UA71059C2 - Спосіб одержання циталопраму - Google Patents

Спосіб одержання циталопраму

Info

Publication number
UA71059C2
UA71059C2 UA2002086988A UA200286988A UA71059C2 UA 71059 C2 UA71059 C2 UA 71059C2 UA 2002086988 A UA2002086988 A UA 2002086988A UA 200286988 A UA200286988 A UA 200286988A UA 71059 C2 UA71059 C2 UA 71059C2
Authority
UA
Ukraine
Prior art keywords
citalopram
preparation
formula
alkylated
aldehyde
Prior art date
Application number
UA2002086988A
Other languages
English (en)
Russian (ru)
Ukrainian (uk)
Inventor
Ханс Петерсен
Майкл Харольд Рок
Original Assignee
Х. Луннбек А/С
X. Луннбек A/C
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8159208&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA71059(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Х. Луннбек А/С, X. Луннбек A/C filed Critical Х. Луннбек А/С
Publication of UA71059C2 publication Critical patent/UA71059C2/uk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87—Benzo [c] furans; Hydrogenated benzo [c] furans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Psychiatry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Furan Compounds (AREA)
UA2002086988A 2000-02-24 2001-02-22 Спосіб одержання циталопраму UA71059C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200000296 2000-02-24
PCT/DK2001/000122 WO2001062754A1 (en) 2000-02-24 2001-02-22 Method for the preparation of citalopram

Publications (1)

Publication Number Publication Date
UA71059C2 true UA71059C2 (uk) 2004-11-15

Family

ID=8159208

Family Applications (1)

Application Number Title Priority Date Filing Date
UA2002086988A UA71059C2 (uk) 2000-02-24 2001-02-22 Спосіб одержання циталопраму

Country Status (29)

Country Link
US (3) US20020004604A1 (enExample)
EP (1) EP1259500A1 (enExample)
JP (1) JP2003524009A (enExample)
KR (1) KR20020080438A (enExample)
CN (1) CN1161350C (enExample)
AU (1) AU2001235357A1 (enExample)
BE (1) BE1012921A6 (enExample)
BG (1) BG107015A (enExample)
BR (1) BR0108947A (enExample)
CA (1) CA2400682A1 (enExample)
EA (1) EA005593B1 (enExample)
FR (1) FR2805813A1 (enExample)
GR (1) GR20010100097A (enExample)
HK (1) HK1054378B (enExample)
HR (1) HRP20020743A2 (enExample)
HU (1) HUP0300078A3 (enExample)
IE (1) IES20010143A2 (enExample)
IL (1) IL151339A0 (enExample)
IS (1) IS6512A (enExample)
IT (1) ITMI20010385A1 (enExample)
MX (1) MXPA02008230A (enExample)
NL (1) NL1017414C1 (enExample)
NO (1) NO20024007L (enExample)
PL (1) PL357178A1 (enExample)
SK (1) SK13662002A3 (enExample)
TR (1) TR200202048T2 (enExample)
UA (1) UA71059C2 (enExample)
WO (1) WO2001062754A1 (enExample)
ZA (2) ZA200206255B (enExample)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR022329A1 (es) 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
PL198024B1 (pl) 1999-04-14 2008-05-30 Lundbeck & Co As H Sposób wytwarzania citalopramu, związki pośrednie i ich zastosowanie do wytwarzania citalopramu
ITMI991581A1 (it) * 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
PT1298124E (pt) 1999-10-25 2007-05-31 Lundbeck & Co As H Método para a preparação de citalopram
US6310222B1 (en) * 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
CN1398263A (zh) 1999-12-28 2003-02-19 H·隆德贝克有限公司 制备西酞普兰的方法
PL198803B1 (pl) 1999-12-30 2008-07-31 Lundbeck & Co As H Sposób wytwarzania 5-cyjano-3H-izobenzofuran-1-onu
EP1254129B1 (en) * 2000-01-14 2003-10-22 H. Lundbeck A/S Method for the preparation of 5-cyanophthalide
US6433196B1 (en) * 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate
IES20010157A2 (en) 2000-03-03 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
GB0005477D0 (en) 2000-03-07 2000-04-26 Resolution Chemicals Limited Process for the preparation of citalopram
CN1427835A (zh) 2000-03-13 2003-07-02 H·隆德贝克有限公司 5－取代的1－(4－氟苯基)－1,3－二氢异苯并呋喃的分步烷基化
JP2003527387A (ja) * 2000-03-13 2003-09-16 ハー・ルンドベック・アクチエゼルスカベット シタロプラムの製造方法
IES20010206A2 (en) 2000-03-13 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
DK1265882T3 (da) 2000-03-14 2004-06-01 Lundbeck & Co As H Fremgangsmåde til fremstilling af citalopram
KR20020080483A (ko) * 2000-03-16 2002-10-23 하. 룬트벡 아크티에 셀스카브 5-시아노-1-(4-플루오로페닐)-1,3-디히드로이소벤조푸란의제조 방법
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IL144817A0 (en) 2000-08-18 2002-06-30 Lundbeck & Co As H Method for the preparation of citalopram
SG167655A1 (en) 2000-12-22 2011-01-28 Lundbeck & Co As H Method for the preparation of pure citalopram
PT1281707E (pt) * 2001-08-02 2005-04-29 Infosint Sa Processo para a preparacao de isobenzofuranos 5-substituidos
AU2002330730A1 (en) * 2002-08-14 2004-03-03 Natco Pharma Limited Process for the preparation of high purity citalopram and its pharmaceutically acceptable salts
US8539533B2 (en) * 2003-03-07 2013-09-17 Siemens Enterprise Communications, Inc. System and method for digital personal video stream manager
TR200504022T1 (tr) * 2003-03-24 2006-08-21 Hetero Drugs Limited (S)-sitalopram oksalatın yeni sıvı kristal formları.
CN100569765C (zh) 2003-12-19 2009-12-16 杭州民生药业集团有限公司 西酞普兰中间体晶体碱
JP2006176490A (ja) * 2004-11-29 2006-07-06 Sumitomo Chemical Co Ltd ５−フタランカルボニトリル及びシタロプラムの製造方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1526331A (en) * 1976-01-14 1978-09-27 Kefalas As Phthalanes
UA62985C2 (en) * 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
PL198024B1 (pl) * 1999-04-14 2008-05-30 Lundbeck & Co As H Sposób wytwarzania citalopramu, związki pośrednie i ich zastosowanie do wytwarzania citalopramu
US6310222B1 (en) * 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate
US6433196B1 (en) * 2000-02-17 2002-08-13 Sumika Fine Chemicals Co., Ltd. Production method of citalopram, intermediate therefor and production method of the intermediate

Also Published As

Publication number Publication date
US20020004604A1 (en) 2002-01-10
BG107015A (bg) 2003-05-30
HUP0300078A3 (en) 2005-02-28
CN1161350C (zh) 2004-08-11
GR20010100097A (el) 2001-10-31
NL1017414C1 (nl) 2001-03-15
ZA200206255B (en) 2003-10-20
CA2400682A1 (en) 2001-08-30
HRP20020743A2 (en) 2003-12-31
HK1054378A1 (en) 2003-11-28
EP1259500A1 (en) 2002-11-27
PL357178A1 (en) 2004-07-26
TR200202048T2 (tr) 2003-01-21
US20030114692A1 (en) 2003-06-19
BR0108947A (pt) 2003-06-03
MXPA02008230A (es) 2003-05-23
IS6512A (is) 2002-08-20
KR20020080438A (ko) 2002-10-23
IES20010143A2 (en) 2001-07-25
SK13662002A3 (sk) 2003-01-09
ITMI20010385A1 (it) 2002-08-26
CN1404475A (zh) 2003-03-19
JP2003524009A (ja) 2003-08-12
NO20024007L (no) 2002-10-07
EA005593B1 (ru) 2005-04-28
EA200200900A1 (ru) 2003-02-27
AU2001235357A1 (en) 2001-09-03
HK1054378B (zh) 2005-04-29
FR2805813A1 (fr) 2001-09-07
IL151339A0 (en) 2003-04-10
NO20024007D0 (no) 2002-08-22
US20030083508A1 (en) 2003-05-01
HUP0300078A2 (en) 2003-05-28
WO2001062754A1 (en) 2001-08-30
ZA200206699B (en) 2003-11-21
BE1012921A6 (fr) 2001-05-08

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