UA86731C2 - Делимая галеновая форма модифицированного высвобождения активного ингредиента - Google Patents

Делимая галеновая форма модифицированного высвобождения активного ингредиента

Info

Publication number
UA86731C2
UA86731C2 UAA200810556A UAA200810556A UA86731C2 UA 86731 C2 UA86731 C2 UA 86731C2 UA A200810556 A UAA200810556 A UA A200810556A UA A200810556 A UAA200810556 A UA A200810556A UA 86731 C2 UA86731 C2 UA 86731C2
Authority
UA
Ukraine
Prior art keywords
divisible
drug release
galenic form
modified drug
galenic
Prior art date
Application number
UAA200810556A
Other languages
English (en)
Ukrainian (uk)
Inventor
Жиль Фонкнехтен
Патрик Женти
Жан-Манюель Пен
Патрик Вютриш
Original Assignee
Ле Лаборатуар Сервье
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39796790&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA86731(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ле Лаборатуар Сервье filed Critical Ле Лаборатуар Сервье
Publication of UA86731C2 publication Critical patent/UA86731C2/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/403Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/64Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Inorganic Chemistry (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)

Abstract

Изобретение относится к делимой галеновой форме модифицированного высвобождения активного ингредиента, где неразделенная галеновая форма и часть указанной формы, которую получают разделением, имеют одинаковые параметры растворения.
UAA200810556A 2008-03-21 2008-08-20 Делимая галеновая форма модифицированного высвобождения активного ингредиента UA86731C2 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0801561A FR2928836B1 (fr) 2008-03-21 2008-03-21 Forme galenique secable permettant une liberation modifiee du principe actif

Publications (1)

Publication Number Publication Date
UA86731C2 true UA86731C2 (ru) 2009-05-12

Family

ID=39796790

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200810556A UA86731C2 (ru) 2008-03-21 2008-08-20 Делимая галеновая форма модифицированного высвобождения активного ингредиента

Country Status (37)

Country Link
US (3) US20090238870A1 (ru)
EP (2) EP2103302A1 (ru)
JP (2) JP5231906B2 (ru)
KR (3) KR20090101048A (ru)
CN (1) CN101347414B (ru)
AP (1) AP2729A (ru)
AR (1) AR067993A1 (ru)
AU (1) AU2008207680B8 (ru)
BR (1) BRPI0803631A2 (ru)
CA (1) CA2629670C (ru)
CL (1) CL2008002486A1 (ru)
CO (1) CO6020017A1 (ru)
CR (2) CR10317A (ru)
CU (1) CU23970B1 (ru)
EA (1) EA200801862A1 (ru)
EC (1) ECSP088727A (ru)
FR (1) FR2928836B1 (ru)
GT (1) GT200800163A (ru)
HK (1) HK1127280A1 (ru)
HN (1) HN2008001466A (ru)
IL (1) IL193611A0 (ru)
JO (1) JO3052B1 (ru)
MA (1) MA31218B1 (ru)
ME (1) ME01031B (ru)
MX (1) MX2008011579A (ru)
MY (1) MY150660A (ru)
NI (1) NI200800256A (ru)
NZ (1) NZ570715A (ru)
PE (1) PE20090991A1 (ru)
SA (1) SA08290555B1 (ru)
SG (1) SG155819A1 (ru)
SV (1) SV2008003023A (ru)
TW (1) TWI396561B (ru)
UA (1) UA86731C2 (ru)
UY (1) UY31307A1 (ru)
WO (1) WO2009125087A1 (ru)
ZA (1) ZA200807354B (ru)

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DK1940467T3 (da) 2005-09-09 2017-02-13 Paladin Labs Inc Lægemiddelsammensætning med langvarig frigivelse
US20070160960A1 (en) * 2005-10-21 2007-07-12 Laser Shot, Inc. System and method for calculating a projectile impact coordinates
WO2011107494A1 (de) 2010-03-03 2011-09-09 Sanofi Neue aromatische glykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung
DE102010015123A1 (de) 2010-04-16 2011-10-20 Sanofi-Aventis Deutschland Gmbh Benzylamidische Diphenylazetidinone, diese Verbindungen enthaltende Arzneimittel und deren Verwendung
US8530413B2 (en) 2010-06-21 2013-09-10 Sanofi Heterocyclically substituted methoxyphenyl derivatives with an oxo group, processes for preparation thereof and use thereof as medicaments
TW201221505A (en) 2010-07-05 2012-06-01 Sanofi Sa Aryloxyalkylene-substituted hydroxyphenylhexynoic acids, process for preparation thereof and use thereof as a medicament
TW201215387A (en) 2010-07-05 2012-04-16 Sanofi Aventis Spirocyclically substituted 1,3-propane dioxide derivatives, processes for preparation thereof and use thereof as a medicament
TW201215388A (en) 2010-07-05 2012-04-16 Sanofi Sa (2-aryloxyacetylamino)phenylpropionic acid derivatives, processes for preparation thereof and use thereof as medicaments
TR201103946A1 (tr) 2011-04-22 2012-11-21 Sanovel İlaç Sanayi̇ Ve Ti̇caret Anoni̇m Şi̇rketi̇ Kontrollü salım sağlayan gliklazid formülasyonları.
WO2013037390A1 (en) 2011-09-12 2013-03-21 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2567959B1 (en) 2011-09-12 2014-04-16 Sanofi 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
EP2760862B1 (en) 2011-09-27 2015-10-21 Sanofi 6-(4-hydroxy-phenyl)-3-alkyl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors
ITFI20130184A1 (it) 2013-08-01 2015-02-02 Valpharma Internat S P A Una formulazione farmaceutica di gliclazide a rilascio modificato, somministrabile per via orale, e suo metodo di produzione.
CN106892856A (zh) * 2017-02-06 2017-06-27 山东科源制药股份有限公司 一种格列齐特粗品重结晶的制备方法
EP4121013A1 (en) 2020-03-16 2023-01-25 Grünenthal GmbH Scored tablet

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CH648754A5 (en) * 1979-08-16 1985-04-15 Ciba Geigy Ag Pharmaceutical slow release tablet
US4851230A (en) * 1983-04-07 1989-07-25 Bristol-Myers Company Capsule shaped tablets
GB8724763D0 (en) * 1987-10-22 1987-11-25 Aps Research Ltd Sustained-release formulations
US5126145A (en) * 1989-04-13 1992-06-30 Upsher Smith Laboratories Inc Controlled release tablet containing water soluble medicament
JPH069375A (ja) * 1992-04-10 1994-01-18 Takeda Chem Ind Ltd 分割可能な連結錠剤
DE4229085C2 (de) * 1992-09-01 1996-07-11 Boehringer Mannheim Gmbh Längliche, teilbare Tablette
US5859037A (en) * 1997-02-19 1999-01-12 Warner-Lambert Company Sulfonylurea-glitazone combinations for diabetes
ES2216335T3 (es) * 1997-12-08 2004-10-16 Bristol-Myers Squibb Company Nuevas sales de metformina y procedimiento.
AP1224A (en) * 1998-03-19 2003-11-14 Bristol Myers Squibb Co Biphasic controlled release delivery system for high solubility pharmaceuticals and method.
JP2006052230A (ja) * 1998-04-03 2006-02-23 Kyowa Hakko Kogyo Co Ltd 分割錠剤及びプレススルーパック
WO1999051207A1 (fr) * 1998-04-03 1999-10-14 Kyowa Hakko Kogyo Co., Ltd. Comprime secable et conditionnement au travers duquel appliquer une force de pression
AP1243A (en) * 1999-02-01 2004-02-02 Servier Lab Core tablet for controlled release of gliclazide after oral administration.
CZ300551B6 (cs) * 1999-03-31 2009-06-17 Janssen Pharmaceutica N. V. Predželatinovaný škrob v rízene se uvolnující formulaci
US6878749B2 (en) * 1999-09-17 2005-04-12 Novartis Ag Method of treating metabolic disorders, especially diabetes, or a disease or condition associated with diabetes
DE10117208A1 (de) * 2001-04-06 2002-10-10 Wolff Walsrode Ag Verfahren zur Herstellung von niederviskosen, wässrigen Celluloseetherlösungen
CN1294908C (zh) * 2003-06-08 2007-01-17 安徽省医药科技实业公司 口服格列齐特缓释制剂
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DK1940467T3 (da) * 2005-09-09 2017-02-13 Paladin Labs Inc Lægemiddelsammensætning med langvarig frigivelse
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Also Published As

Publication number Publication date
NI200800256A (es) 2010-02-11
JP2009227651A (ja) 2009-10-08
AR067993A1 (es) 2009-10-28
AU2008207680A1 (en) 2009-10-08
CN101347414A (zh) 2009-01-21
CU23970B1 (es) 2013-12-27
EP2103302A1 (fr) 2009-09-23
CA2629670A1 (fr) 2008-10-01
JP5231906B2 (ja) 2013-07-10
MY150660A (en) 2014-02-14
EA200801862A1 (ru) 2009-10-30
UY31307A1 (es) 2008-10-31
KR20110112266A (ko) 2011-10-12
SG155819A1 (en) 2009-10-29
JO3052B1 (ar) 2017-03-15
BRPI0803631A2 (pt) 2011-03-29
HK1127280A1 (en) 2009-09-25
US20140221449A1 (en) 2014-08-07
US20130295176A1 (en) 2013-11-07
IL193611A0 (en) 2009-08-03
MA31218B1 (fr) 2010-03-01
FR2928836A1 (fr) 2009-09-25
SV2008003023A (es) 2010-07-29
CO6020017A1 (es) 2009-03-31
FR2928836B1 (fr) 2011-08-26
US20090238870A1 (en) 2009-09-24
GT200800163A (es) 2010-05-21
CU20080179A7 (es) 2011-04-26
CL2008002486A1 (es) 2008-12-26
MX2008011579A (es) 2009-09-21
ECSP088727A (es) 2008-10-31
CN101347414B (zh) 2011-11-23
AP2729A (en) 2013-08-31
NZ570715A (en) 2010-10-29
AU2008207680B8 (en) 2010-05-13
CA2629670C (fr) 2012-04-17
JP2010209103A (ja) 2010-09-24
AP2008004614A0 (en) 2008-10-31
SA08290555B1 (ar) 2011-07-20
TW200940109A (en) 2009-10-01
CR20140334A (es) 2014-08-20
KR20150035829A (ko) 2015-04-07
ZA200807354B (en) 2008-11-26
KR20090101048A (ko) 2009-09-24
CR10317A (es) 2008-11-26
HN2008001466A (es) 2011-04-25
KR101693189B1 (ko) 2017-01-05
ME01031B (me) 2012-10-20
AU2008207680B2 (en) 2010-04-22
TWI396561B (zh) 2013-05-21
PE20090991A1 (es) 2009-07-18
WO2009125087A1 (fr) 2009-10-15
EP3025706A1 (fr) 2016-06-01

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