YU49485B - Nova kristalna modifikacija cdch, postupak za njeno pripremanje i farmaceutski preparati koji je sadrže - Google Patents

Nova kristalna modifikacija cdch, postupak za njeno pripremanje i farmaceutski preparati koji je sadrže

Info

Publication number
YU49485B
YU49485B YU65096A YU65096A YU49485B YU 49485 B YU49485 B YU 49485B YU 65096 A YU65096 A YU 65096A YU 65096 A YU65096 A YU 65096A YU 49485 B YU49485 B YU 49485B
Authority
YU
Yugoslavia
Prior art keywords
cdch
preparation
pharmaceutical preparations
preparations containing
crystal modification
Prior art date
Application number
YU65096A
Other languages
English (en)
Serbo-Croatian (sh)
Other versions
YU65096A (sh
Inventor
Alfons Grunenberg
Patrick Bosché
Original Assignee
Bayer Health Care Ag.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7779831&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=YU49485(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Health Care Ag. filed Critical Bayer Health Care Ag.
Publication of YU65096A publication Critical patent/YU65096A/sh
Publication of YU49485B publication Critical patent/YU49485B/sh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
YU65096A 1995-12-12 1996-12-06 Nova kristalna modifikacija cdch, postupak za njeno pripremanje i farmaceutski preparati koji je sadrže YU49485B (sh)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19546249A DE19546249A1 (de) 1995-12-12 1995-12-12 Neue Kristallmodifikation des 1-Cyclopropyl-7-([S,S]-2,8-diazabicyclo[4,3,0]non-8-yl)-6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäure Hydrochlorid (CDCH), Verfahren zu dessen Herstellung und diese enthaltende pharmazeutische Zubereitungen

Publications (2)

Publication Number Publication Date
YU65096A YU65096A (sh) 1998-12-23
YU49485B true YU49485B (sh) 2006-08-17

Family

ID=7779831

Family Applications (1)

Application Number Title Priority Date Filing Date
YU65096A YU49485B (sh) 1995-12-12 1996-12-06 Nova kristalna modifikacija cdch, postupak za njeno pripremanje i farmaceutski preparati koji je sadrže

Country Status (42)

Country Link
US (1) US5849752A (OSRAM)
EP (1) EP0780390B1 (OSRAM)
JP (1) JP4104687B2 (OSRAM)
KR (1) KR100525146B1 (OSRAM)
CN (1) CN1061348C (OSRAM)
AR (1) AR005009A1 (OSRAM)
AT (1) ATE221531T1 (OSRAM)
AU (1) AU708006B2 (OSRAM)
BG (1) BG62258B1 (OSRAM)
BR (1) BR9605968A (OSRAM)
CA (1) CA2192418C (OSRAM)
CO (1) CO4480105A1 (OSRAM)
CU (1) CU22774A3 (OSRAM)
CZ (1) CZ288657B6 (OSRAM)
DE (2) DE19546249A1 (OSRAM)
DK (1) DK0780390T3 (OSRAM)
EE (1) EE03474B1 (OSRAM)
ES (1) ES2179910T3 (OSRAM)
HR (1) HRP960558B1 (OSRAM)
HU (1) HU226521B1 (OSRAM)
ID (1) ID22625A (OSRAM)
IL (1) IL119795A (OSRAM)
IN (1) IN185805B (OSRAM)
MA (1) MA24342A1 (OSRAM)
MY (1) MY117492A (OSRAM)
NL (1) NL300109I1 (OSRAM)
NO (1) NO306725B1 (OSRAM)
NZ (1) NZ299905A (OSRAM)
PL (1) PL184885B1 (OSRAM)
PT (1) PT780390E (OSRAM)
RO (1) RO119782B1 (OSRAM)
RU (1) RU2162468C2 (OSRAM)
SA (1) SA96170492B1 (OSRAM)
SG (1) SG47201A1 (OSRAM)
SI (1) SI0780390T1 (OSRAM)
SK (1) SK282805B6 (OSRAM)
SV (1) SV1996000109A (OSRAM)
TR (1) TR199600970A2 (OSRAM)
TW (1) TW411340B (OSRAM)
UA (1) UA35638C2 (OSRAM)
YU (1) YU49485B (OSRAM)
ZA (1) ZA9610405B (OSRAM)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6270799B1 (en) * 1997-09-25 2001-08-07 Bayer Aktiengesellscahft Medicament formulation with a controlled release of an active agent
DE19751948A1 (de) 1997-11-24 1999-05-27 Bayer Ag Verfahren zur Herstellung von 8-Methoxy-Chinoloncarbonsäuren
US6716830B2 (en) 1998-09-30 2004-04-06 Alcon, Inc. Ophthalmic antibiotic compositions containing moxifloxacin
US6395746B1 (en) 1998-09-30 2002-05-28 Alcon Manufacturing, Ltd. Methods of treating ophthalmic, otic and nasal infections and attendant inflammation
US6509327B1 (en) 1998-09-30 2003-01-21 Alcon Manufacturing, Ltd. Compositions and methods for treating otic, ophthalmic and nasal infections
KR100650489B1 (ko) * 1998-11-10 2006-11-28 바이엘 헬스케어 아게 목시플록사신 제약 제제
DE19854357A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Semi-Hydrochlorid von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo/4.3.0/ -nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854356A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation A von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo-/4.3.0/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854355A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation B von 8-Cyan-1-cyclopropyl-7-(1S, 6S-2,8-diazabicyclo-/4.3.O/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19908449A1 (de) * 1999-02-26 2000-08-31 Bayer Ag Kristallmodifikation C von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicylo-[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chino/incarbonsäure
US20060252789A1 (en) * 2002-10-31 2006-11-09 Sujay Biswas Amorphous moxifloxacin hydrochloride
EP2113505A1 (en) 2003-04-09 2009-11-04 Dr. Reddy's Laboratories, Ltd. A crystalline form III of anhydrous moxifloxacin hydrochloride and processes for the preparation thereof
US20060264635A1 (en) * 2003-08-05 2006-11-23 Chava Satyanarayana Process for the preparation of moxifloxacin hydrochloride
ITMI20032259A1 (it) 2003-11-20 2005-05-21 Chemi Spa Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione
ES2319125T3 (es) * 2003-11-20 2009-05-04 Chemi S.P.A. Polimorfos del clorhidrato del acido 1-ciclopropil-7-((s,s)-2,8-diazadiciclo(4.3.0)-non-8-il)-6-fluoro-1,4-dihidro-8-metoxi-4-oxo-3-quinolina carboxilico y metodos para la preparacion de los mismos.
US7491725B2 (en) 2004-02-06 2009-02-17 Bristol-Myers Squibb Company Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
DE102004015981A1 (de) * 2004-04-01 2005-10-20 Bayer Healthcare Ag Neue kirstalline Form von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE102004063347A1 (de) * 2004-12-23 2006-07-13 Stada Arzneimittel Ag Gebrauchsfertige Gemcitabinlösungen und Gemcitabinlösungskonzentrate
WO2007033515A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation orale contenant de la moxifloxacine et son procédé de préparation
GB0612422D0 (en) * 2006-06-23 2006-08-02 Generics Uk Ltd Novel hydrate form
SI2032521T1 (sl) 2006-06-27 2010-02-26 Sandoz Ag Nov postopek za pripravo soli
ES2303768B1 (es) * 2006-09-08 2009-06-05 Quimica Sintetica, S.A. Nueva forma cristalina de moxifloxacino clorhidrato.
NZ576929A (en) 2006-11-13 2012-07-27 Cipla Ltd Crystalline anhydrous form C of moxifloxacin hydrochloride
EP1992626A1 (en) * 2007-05-10 2008-11-19 Sandoz AG Process for the preparation of moxifloxacin hydrochloride
EP2083010A1 (en) * 2008-01-08 2009-07-29 Chemo Ibérica, S.A. Polymorphic Forms of Moxifloxacin hydrochloride and processes for preparation thereof
EP2154137A1 (en) 2008-08-04 2010-02-17 Chemo Ibérica, S.A. Crystalline form of moxifloxacin base
EA201170545A1 (ru) * 2008-10-09 2012-01-30 Абды Ибрахым Иладж Санайи Ве Тыджарет Аноным Сыркеты Применение органических растворителей в способе влажного гранулирования моксифлоксацина
WO2010052726A1 (en) * 2008-11-06 2010-05-14 Hetero Research Foundation Novel polymorph of moxifloxacin hydrochloride
US20110293717A1 (en) 2008-12-08 2011-12-01 Ratiopharm Gmbh Compacted moxifloxacin
EA201101564A1 (ru) 2009-05-15 2012-07-30 Редкс Фарма Лимитед Редокс производные лекарственных средств
WO2011121596A2 (en) * 2010-04-01 2011-10-06 Neuland Laboratories Ltd. Crystal modification of moxifloxacin hydrochloride
BRPI1106900A2 (pt) 2011-12-26 2013-11-05 Ems Sa Composição farmacêutica sólida compreendendo antibótico da familia das quinolonas e processo de sua obtenção
FR2992218B1 (fr) 2012-06-22 2015-01-23 Rivopharm Sa Composition pharmaceutique de chlorhydrate de moxifloxacine et procede de preparation
CN102924449B (zh) * 2012-10-30 2015-08-12 重庆福安药业集团庆余堂制药有限公司 盐酸莫西沙星h晶型及其制备方法和药物组合物
EP2928892B1 (en) 2012-12-04 2018-03-21 Mankind Pharma Ltd. An improved process for the preparation of moxifloxacin hydrochloride
RU2561037C2 (ru) * 2013-02-07 2015-08-20 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Антибактериальная фармацевтическая композиция и способ ее получения
EP2969004A4 (en) 2013-03-15 2016-09-21 Melinta Therapeutics Inc METHOD FOR THE TREATMENT OF INFECTIONS IN OVERWEIGHT AND ADIPOSIVE PATIENTS USING ANTIBIOTICS

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3601567A1 (de) * 1986-01-21 1987-07-23 Bayer Ag 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
FI871419A7 (fi) * 1986-03-31 1987-10-01 Sankyo Co Kinoliini-3-karboksyylihappojohdannaiset, niiden valmistus ja käyttö
AU609974B2 (en) * 1988-05-18 1991-05-09 Warner-Lambert Company Improved process for the preparation of 5-amino-7- (substituted amino)-quinoline-3-carboxylic acids
DE3910663A1 (de) * 1989-04-03 1990-10-04 Bayer Ag 5-alkylchinoloncarbonsaeuren
RO108347B1 (ro) * 1989-10-30 1994-04-28 Bellon Labor Sa Roger DERIVATI DE BENZO-(b)-NAFTIRIDIN-1,8 SI PROCEDEU DE PREPARARE A ACESTORA
TW209865B (OSRAM) 1992-01-10 1993-07-21 Bayer Ag
ATE207479T1 (de) * 1992-01-31 2001-11-15 Chugai Pharmaceutical Co Ltd Kristalle von derivaten von chinozon carbonsäure- hydraten
DE4234078A1 (de) * 1992-10-09 1994-04-14 Bayer Ag Chinoloncarbonsäuren
CA2112165C (en) * 1992-12-25 2003-04-08 Makoto Takemura Bicyclic amine derivatives
ZA946853B (en) * 1993-09-10 1995-04-24 Daiichi Seiyaku Co Crystals of antimicrobial compound.
ES2121293T3 (es) * 1994-04-07 1998-11-16 Pfizer Uso de trovafloxacina o derivados de la misma para la fabricacion de un medicamento para el tratamiento de infecciones por h. pylori.

Also Published As

Publication number Publication date
ATE221531T1 (de) 2002-08-15
CZ288657B6 (cs) 2001-08-15
SV1996000109A (es) 1997-10-23
AU708006B2 (en) 1999-07-29
ES2179910T3 (es) 2003-02-01
NO965298L (no) 1997-06-13
CN1160052A (zh) 1997-09-24
BG62258B1 (bg) 1999-06-30
HU9603428D0 (en) 1997-01-28
NZ299905A (en) 1998-09-24
SA96170492B1 (ar) 2006-05-23
SI0780390T1 (en) 2002-10-31
CO4480105A1 (es) 1997-07-09
EP0780390A1 (de) 1997-06-25
DE59609501D1 (de) 2002-09-05
EE03474B1 (et) 2001-08-15
PT780390E (pt) 2002-11-29
AR005009A1 (es) 1999-04-07
NO965298D0 (no) 1996-12-11
CU22774A3 (es) 2002-07-24
JPH09169757A (ja) 1997-06-30
CN1061348C (zh) 2001-01-31
BR9605968A (pt) 1998-08-18
HRP960558A2 (en) 1998-02-28
SK282805B6 (sk) 2002-12-03
NL300109I1 (nl) 2003-02-03
HUP9603428A2 (en) 1997-08-28
KR970042550A (ko) 1997-07-24
RO119782B1 (ro) 2005-03-30
MY117492A (en) 2004-07-31
TW411340B (en) 2000-11-11
MX9606325A (es) 1997-10-31
KR100525146B1 (ko) 2006-01-27
RU2162468C2 (ru) 2001-01-27
PL317415A1 (en) 1997-06-23
CA2192418C (en) 2001-06-12
ID22625A (id) 1999-12-02
HRP960558B1 (en) 2002-04-30
AU7421696A (en) 1997-06-19
HU226521B1 (en) 2009-03-30
IL119795A0 (en) 1997-03-18
ZA9610405B (en) 1997-06-23
TR199600970A2 (tr) 1997-06-21
IL119795A (en) 1998-12-27
DK0780390T3 (da) 2002-11-11
JP4104687B2 (ja) 2008-06-18
HUP9603428A3 (en) 1997-10-28
BG101043A (en) 1998-04-30
EE9600201A (et) 1997-06-16
YU65096A (sh) 1998-12-23
UA35638C2 (uk) 2001-04-16
CA2192418A1 (en) 1997-06-13
MA24342A1 (fr) 1998-07-01
SG47201A1 (en) 1998-03-20
CZ364696A3 (en) 1997-07-16
US5849752A (en) 1998-12-15
EP0780390B1 (de) 2002-07-31
SK159196A3 (en) 1997-10-08
PL184885B1 (pl) 2003-01-31
NO306725B1 (no) 1999-12-13
IN185805B (OSRAM) 2001-05-05
DE19546249A1 (de) 1997-06-19

Similar Documents

Publication Publication Date Title
YU49485B (sh) Nova kristalna modifikacija cdch, postupak za njeno pripremanje i farmaceutski preparati koji je sadrže
TW334418B (en) Stilbene derivatives and pharmaceutical compositions
BR9408246A (pt) Composto derivado de 3-azabicicloalcano N-substituído
BG103485A (en) Ketobanzamides as calpain inhibitors
MEP24608A (en) Azetidine derivatives, preparation thereof and pharmaceutical compositions containing same
CA2338600A1 (en) Novel thiazolopyrimidine compounds
HUP9900617A3 (en) Novel indole-, indoline- or tetrahydrokinoline derivatives as acat and lipid peroxidation inhibitors, use thereof, pharmaceutical compositions containing these compounds
MY119042A (en) Dolastatin derivatives, their preparation and use
GR3033661T3 (en) Novel mercaptoacetylamido 1,3,4,5-tetrahydro-benzo(c)azepin-3-one disulfide derivatives useful as inhibitors of enkephalinase and ace
DK537389D0 (da) Glycosidase-inhibitoren salbostatin, dens fremstilling og anvendelse
IT1293778B1 (it) 1,4,7,10-tetraazabiciclo(8.2.2.)tetradecan-2 one, sua preparazione e suo uso per la preparazione di tetraazamacrocicli
CA2245267A1 (en) Crystal form of n-(4-trifluoromethylphenyl)-5-methylisoxazole-4-carboxamide
PT722319E (pt) Derivados de antraciclinona e a sua utilizacao no tratamento da amiloidose
RU94022277A (ru) Новые 19-норстероиды, имеющие в положении 11 - бета феноксиалкилсульфонамидную или феноксиалкилсульфонилкарбамидную цепь, метод и промежуточные продукты их получения, и содержащая их фармацевтическая композиция
CA2152771A1 (en) 7-o-ethers of taxane derivatives
PT736029E (pt) Sulfamatos de pseudofructopiranose anticonvulsivos
SG64906A1 (en) New bis-naphthalimides for the treatment of cancer
RU95112519A (ru) (3,4-ди-фторфенокси)метил оксиран и способ его получения
MY114282A (en) Anthracycline derivatives
DK0490816T3 (da) Fluorforbindelser som aromatase-inhibitorer.
CA2092694A1 (en) Use of pyridylmethylsulphinyl-1h-benzimidazole derivates in the treatment of illnesses caused by helicobacter bacteria
ITMI932189A0 (it) Composizioni farmaceutiche contenenti n-acetilcarnosina per il trattamento della cataratta
ATE40987T1 (de) Acetylenische phenoxypropanolderivate und pharmazeutische zusammensetzungen fuer die behandlung von bluthochdruck.
MY115430A (en) Glutaramide derivatives.
NO960812L (no) Alkoksysubstituerte ptoren