UA83509C2 - Imidazopyrazines as tyrosine kinase inhibitors - Google Patents

Imidazopyrazines as tyrosine kinase inhibitors Download PDF

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Publication number
UA83509C2
UA83509C2 UAA200605222A UAA200605222A UA83509C2 UA 83509 C2 UA83509 C2 UA 83509C2 UA A200605222 A UAA200605222 A UA A200605222A UA A200605222 A UAA200605222 A UA A200605222A UA 83509 C2 UA83509 C2 UA 83509C2
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aai
seiai
web
basei
iaiei
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UAA200605222A
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Патрисия Энн Бек
Кара Сесарио
Хань-Цин Дун
Кеннет Форман
Марк Джозеф Малвихилл
Энтони Инноченцо Найгро
Лидия Сароглоу
Арно Г. Штайниг
Инчуань Суй
Цинхуа Вен
Дуглас Вернер
Робин Уилкес
Джонатан Уилльямс
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Оси Фармасьютикалз, Инк.
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Application filed by Оси Фармасьютикалз, Инк. filed Critical Оси Фармасьютикалз, Инк.
Publication of UA83509C2 publication Critical patent/UA83509C2/uk

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    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
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Abstract

Соединения формулы (І) и их фармацевтически приемлемые соли, где Qи Rимеют значения, указанные здесь, ингибируют фермент IGF-1R и являются пригодными для лечения и/или профилактики разных заболеваний и состояний, которые восприимчивы к лечению ингибированием тирозинкиназы.
UAA200605222A 2003-10-15 2004-10-14 Imidazopyrazines as tyrosine kinase inhibitors UA83509C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US51171203P 2003-10-15 2003-10-15
PCT/US2004/034219 WO2005037836A2 (en) 2003-10-15 2004-10-14 Imidazo ‘1, 5 - a ! pyrazine tyrosine kinase inhibitors

Publications (1)

Publication Number Publication Date
UA83509C2 true UA83509C2 (en) 2008-07-25

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ID=34465267

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Application Number Title Priority Date Filing Date
UAA200605222A UA83509C2 (en) 2003-10-15 2004-10-14 Imidazopyrazines as tyrosine kinase inhibitors

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US (2) US7459554B2 (ru)
EP (1) EP1675860B1 (ru)
JP (1) JP4916883B2 (ru)
KR (1) KR100872204B1 (ru)
CN (1) CN1898240B (ru)
AP (1) AP2006003620A0 (ru)
AR (1) AR046337A1 (ru)
AT (1) ATE525377T1 (ru)
AU (1) AU2004282219C1 (ru)
BR (1) BRPI0415395A (ru)
CA (1) CA2542481A1 (ru)
ES (1) ES2372694T3 (ru)
IL (1) IL174948A0 (ru)
NO (1) NO20062136L (ru)
RU (1) RU2405784C2 (ru)
SG (1) SG132683A1 (ru)
TW (1) TW200530238A (ru)
UA (1) UA83509C2 (ru)
WO (1) WO2005037836A2 (ru)

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