UA78265C2 - Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function - Google Patents

Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function Download PDF

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Publication number
UA78265C2
UA78265C2 UA20040705945A UA20040705945A UA78265C2 UA 78265 C2 UA78265 C2 UA 78265C2 UA 20040705945 A UA20040705945 A UA 20040705945A UA 20040705945 A UA20040705945 A UA 20040705945A UA 78265 C2 UA78265 C2 UA 78265C2
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UA
Ukraine
Prior art keywords
substituted
epoxy
dioxo
dimethyl
octahydro
Prior art date
Application number
UA20040705945A
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English (en)
Ukrainian (uk)
Inventor
Mark E Salvati
James Aaron Balog
Dacia A Pickering
Ramesh N Patel
Ronald L Hanson
James R Corte
Steven H Spergel
Richard A Rampulla
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Bristol Myers Squibb Co
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Publication of UA78265C2 publication Critical patent/UA78265C2/uk

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    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/18—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/18—Bridged systems
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    • A61P5/32—Antioestrogens
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    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones
    • A61P5/46—Drugs for disorders of the endocrine system of the suprarenal hormones for decreasing, blocking or antagonising the activity of glucocorticosteroids
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/08—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
UA20040705945A 2001-12-19 2002-12-18 Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function UA78265C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2511601A 2001-12-19 2001-12-19
PCT/US2002/040598 WO2003062241A1 (en) 2001-12-19 2002-12-18 Fused heterocyclic succinimidecompounds and analogs thereof, modulators of nuclear hormone receptor function

Publications (1)

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UA78265C2 true UA78265C2 (en) 2007-03-15

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JP (1) JP2005523257A (is)
KR (1) KR20040086248A (is)
CN (1) CN1589271A (is)
AR (1) AR037950A1 (is)
AT (1) ATE411319T1 (is)
AU (1) AU2002361785B2 (is)
BR (1) BR0215281A (is)
CA (1) CA2471342A1 (is)
CO (1) CO5640082A2 (is)
DE (1) DE60229435D1 (is)
DK (1) DK1458723T3 (is)
ES (1) ES2314127T3 (is)
GE (1) GEP20063817B (is)
HR (1) HRP20040567A2 (is)
HU (1) HUP0402554A3 (is)
IL (1) IL162547A0 (is)
IS (1) IS7324A (is)
MX (1) MXPA04005876A (is)
NO (1) NO20043068L (is)
NZ (1) NZ533471A (is)
PL (1) PL370904A1 (is)
PT (1) PT1458723E (is)
RU (1) RU2330038C2 (is)
SI (1) SI1458723T1 (is)
TW (1) TWI263640B (is)
UA (1) UA78265C2 (is)
UY (1) UY27595A1 (is)
WO (1) WO2003062241A1 (is)
YU (1) YU53604A (is)
ZA (1) ZA200404812B (is)

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RU2330038C2 (ru) 2008-07-27
MXPA04005876A (es) 2005-05-16
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