ZA200303432B - SN-38 lipid complexes and methods of use. - Google Patents

SN-38 lipid complexes and methods of use. Download PDF

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Publication number
ZA200303432B
ZA200303432B ZA200303432A ZA200303432A ZA200303432B ZA 200303432 B ZA200303432 B ZA 200303432B ZA 200303432 A ZA200303432 A ZA 200303432A ZA 200303432 A ZA200303432 A ZA 200303432A ZA 200303432 B ZA200303432 B ZA 200303432B
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ZA
South Africa
Prior art keywords
composition
lipid
compound
liposomes
cardiolipin
Prior art date
Application number
ZA200303432A
Other languages
English (en)
Inventor
Imran Ahmad
Aquilur Rahman
Jia-Ai Allen Zhang
Original Assignee
Neopharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neopharm Inc filed Critical Neopharm Inc
Publication of ZA200303432B publication Critical patent/ZA200303432B/en

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/127—Liposomes
    • A61K9/1271—Non-conventional liposomes, e.g. PEGylated liposomes, liposomes coated with polymers
    • A61K9/1272—Non-conventional liposomes, e.g. PEGylated liposomes, liposomes coated with polymers with substantial amounts of non-phosphatidyl, i.e. non-acylglycerophosphate, surfactants as bilayer-forming substances, e.g. cationic lipids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/69—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit
    • A61K47/6905—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit the form being a colloid or an emulsion
    • A61K47/6911—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit the form being a colloid or an emulsion the form being a liposome
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dispersion Chemistry (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
ZA200303432A 2000-11-09 2003-05-05 SN-38 lipid complexes and methods of use. ZA200303432B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US24730600P 2000-11-09 2000-11-09

Publications (1)

Publication Number Publication Date
ZA200303432B true ZA200303432B (en) 2004-08-05

Family

ID=22934406

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200303432A ZA200303432B (en) 2000-11-09 2003-05-05 SN-38 lipid complexes and methods of use.

Country Status (22)

Country Link
US (1) US7390502B2 (fr)
EP (1) EP1355634B8 (fr)
JP (1) JP4524071B2 (fr)
KR (1) KR100869824B1 (fr)
CN (1) CN1531424A (fr)
AT (1) ATE413164T1 (fr)
AU (1) AU2002246510B2 (fr)
BG (1) BG107862A (fr)
BR (1) BR0115260A (fr)
CA (1) CA2427467C (fr)
CZ (1) CZ20031515A3 (fr)
DE (1) DE60136490D1 (fr)
EA (1) EA006741B1 (fr)
HU (1) HUP0302352A3 (fr)
IL (1) IL155696A0 (fr)
MX (1) MXPA03004095A (fr)
NO (1) NO20032069L (fr)
NZ (1) NZ525552A (fr)
PL (1) PL363618A1 (fr)
SK (1) SK7092003A3 (fr)
WO (1) WO2002058622A2 (fr)
ZA (1) ZA200303432B (fr)

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WO2004035032A2 (fr) * 2002-08-20 2004-04-29 Neopharm, Inc. Formulation de sn-38 a base de lipides pharmaceutiquement actifs
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US20050277611A1 (en) * 2002-10-16 2005-12-15 Neopharm, Inc. Cationic cardiolipin analoges and its use thereof
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MX2016010998A (es) 2014-02-27 2017-03-31 Lycera Corp Terapia celular adoptiva que usa un agonista de receptor huérfano gamma relacionado con receptor de ácido retinoico y métodos terapéuticos relacionados.
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US10611740B2 (en) 2015-06-11 2020-04-07 Lycera Corporation Aryl dihydro-2H-benzo[b][1,4]oxazine sulfonamide and related compounds for use as agonists of RORγ and the treatment of disease
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HUP0302352A3 (en) 2007-03-28
KR100869824B1 (ko) 2008-11-21
EP1355634A2 (fr) 2003-10-29
BR0115260A (pt) 2005-08-16
CN1531424A (zh) 2004-09-22
EA200300550A1 (ru) 2004-06-24
EP1355634B1 (fr) 2008-11-05
CA2427467A1 (fr) 2002-08-01
EA006741B1 (ru) 2006-04-28
KR20030072352A (ko) 2003-09-13
IL155696A0 (en) 2003-11-23
US20030215492A1 (en) 2003-11-20
DE60136490D1 (de) 2008-12-18
JP2004529086A (ja) 2004-09-24
CA2427467C (fr) 2010-01-12
EP1355634A4 (fr) 2005-07-06
MXPA03004095A (es) 2004-09-10
US7390502B2 (en) 2008-06-24
NO20032069D0 (no) 2003-05-08
EP1355634B8 (fr) 2009-03-04
ATE413164T1 (de) 2008-11-15
CZ20031515A3 (cs) 2003-09-17
AU2002246510B2 (en) 2007-09-20
NO20032069L (no) 2003-07-02
SK7092003A3 (en) 2004-06-08
WO2002058622A2 (fr) 2002-08-01
HUP0302352A2 (hu) 2003-11-28
AU2002246510A2 (en) 2002-08-06
BG107862A (bg) 2004-06-30
WO2002058622A3 (fr) 2003-08-28
JP4524071B2 (ja) 2010-08-11
PL363618A1 (en) 2004-11-29
NZ525552A (en) 2005-04-29

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