UY35831A - ?proceso para fluorar compuestos?. - Google Patents

?proceso para fluorar compuestos?.

Info

Publication number
UY35831A
UY35831A UY0001035831A UY35831A UY35831A UY 35831 A UY35831 A UY 35831A UY 0001035831 A UY0001035831 A UY 0001035831A UY 35831 A UY35831 A UY 35831A UY 35831 A UY35831 A UY 35831A
Authority
UY
Uruguay
Prior art keywords
fluorate
compounds
substrate
fluorinated
sulfonyl
Prior art date
Application number
UY0001035831A
Other languages
English (en)
Inventor
Allen Laura
Sanford Melanie
Shin Hee Lee
Bland Douglas
Cheng Yeng
Roth Gary
Muhuhi Joseck
Original Assignee
Dow Agrosciences Llc
Univ Michigan
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow Agrosciences Llc, Univ Michigan filed Critical Dow Agrosciences Llc
Publication of UY35831A publication Critical patent/UY35831A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C07D213/803—Processes of preparation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/06—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
    • C07D213/127—Preparation from compounds containing pyridine rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Se describen métodos de preparación de un sustrato fluorado mediante la combinación de fluoruro de potasio, una sal de amonio cuaternario y un sustrato sustituido con al menos un grupo de cloro, bromo, sulfonilo o nitro, para proveer de ese modo el sustrato fluorado.
UY0001035831A 2013-11-12 2014-11-12 ?proceso para fluorar compuestos?. UY35831A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201361902989P 2013-11-12 2013-11-12

Publications (1)

Publication Number Publication Date
UY35831A true UY35831A (es) 2015-06-30

Family

ID=51999557

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001035831A UY35831A (es) 2013-11-12 2014-11-12 ?proceso para fluorar compuestos?.

Country Status (14)

Country Link
US (1) US9493415B2 (es)
EP (1) EP3068764B1 (es)
JP (1) JP6563391B2 (es)
CN (1) CN105899488B (es)
AR (1) AR098398A1 (es)
BR (1) BR102014028162A2 (es)
CA (1) CA2929940A1 (es)
ES (1) ES2720234T3 (es)
HU (1) HUE043300T2 (es)
IL (1) IL245542B (es)
PL (1) PL3068764T3 (es)
TW (1) TW201609652A (es)
UY (1) UY35831A (es)
WO (1) WO2015073525A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201524956A (zh) * 2013-11-12 2015-07-01 Dow Agrosciences Llc 用於氟化化合物之過程（二）
TW201609651A (zh) 2013-11-12 2016-03-16 陶氏農業科學公司 用於氟化化合物之過程（一）
TWI726900B (zh) 2015-08-04 2021-05-11 美商陶氏農業科學公司 用於氟化化合物之過程

Family Cites Families (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1292746C (en) 1983-12-23 1991-12-03 Charles A. Wilson Preparation of difluoropyridine compounds
GB8504268D0 (en) * 1985-02-19 1985-03-20 Shell Int Research Preparation of fluorinated pyridines
DE3827436A1 (de) * 1988-08-12 1990-02-15 Bayer Ag Verfahren zum einfuehren von fluoratomen an aromatische kerne durch nucleophilen austausch
EP0523671B1 (de) * 1991-07-17 1996-01-17 Hoechst Aktiengesellschaft Verfahren zur Herstellung von Chlorfluornitrobenzolen
BR9612862B8 (pt) * 1995-09-22 2014-08-05 Wakunaga Pharma Co Ltd Derivado de ácido piridono carboxílico e agentes antibacteriais.
DE19817264A1 (de) * 1998-04-18 1999-10-21 Bayer Ag Neue Dihydropyrimidine
CA2445459A1 (fr) 2001-05-17 2002-11-21 Maxime Garayt Utilisation d'une composition de nature ionique comme reactif de substitution, composition constituant un reactif de fluoration et procede l'utilisant
CN1357530A (zh) * 2001-07-23 2002-07-10 昆山双鹤药业有限责任公司 用邻氯硝基苯制备2,3,4－三氟硝基苯的生产工艺
KR100441153B1 (ko) 2002-03-14 2004-07-21 주식회사 씨트리 유기 불소화합물의 제조방법
DE10227223A1 (de) 2002-06-18 2004-01-08 Kühlein, Klaus, Prof.Dr. Verfahren zur Herstellung substituierter organischer Verbindungen und Verwendung von Katalysatoren für Substitutionsreaktionen
JP2006515601A (ja) 2002-11-28 2006-06-01 アストラゼネカ アクチボラグ 抗細菌性薬剤としてのオキサゾリジノン
WO2005063661A1 (ja) 2003-12-25 2005-07-14 Sumitomo Chemical Company, Limited フッ素化剤およびそれを用いる含フッ素化合物の製造方法
DE102004033525A1 (de) 2004-07-08 2006-02-02 Lanxess Deutschland Gmbh Verbessertes Verfahren zur Herstellung kernfluorierter Aromaten
US7592486B2 (en) 2004-09-16 2009-09-22 Board Of Regents Of The University Of Nebraska Anhydrous fluoride salts and reagents and methods for their production
BRPI0517854A (pt) 2004-11-17 2008-10-21 Minrad Inc processo para a preparação de um composto, mistura de produtos, e, sevoflurano
CN100344605C (zh) * 2006-06-30 2007-10-24 上海万溯化学有限公司 一种3－氟－5－硝基三氟甲苯的制备方法
AR068509A1 (es) * 2007-09-19 2009-11-18 Jerini Ag Antagosnistas del receptor de bradiquinina b1
CN101591211B (zh) * 2008-05-30 2012-10-03 南京理工大学 微波卤素交换氟化制备氟代化合物的方法
CN101519373B (zh) * 2008-12-30 2011-10-05 凯莱英医药化学（天津）有限公司 一种2,6-二氟吡啶的合成方法
CN101602712B (zh) * 2009-07-21 2011-04-06 南京第一农药集团有限公司 一种合成2-氟-3-氯-5-三氟甲基吡啶的方法
CN101648904B (zh) * 2009-09-14 2011-08-03 南京第一农药集团有限公司 一种2,3-二氟-5-氯吡啶的合成方法
CN101671217A (zh) * 2009-09-28 2010-03-17 南京第一农药集团有限公司 由有机多氯化合物制备有机氟氯化合物的方法
CN102531962A (zh) * 2010-12-30 2012-07-04 上海恩氟佳科技有限公司 2-氟-5-氯苯腈的制备方法
TWI537252B (zh) 2011-01-25 2016-06-11 陶氏農業科學公司 用於製備４－胺基－５－氟－３－鹵素－６－（經取代之）吡啶甲酸酯的方法（一）
TWI529163B (zh) * 2011-01-25 2016-04-11 陶氏農業科學公司 用於製備４－胺基－５－氟－３－鹵素－６－（經取代之）吡啶甲酸酯的方法
TWI592401B (zh) 2011-01-25 2017-07-21 陶氏農業科學公司 用於製備４－胺基－３－氯－５－氟－６－（經取代的）吡啶甲酸酯的方法（一）
TWI547482B (zh) 2011-01-25 2016-09-01 陶氏農業科學公司 增加可回收之3-氯-4,5,6-三氟-2-氰吡啶之量的改良方法
FR2975990B1 (fr) 2011-06-01 2013-05-24 Rhodia Operations Procede de preparation d'un compose organique fluore
CN102617360B (zh) * 2012-03-01 2013-11-06 江西吉翔医药化工有限公司 3,5-二氯-2,4-二氟苯胺的合成方法
AR092355A1 (es) 2012-07-24 2015-04-15 Dow Agrosciences Llc Fluoruros de fluoropicolinoilo y procesos para su preparacion
AR091856A1 (es) 2012-07-24 2015-03-04 Dow Agrosciences Llc Proceso para la preparacion de 4-amino-5-fluor-3-halo-6-(substituido) picolinatos
CN103012279B (zh) * 2012-11-27 2015-01-28 浙江工业大学 一种4,5,6-三氟嘧啶化合物的制备方法
WO2014093591A1 (en) 2012-12-13 2014-06-19 Dow Agrosciences Llc Processes for the preparation of 4-amino-3-halo-6- (substituted)picolinates and 4-amino-5-fluoro-3-halo-6- (substituted)picolinates
US9260392B2 (en) 2012-12-13 2016-02-16 Dow Agrosciences Llc Process for the preparation of 4-Amino-5-fluoro-3-chloro-6-(substituted)picolinates
PL2931043T3 (pl) 2012-12-13 2018-01-31 Dow Agrosciences Llc Sposób wytwarzania 4-amino-5-fluoro-3-chloro 6-(podstawionych) pikolinianów
TW201524956A (zh) 2013-11-12 2015-07-01 Dow Agrosciences Llc 用於氟化化合物之過程（二）
TW201609651A (zh) 2013-11-12 2016-03-16 陶氏農業科學公司 用於氟化化合物之過程（一）

Also Published As

Publication number Publication date
CN105899488B (zh) 2019-09-03
PL3068764T3 (pl) 2019-08-30
HUE043300T2 (hu) 2019-08-28
EP3068764B1 (en) 2019-02-20
US9493415B2 (en) 2016-11-15
CN105899488A (zh) 2016-08-24
ES2720234T3 (es) 2019-07-18
IL245542A0 (en) 2016-06-30
JP6563391B2 (ja) 2019-08-21
US20150141654A1 (en) 2015-05-21
JP2016538278A (ja) 2016-12-08
TW201609652A (zh) 2016-03-16
BR102014028162A2 (pt) 2015-09-08
AR098398A1 (es) 2016-05-26
IL245542B (en) 2019-01-31
CA2929940A1 (en) 2015-05-21
EP3068764A1 (en) 2016-09-21
WO2015073525A1 (en) 2015-05-21

Similar Documents

Publication Publication Date Title
EA201891360A1 (ru) Тройной агонист рецепторов глюкагона/glp-1/gip
CU20200004A7 (es) Compuestos para tratar afecciones asociadas con la actividad nlrp
SV2018005684A (es) Anticuerpos que se unen especificamente a pd-1 y sus usos
EA201891211A1 (ru) Ингибиторы cxcr2
DK2970283T3 (da) Substituerede 2-aza-bicyclo[2.2.1]heptan-3-carboxylsyre-(benzyl-cyano-methyl)-amider som inhibitorer af cathepsin-c
EA201692219A1 (ru) Способы получения противовирусных соединений
PE20190734A1 (es) Composiciones de colector y metodos de uso de las mismas
AR096344A1 (es) Compuestos de elastómeros, mezclas y métodos para preparar los mismos
BR112016007581A2 (pt) pigmentos à base de compostos de bismuto
DK3279202T3 (da) Krystal af 3,5-disubstitueret benzenalkynylforbindelse
CL2017002427A1 (es) Producción de ácido ribonucleico libre de células.
BR112016018358A2 (pt) Composição reativa, e, processo
BR112017008154A2 (pt) construção de gerenciamento de luz
CL2016001095A1 (es) Silicato de zirconio microporoso para el tratamiento de hipercalemia.
PE20170329A1 (es) Polipeptidos que tienen actividad xilanasa con una tasa de conversion alta de polisacaridos que contienen xilosa
PH12018500903A1 (en) Pyranodipyridine compound
AR105812A1 (es) Métodos para la preparación de inhibidores de proteína deacetilasa
CL2017002255A1 (es) Procesos para preparar fluorocetólidos.
UY35831A (es) ?proceso para fluorar compuestos?.
UY35832A (es) ?proceso para fluorar compuestos?
BR112016027455A2 (pt) moduladores ppar
BR112015020373A2 (pt) processo para produção de um poliuretano, poliuretano e uso de um poliuretano.
CL2018000962A1 (es) Oportunidades para el proceso de aumento de recuperación según se aplica a la producción de molibdeno
ITUB20152959A1 (it) Sali di composti a struttura benzimidazolica, loro usi e procedimento di preparazione.
UY35833A (es) ?proceso de fluoración de compuestos?

Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20211215