 3-B) pyridine derivatives as protein kinase inhibitors
WO2008063888A2 (en) 2006-11-22 2008-05-29 Plexxikon, Inc. Compounds modulating c-fms and/or c-kit activity and uses therefor
US20100168197A1 (en) * 2007-02-28 2010-07-01 Naresh Kumar Muscarinic receptor antagonists
EP2170830B1 (en) 2007-07-17 2014-10-15 Plexxikon, Inc. 2-FLUORO-BENZENESULFONAMIDE COMPOUNDS AS Raf KINASE MODULATORS
AU2010232670B2 (en) 2009-04-03 2015-07-09 F. Hoffmann-La Roche Ag Propane- I-sulfonic acid {3- [5- (4 -chloro-phenyl) -1H-pyrrolo [2, 3-b] pyridine-3-carbonyl] -2, 4-difluoro-pheny l } -amide compositions and uses thereof
PE20121327A1 (es) 2009-11-06 2012-10-18 Plexxikon Inc Compuestos y metodos para la modulacion de cinasas, e indicaciones para ello
PL2672967T3 (pl) 2011-02-07 2019-04-30 Plexxikon Inc Związki i sposoby modulacji kinaz i wskazania ku temu
TWI558702B (zh) 2011-02-21 2016-11-21 普雷辛肯公司 醫藥活性物質的固態形式
US9150570B2 (en) 2012-05-31 2015-10-06 Plexxikon Inc. Synthesis of heterocyclic compounds
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CN110615774B (zh) * 2019-09-19 2022-11-11 安徽中医药大学 具有抗炎活性的苄基哌嗪类化合物、制法及医药用途
JP2022090346A (ja) 2020-12-07 2022-06-17 三星電子株式会社 共重合体、ならびに当該共重合体を用いるエレクトロルミネッセンス素子材料およびエレクトロルミネッセンス素子

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