ZA200307474B - CCR5 antagonists useful for treating AIDS. - Google Patents
CCR5 antagonists useful for treating AIDS. Download PDFInfo
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- ZA200307474B ZA200307474B ZA200307474A ZA200307474A ZA200307474B ZA 200307474 B ZA200307474 B ZA 200307474B ZA 200307474 A ZA200307474 A ZA 200307474A ZA 200307474 A ZA200307474 A ZA 200307474A ZA 200307474 B ZA200307474 B ZA 200307474B
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Landscapes
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| PE20040769A1 (es) | 2002-12-18 | 2004-11-06 | Schering Corp | Derivados de piperidina utiles como antagonisas ccr5 |
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| US7705153B2 (en) * | 2004-02-05 | 2010-04-27 | Schering Corporation | Bipiperdine derivatives useful as CCR3 antagonists |
| SE0400925D0 (sv) * | 2004-04-06 | 2004-04-06 | Astrazeneca Ab | Chemical compounds |
| US7678798B2 (en) * | 2004-04-13 | 2010-03-16 | Incyte Corporation | Piperazinylpiperidine derivatives as chemokine receptor antagonists |
| NZ553696A (en) | 2004-09-13 | 2010-02-26 | Ono Pharmaceutical Co | Nitrogenous heterocyclic derivative and medicine containing the same as an active ingredient |
| US7635698B2 (en) | 2004-12-29 | 2009-12-22 | Millennium Pharmaceuticals, Inc. | Compounds useful as chemokine receptor antagonists |
| WO2006071875A1 (fr) * | 2004-12-29 | 2006-07-06 | Millennium Pharmaceuticals, Inc. | Composes utilises comme antagonistes des recepteurs de la chemokine |
| AR054422A1 (es) * | 2005-01-06 | 2007-06-27 | Schering Corp | Sintesis de los antagonistas del receptor ccr5. compuestos relacionados |
| SG158858A1 (en) * | 2005-01-06 | 2010-02-26 | Schering Corp | Preparation of pharmaceutical salts of piperazine compounds |
| JP4769257B2 (ja) * | 2005-02-23 | 2011-09-07 | シェーリング コーポレイション | ケモカインレセプターのインヒビターとして有用なピペリジニルピペラジン誘導体 |
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| US7462485B2 (en) * | 2005-10-07 | 2008-12-09 | Glaser Lawrence F | Modified erythrocytes and uses thereof |
| TW200745087A (en) * | 2006-02-24 | 2007-12-16 | Schering Corp | CCR5 antagonists useful for treating HIV |
| WO2008030853A2 (fr) * | 2006-09-06 | 2008-03-13 | Incyte Corporation | Thérapie de combinaison contre l'infection par le virus de l'immunodéficience humaine |
| US20100063280A1 (en) * | 2006-12-22 | 2010-03-11 | Schering Corporation | Process for preparing ccr-5 receptor antagonists utilizing 4-substituted 1-cyclopropane-sulfonyl-piperidinyl compounds |
| AU2009220462A1 (en) * | 2008-02-29 | 2009-09-11 | Merck Sharp & Dohme Corp. | CCR5 antagonists as prophylactics for preventing HIV infection and methods of inhibiting transmission of same |
| US11629196B2 (en) | 2020-04-27 | 2023-04-18 | Incelldx, Inc. | Method of treating SARS-CoV-2-associated hypercytokinemia by administering a human monoclonal antibody (PRO-140) that inhibits CCR5/CCL5 binding interactions |
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| US5368854A (en) | 1992-08-20 | 1994-11-29 | Schering Corporation | Use of IL-10 to treat inflammatory bowel disease |
| WO1994018192A1 (fr) | 1993-02-12 | 1994-08-18 | Merck & Co., Inc. | Derives de piperazine utiles comme inhibiteurs de la protease du vih |
| US5889006A (en) | 1995-02-23 | 1999-03-30 | Schering Corporation | Muscarinic antagonists |
| IL117149A0 (en) | 1995-02-23 | 1996-06-18 | Schering Corp | Muscarinic antagonists |
| WO1996040300A2 (fr) | 1995-06-07 | 1996-12-19 | Kimberly-Clark Worldwide, Inc. | Inhibition d'exoproteines dans un article absorbant |
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| TW531537B (en) | 1995-12-27 | 2003-05-11 | Janssen Pharmaceutica Nv | 1-(1,2-disubstituted piperidinyl)-4-substituted piperidine derivatives |
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| WO2000066558A1 (fr) * | 1999-05-04 | 2000-11-09 | Schering Corporation | Derives de piperazine faisant office d'antagonistes ccr5 |
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2002
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- 2002-03-27 PE PE2002000251A patent/PE20020996A1/es not_active Application Discontinuation
- 2002-03-27 EP EP05009882A patent/EP1591444B1/fr not_active Expired - Lifetime
- 2002-03-27 US US10/107,940 patent/US6720325B2/en not_active Expired - Lifetime
- 2002-03-27 SK SK1196-2003A patent/SK287521B6/sk not_active IP Right Cessation
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- 2002-03-27 WO PCT/US2002/009491 patent/WO2002079194A1/fr active IP Right Grant
- 2002-03-27 EP EP02725381A patent/EP1373256B1/fr not_active Expired - Lifetime
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- 2002-03-27 IL IL15755102A patent/IL157551A0/xx not_active IP Right Cessation
- 2002-03-27 SI SI200230169T patent/SI1373256T1/sl unknown
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- 2002-03-27 CA CA002442227A patent/CA2442227C/fr not_active Expired - Fee Related
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- 2002-03-27 AT AT02725381T patent/ATE299139T1/de active
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- 2002-03-27 DK DK02725381T patent/DK1373256T3/da active
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2006
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