UY30170A1 - Proceso para la preparacion de compuestos de dibenzotiazepina - Google Patents

Proceso para la preparacion de compuestos de dibenzotiazepina

Info

Publication number
UY30170A1
UY30170A1 UY30170A UY30170A UY30170A1 UY 30170 A1 UY30170 A1 UY 30170A1 UY 30170 A UY30170 A UY 30170A UY 30170 A UY30170 A UY 30170A UY 30170 A1 UY30170 A1 UY 30170A1
Authority
UY
Uruguay
Prior art keywords
compound
carboxy
diphenylsulfide
dibenzotiazepine
compounds
Prior art date
Application number
UY30170A
Other languages
English (en)
Inventor
Kiyotaka Yoshh
Shigeyoshi Nishino
Katsumasa Harada
Debra Ainge
Luis-Manuel Vaz
Paul Michael Murray
Original Assignee
Ube Industries
Astrazeneca Uk Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ube Industries, Astrazeneca Uk Ltd filed Critical Ube Industries
Publication of UY30170A1 publication Critical patent/UY30170A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/18—Eight-membered rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C319/00—Preparation of thiols, sulfides, hydropolysulfides or polysulfides
    • C07C319/14—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides
    • C07C319/18—Preparation of thiols, sulfides, hydropolysulfides or polysulfides of sulfides by addition of thiols to unsaturated compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with two six-membered rings
    • C07D281/16—[b, f]-condensed

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)

Abstract

Un compuesto de di-benzotiazepina se prepara apropiadamente sometiendo un compuesto de 2-amino-2`-carboxi-difenilsufuroide a reaccinn de deshidratacinn. condensacinn en la presencia de un catalizador rcido; el compuesto de 2-amino-2`- carboxi-difenilsulfuro se prepara aproximadamente reduciendo el compuesto de 2-nitro-2`carboxi-difenilsulfuro en un solvente mas bajo de cster alifrtico; y el compuesto de 2-nitro-2`carboxi-difenilsulfuro se prepara apropiadamente reaccionando un compuesto de nitrobenceno con un compuesto de rcido tiosalicelico en una mezcla de un alcohol alifrtico inferior y agua.
UY30170A 2006-02-22 2007-02-21 Proceso para la preparacion de compuestos de dibenzotiazepina UY30170A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US77548306P 2006-02-22 2006-02-22

Publications (1)

Publication Number Publication Date
UY30170A1 true UY30170A1 (es) 2007-09-28

Family

ID=38220043

Family Applications (1)

Application Number Title Priority Date Filing Date
UY30170A UY30170A1 (es) 2006-02-22 2007-02-21 Proceso para la preparacion de compuestos de dibenzotiazepina

Country Status (17)

Country Link
US (1) US7671195B2 (es)
EP (1) EP1996568A2 (es)
JP (1) JP2009527458A (es)
KR (1) KR20080108468A (es)
CN (1) CN101389615A (es)
AR (1) AR059613A1 (es)
AU (1) AU2007223597A1 (es)
BR (1) BRPI0708096A2 (es)
CA (1) CA2642659A1 (es)
EC (1) ECSP088679A (es)
IL (1) IL193264A0 (es)
NO (1) NO20083544L (es)
RU (1) RU2008137615A (es)
TW (1) TW200811119A (es)
UY (1) UY30170A1 (es)
WO (1) WO2007102352A2 (es)
ZA (1) ZA200806903B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20030216376A1 (en) * 2002-03-20 2003-11-20 Revital Lifshitz-Liron Crystalline forms of quetiapine hemifumarate
WO2006113425A1 (en) * 2005-04-14 2006-10-26 Teva Pharmaceutical Industries Ltd. Process for preparing quetiapine fumarate
EP2144892A2 (en) * 2007-03-29 2010-01-20 Teva Pharmaceutical Industries Ltd. Improved process for preparing quetiapine fumarate
CN104177311B (zh) * 2013-05-27 2016-09-14 许昌恒生制药有限公司 一种喹硫平中间体的制备方法
CN103772319A (zh) * 2014-01-02 2014-05-07 成都医路康医学技术服务有限公司 一种硫氮杂卓类化合物的合成方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL201699B1 (pl) * 1999-07-09 2009-04-30 Astrazeneca Uk Ltd Sposób wytwarzania pochodnej dibenzotiazepiny
KR100707050B1 (ko) * 2002-11-28 2007-04-13 에스케이 주식회사 10Ｈ-디벤조[ｂ,ｆ][1,4]티아제핀-11-온의 제조방법
PL195728B1 (pl) * 2003-07-18 2007-10-31 Helm Ag Sposób wytwarzania 11-(1-piperazynylo)dibenzo[b,f][1,4]tiazepiny
EP1682537B1 (en) * 2003-11-05 2012-03-28 SARcode Bioscience Inc. Modulators of cellular adhesion

Also Published As

Publication number Publication date
AR059613A1 (es) 2008-04-16
AU2007223597A8 (en) 2008-09-11
WO2007102352A2 (en) 2007-09-13
JP2009527458A (ja) 2009-07-30
KR20080108468A (ko) 2008-12-15
EP1996568A2 (en) 2008-12-03
TW200811119A (en) 2008-03-01
CN101389615A (zh) 2009-03-18
BRPI0708096A2 (pt) 2011-05-17
RU2008137615A (ru) 2010-03-27
US20070203336A1 (en) 2007-08-30
US7671195B2 (en) 2010-03-02
ECSP088679A (es) 2008-09-29
WO2007102352A3 (en) 2008-01-10
IL193264A0 (en) 2009-02-11
CA2642659A1 (en) 2007-09-13
AU2007223597A1 (en) 2007-09-13
NO20083544L (no) 2008-09-16
ZA200806903B (en) 2010-10-27

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20170526