ID22625A - Modifikasi kristal baru dari cdch, suatu proses untuk preparatnya dan formulasi farmasi terdiri dari modifikasi - Google Patents

Modifikasi kristal baru dari cdch, suatu proses untuk preparatnya dan formulasi farmasi terdiri dari modifikasi

Info

Publication number
ID22625A
ID22625A IDP963684A ID963684A ID22625A ID 22625 A ID22625 A ID 22625A ID P963684 A IDP963684 A ID P963684A ID 963684 A ID963684 A ID 963684A ID 22625 A ID22625 A ID 22625A
Authority
ID
Indonesia
Prior art keywords
modification
cdch
preparation
formulation containing
new crystals
Prior art date
Application number
IDP963684A
Other languages
English (en)
Indonesian (id)
Inventor
Alfons Dr Grunenberg
Patrick Dr Bosche
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7779831&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ID22625(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of ID22625A publication Critical patent/ID22625A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IDP963684A 1995-12-12 1996-12-10 Modifikasi kristal baru dari cdch, suatu proses untuk preparatnya dan formulasi farmasi terdiri dari modifikasi ID22625A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19546249A DE19546249A1 (de) 1995-12-12 1995-12-12 Neue Kristallmodifikation des 1-Cyclopropyl-7-([S,S]-2,8-diazabicyclo[4,3,0]non-8-yl)-6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäure Hydrochlorid (CDCH), Verfahren zu dessen Herstellung und diese enthaltende pharmazeutische Zubereitungen

Publications (1)

Publication Number Publication Date
ID22625A true ID22625A (id) 1999-12-02

Family

ID=7779831

Family Applications (1)

Application Number Title Priority Date Filing Date
IDP963684A ID22625A (id) 1995-12-12 1996-12-10 Modifikasi kristal baru dari cdch, suatu proses untuk preparatnya dan formulasi farmasi terdiri dari modifikasi

Country Status (42)

Country Link
US (1) US5849752A (OSRAM)
EP (1) EP0780390B1 (OSRAM)
JP (1) JP4104687B2 (OSRAM)
KR (1) KR100525146B1 (OSRAM)
CN (1) CN1061348C (OSRAM)
AR (1) AR005009A1 (OSRAM)
AT (1) ATE221531T1 (OSRAM)
AU (1) AU708006B2 (OSRAM)
BG (1) BG62258B1 (OSRAM)
BR (1) BR9605968A (OSRAM)
CA (1) CA2192418C (OSRAM)
CO (1) CO4480105A1 (OSRAM)
CU (1) CU22774A3 (OSRAM)
CZ (1) CZ288657B6 (OSRAM)
DE (2) DE19546249A1 (OSRAM)
DK (1) DK0780390T3 (OSRAM)
EE (1) EE03474B1 (OSRAM)
ES (1) ES2179910T3 (OSRAM)
HR (1) HRP960558B1 (OSRAM)
HU (1) HU226521B1 (OSRAM)
ID (1) ID22625A (OSRAM)
IL (1) IL119795A (OSRAM)
IN (1) IN185805B (OSRAM)
MA (1) MA24342A1 (OSRAM)
MY (1) MY117492A (OSRAM)
NL (1) NL300109I1 (OSRAM)
NO (1) NO306725B1 (OSRAM)
NZ (1) NZ299905A (OSRAM)
PL (1) PL184885B1 (OSRAM)
PT (1) PT780390E (OSRAM)
RO (1) RO119782B1 (OSRAM)
RU (1) RU2162468C2 (OSRAM)
SA (1) SA96170492B1 (OSRAM)
SG (1) SG47201A1 (OSRAM)
SI (1) SI0780390T1 (OSRAM)
SK (1) SK282805B6 (OSRAM)
SV (1) SV1996000109A (OSRAM)
TR (1) TR199600970A2 (OSRAM)
TW (1) TW411340B (OSRAM)
UA (1) UA35638C2 (OSRAM)
YU (1) YU49485B (OSRAM)
ZA (1) ZA9610405B (OSRAM)

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CZ293062B6 (cs) * 1997-09-25 2004-01-14 Bayer Aktiengesellschaft Léčivo s regulovaným uvolněním aktivní sloučeniny
DE19751948A1 (de) 1997-11-24 1999-05-27 Bayer Ag Verfahren zur Herstellung von 8-Methoxy-Chinoloncarbonsäuren
US6509327B1 (en) 1998-09-30 2003-01-21 Alcon Manufacturing, Ltd. Compositions and methods for treating otic, ophthalmic and nasal infections
US6395746B1 (en) 1998-09-30 2002-05-28 Alcon Manufacturing, Ltd. Methods of treating ophthalmic, otic and nasal infections and attendant inflammation
US6716830B2 (en) 1998-09-30 2004-04-06 Alcon, Inc. Ophthalmic antibiotic compositions containing moxifloxacin
CA2349161C (en) * 1998-11-10 2008-01-29 Bayer Aktiengesellschaft Pharmaceutical moxifloxacin preparation
DE19854357A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Semi-Hydrochlorid von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo/4.3.0/ -nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854356A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation A von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo-/4.3.0/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854355A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation B von 8-Cyan-1-cyclopropyl-7-(1S, 6S-2,8-diazabicyclo-/4.3.O/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19908449A1 (de) * 1999-02-26 2000-08-31 Bayer Ag Kristallmodifikation C von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicylo-[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chino/incarbonsäure
EP1562942A1 (en) * 2002-10-31 2005-08-17 Ranbaxy Laboratories, Ltd. Amorphous moxifloxacin hydrochloride
CA2521398C (en) 2003-04-09 2011-03-22 Dr. Reddy's Laboratories Limited A crystalline form iii of anhydrous moxifloxacin hydrochloride and a process for preparation thereof
WO2005012285A1 (en) * 2003-08-05 2005-02-10 Matrix Laboratories Ltd An improved process for the preparation of moxifloxacin hydrochloride
ES2319125T3 (es) * 2003-11-20 2009-05-04 Chemi S.P.A. Polimorfos del clorhidrato del acido 1-ciclopropil-7-((s,s)-2,8-diazadiciclo(4.3.0)-non-8-il)-6-fluoro-1,4-dihidro-8-metoxi-4-oxo-3-quinolina carboxilico y metodos para la preparacion de los mismos.
ITMI20032259A1 (it) 2003-11-20 2005-05-21 Chemi Spa Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione
US7491725B2 (en) 2004-02-06 2009-02-17 Bristol-Myers Squibb Company Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
DE102004015981A1 (de) * 2004-04-01 2005-10-20 Bayer Healthcare Ag Neue kirstalline Form von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE102004063347A1 (de) * 2004-12-23 2006-07-13 Stada Arzneimittel Ag Gebrauchsfertige Gemcitabinlösungen und Gemcitabinlösungskonzentrate
WO2007033515A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation orale contenant de la moxifloxacine et son procédé de préparation
GB0612422D0 (en) * 2006-06-23 2006-08-02 Generics Uk Ltd Novel hydrate form
DE602007003024D1 (de) 2006-06-27 2009-12-10 Sandoz Ag Neues verfahren zur salzherstellung
ES2303768B1 (es) * 2006-09-08 2009-06-05 Quimica Sintetica, S.A. Nueva forma cristalina de moxifloxacino clorhidrato.
IN2014MN02582A (OSRAM) 2006-11-13 2015-09-11 Cipla Ltd
EP1992626A1 (en) * 2007-05-10 2008-11-19 Sandoz AG Process for the preparation of moxifloxacin hydrochloride
EP2083010A1 (en) * 2008-01-08 2009-07-29 Chemo Ibérica, S.A. Polymorphic Forms of Moxifloxacin hydrochloride and processes for preparation thereof
EP2154137A1 (en) 2008-08-04 2010-02-17 Chemo Ibérica, S.A. Crystalline form of moxifloxacin base
PL2349220T3 (pl) 2008-10-09 2012-12-31 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi Zastosowanie rozpuszczalników organicznych w granulacji na mokro moksyfloksacyny
WO2010052726A1 (en) * 2008-11-06 2010-05-14 Hetero Research Foundation Novel polymorph of moxifloxacin hydrochloride
PL2364141T5 (pl) 2008-12-08 2018-02-28 Ratiopharm Gmbh Kompaktorowana moksyfloksacyna
NZ610978A (en) 2009-05-15 2014-11-28 Redx Pharma Ltd Redox drug derivatives
WO2011121596A2 (en) * 2010-04-01 2011-10-06 Neuland Laboratories Ltd. Crystal modification of moxifloxacin hydrochloride
BRPI1106900A2 (pt) 2011-12-26 2013-11-05 Ems Sa Composição farmacêutica sólida compreendendo antibótico da familia das quinolonas e processo de sua obtenção
FR2992218B1 (fr) 2012-06-22 2015-01-23 Rivopharm Sa Composition pharmaceutique de chlorhydrate de moxifloxacine et procede de preparation
CN102924449B (zh) * 2012-10-30 2015-08-12 重庆福安药业集团庆余堂制药有限公司 盐酸莫西沙星h晶型及其制备方法和药物组合物
US9388178B2 (en) 2012-12-04 2016-07-12 Mankind Research Centre Process for the preparation of moxifloxacin hydrochloride
RU2561037C2 (ru) * 2013-02-07 2015-08-20 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Антибактериальная фармацевтическая композиция и способ ее получения
HK1219690A1 (zh) 2013-03-15 2017-04-13 Melinta Subsidiary Corp. 利用抗生素来治疗超重和肥胖患者感染的方法

Family Cites Families (11)

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Publication number Priority date Publication date Assignee Title
DE3601567A1 (de) * 1986-01-21 1987-07-23 Bayer Ag 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
CN1019114B (zh) * 1986-03-31 1992-11-18 三共株式会社 喹啉-3-羟酸衍生物的制备方法
AU609974B2 (en) * 1988-05-18 1991-05-09 Warner-Lambert Company Improved process for the preparation of 5-amino-7- (substituted amino)-quinoline-3-carboxylic acids
DE3910663A1 (de) * 1989-04-03 1990-10-04 Bayer Ag 5-alkylchinoloncarbonsaeuren
RO108347B1 (ro) * 1989-10-30 1994-04-28 Bellon Labor Sa Roger DERIVATI DE BENZO-(b)-NAFTIRIDIN-1,8 SI PROCEDEU DE PREPARARE A ACESTORA
TW209865B (OSRAM) 1992-01-10 1993-07-21 Bayer Ag
DE69331003T2 (de) * 1992-01-31 2002-06-20 Chugai Seiyaku K.K., Tokio/Tokyo Kristalle von derivaten von chinozon carbonsäure-hydraten
DE4234078A1 (de) 1992-10-09 1994-04-14 Bayer Ag Chinoloncarbonsäuren
JP3268098B2 (ja) * 1992-12-25 2002-03-25 第一製薬株式会社 二環性環状アミン誘導体
ZA946853B (en) * 1993-09-10 1995-04-24 Daiichi Seiyaku Co Crystals of antimicrobial compound.
EP0676199B1 (en) * 1994-04-07 1998-09-02 Pfizer Inc. Use of trovafloxacin or derivatives thereof for the manufacture of a medicament for the treatment of H. pylori infections

Also Published As

Publication number Publication date
JPH09169757A (ja) 1997-06-30
CA2192418C (en) 2001-06-12
CZ288657B6 (cs) 2001-08-15
ATE221531T1 (de) 2002-08-15
PL317415A1 (en) 1997-06-23
US5849752A (en) 1998-12-15
CA2192418A1 (en) 1997-06-13
DE59609501D1 (de) 2002-09-05
EP0780390B1 (de) 2002-07-31
UA35638C2 (uk) 2001-04-16
CO4480105A1 (es) 1997-07-09
AU708006B2 (en) 1999-07-29
BG62258B1 (bg) 1999-06-30
HU226521B1 (en) 2009-03-30
DK0780390T3 (da) 2002-11-11
NZ299905A (en) 1998-09-24
PT780390E (pt) 2002-11-29
HU9603428D0 (en) 1997-01-28
MY117492A (en) 2004-07-31
RU2162468C2 (ru) 2001-01-27
EE9600201A (et) 1997-06-16
IL119795A0 (en) 1997-03-18
CU22774A3 (es) 2002-07-24
IN185805B (OSRAM) 2001-05-05
HRP960558A2 (en) 1998-02-28
TW411340B (en) 2000-11-11
NO965298L (no) 1997-06-13
JP4104687B2 (ja) 2008-06-18
IL119795A (en) 1998-12-27
EE03474B1 (et) 2001-08-15
ZA9610405B (en) 1997-06-23
YU65096A (sh) 1998-12-23
RO119782B1 (ro) 2005-03-30
KR970042550A (ko) 1997-07-24
YU49485B (sh) 2006-08-17
SK159196A3 (en) 1997-10-08
MX9606325A (es) 1997-10-31
SI0780390T1 (en) 2002-10-31
HUP9603428A3 (en) 1997-10-28
DE19546249A1 (de) 1997-06-19
AU7421696A (en) 1997-06-19
NL300109I1 (nl) 2003-02-03
BR9605968A (pt) 1998-08-18
BG101043A (en) 1998-04-30
NO306725B1 (no) 1999-12-13
SA96170492B1 (ar) 2006-05-23
SV1996000109A (es) 1997-10-23
CZ364696A3 (en) 1997-07-16
HRP960558B1 (en) 2002-04-30
AR005009A1 (es) 1999-04-07
EP0780390A1 (de) 1997-06-25
NO965298D0 (no) 1996-12-11
SK282805B6 (sk) 2002-12-03
KR100525146B1 (ko) 2006-01-27
ES2179910T3 (es) 2003-02-01
CN1160052A (zh) 1997-09-24
MA24342A1 (fr) 1998-07-01
TR199600970A2 (tr) 1997-06-21
SG47201A1 (en) 1998-03-20
PL184885B1 (pl) 2003-01-31
CN1061348C (zh) 2001-01-31
HUP9603428A2 (en) 1997-08-28

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