UA41327C2 - Ендопаразитицидний засіб - Google Patents

Ендопаразитицидний засіб

Info

Publication number
UA41327C2
UA41327C2 UA95018024A UA95018024A UA41327C2 UA 41327 C2 UA41327 C2 UA 41327C2 UA 95018024 A UA95018024 A UA 95018024A UA 95018024 A UA95018024 A UA 95018024A UA 41327 C2 UA41327 C2 UA 41327C2
Authority
UA
Ukraine
Prior art keywords
endoparasiticide
agent
cyclohexylcarbonyl
hexahydropyrazino
benzazepine
Prior art date
Application number
UA95018024A
Other languages
English (en)
Russian (ru)
Inventor
Норберт МЕНКЕ
Ахім Хардер
Ахим ХАРДЕР
Петер Ієшке
Петер Иешке
Original Assignee
Байєр Аг
Байер Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Байєр Аг, Байер Аг filed Critical Байєр Аг
Publication of UA41327C2 publication Critical patent/UA41327C2/uk

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15—Depsipeptides; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N33/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic nitrogen compounds
    • A01N33/02—Amines; Quaternary ammonium compounds
    • A01N33/04—Nitrogen directly attached to aliphatic or cycloaliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Luminescent Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Peptides Or Proteins (AREA)
  • Compositions Of Oxide Ceramics (AREA)
  • Cosmetics (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Винахід відноситься до засобів для боротьби з комахами, зокрема до ендопаразитицидного засобу. Ендопаразитицидний засіб містить циклічний депсипептид з 6-30 кільцевих атомів, що складається з амінокислот і гідроксикарбонових кислот, які є кільцевими ланками, або його оптичний ізомер або рацемат. Засіб додатково містить 2-(циклогексилкарбоніл) -1,2,3,6,7,11b-гексагідро-4Н-піразино[2,1-р]ізохінолін-4-он або 2-(циклогексилкарбоніл) -2,3,6,7,8,12b-гексагідропіразино[2,1-р][2]-бензазепін-4(1Н) -он.
UA95018024A 1994-01-11 1995-01-10 Ендопаразитицидний засіб UA41327C2 (uk)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4400464A DE4400464A1 (de) 1994-01-11 1994-01-11 Endoparasitizide Mittel

Publications (1)

Publication Number Publication Date
UA41327C2 true UA41327C2 (uk) 2001-09-17

Family

ID=6507651

Family Applications (1)

Application Number Title Priority Date Filing Date
UA95018024A UA41327C2 (uk) 1994-01-11 1995-01-10 Ендопаразитицидний засіб

Country Status (27)

Country Link
US (1) US5589503A (uk)
EP (1) EP0662326B1 (uk)
JP (2) JP4033920B2 (uk)
KR (1) KR100359618B1 (uk)
CN (1) CN1165338C (uk)
AT (1) ATE209501T1 (uk)
AU (1) AU685535B2 (uk)
CA (1) CA2139725C (uk)
CZ (1) CZ290246B6 (uk)
DE (3) DE4400464A1 (uk)
DK (1) DK0662326T5 (uk)
ES (1) ES2168285T3 (uk)
FI (1) FI116885B (uk)
FR (1) FR06C0002I2 (uk)
HU (1) HU226207B1 (uk)
IL (1) IL112285A (uk)
NL (1) NL300218I2 (uk)
NO (2) NO307030B1 (uk)
NZ (1) NZ270300A (uk)
PH (1) PH31462A (uk)
PL (1) PL180019B1 (uk)
PT (1) PT662326E (uk)
RU (1) RU2124364C1 (uk)
SK (1) SK283367B6 (uk)
TW (1) TW364850B (uk)
UA (1) UA41327C2 (uk)
ZA (1) ZA95136B (uk)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
DE19520275A1 (de) * 1995-06-02 1996-12-05 Bayer Ag Endoparasitizide Mittel
CA2306883C (en) * 1997-10-20 2007-11-27 Dainippon Pharmaceutical Co., Ltd. Fast-dissolving pharmaceutical composition comprising as-3201
DE19921887A1 (de) * 1999-05-12 2000-11-16 Bayer Ag Endoparasitizide Mittel
DE10008128A1 (de) * 2000-02-22 2001-08-23 Bayer Ag Endoparasitizide Mittel
KR100358084B1 (ko) * 2000-10-04 2002-10-25 주식회사대성미생물연구소 프라지콴텔과 시메티딘 합제를 이용한 어류의아가미흡충증 치료방법
DE10104362A1 (de) * 2001-02-01 2002-08-08 Bayer Ag Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit
KR20040012990A (ko) * 2001-06-28 2004-02-11 제온 코포레이션 시클로알킬 알킬 에테르 화합물을 함유하여 이루어지는용제 및 시클로알킬 알킬 에테르 화합물의 제조방법
EP1450860B1 (en) * 2001-10-05 2013-09-18 Rubicon Scientific LLC Animal feeds including actives
DE10358525A1 (de) * 2003-12-13 2005-07-07 Bayer Healthcare Ag Endoparasitizide Mittel zur topischen Applikation
DE10359798A1 (de) 2003-12-19 2005-07-21 Bayer Healthcare Ag Cyclohexadepsipeptide zur Bekämpfung von Endoparasiten und ein Verfahren zu ihrer Herstellung
DE102004055316A1 (de) * 2004-11-16 2006-05-18 Bayer Healthcare Ag Verhinderung vertikaler Endoparasiten-Infektionen
DE102005011779A1 (de) * 2005-03-11 2006-09-14 Bayer Healthcare Ag Endoparasitizide Mittel
CN102149717B (zh) * 2008-08-28 2014-05-14 辉瑞大药厂 二氧杂-双环[3.2.1]辛烷-2，3，4-三醇衍生物
DE102009012423A1 (de) 2009-03-10 2010-09-16 Bayer Animal Health Gmbh Zubereitung auf Ölbasis
UA114287C2 (uk) * 2011-03-02 2017-05-25 Дзе Юніверсіті Оф Токіо Засіб для боротьби з ендопаразитами
SI2782565T1 (sl) * 2011-11-25 2019-12-31 Bayer Intellectual Property Gmbh Uporaba aril in hetaril karboksamidov kot endoparaziticid
PL3298027T3 (pl) 2015-05-20 2021-11-08 Boehringer Ingelheim Animal Health USA Inc. Przeciwrobacze związki depsipeptydów
AU2016380868B2 (en) 2015-12-28 2019-11-28 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
US11382949B2 (en) 2016-11-16 2022-07-12 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
CA3147171A1 (en) 2019-08-14 2021-02-18 Vetoquinol Sa Compositions comprising tigolaner for controlling parasites
CN113943350B (zh) * 2021-11-02 2023-08-15 海南大学三亚南繁研究院 一种环肽化合物或其药学上可接受的盐及其制备方法和应用、药物及其应用

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO176766C (no) * 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
GB9024924D0 (en) * 1990-11-16 1991-01-02 Beecham Group Plc Novel compositions
NZ247278A (en) * 1991-02-12 1995-03-28 Ancare Distributors Veterinary anthelmintic drench comprising a suspension of praziquantel in a liquid carrier
DK0634408T3 (da) * 1992-03-17 2002-04-22 Fujisawa Pharmaceutical Co Depsipeptidderivater, fremstilling og anvendelse deraf
DE4317458A1 (de) * 1992-06-11 1993-12-16 Bayer Ag Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung
CN1073560C (zh) * 1993-02-19 2001-10-24 明治制果株式会社 环缩酚酸肽pf1022衍生物
DE4317457A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4317432A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung

Also Published As

Publication number Publication date
CZ6195A3 (en) 1995-07-12
DE4400464A1 (de) 1995-07-13
NO950093L (no) 1995-07-12
EP0662326A2 (de) 1995-07-12
FR06C0002I2 (uk) 2006-12-29
AU8159294A (en) 1995-07-20
FR06C0002I1 (uk) 2006-03-10
CN1121429A (zh) 1996-05-01
RU2124364C1 (ru) 1999-01-10
NO2006001I1 (no) 2006-02-13
NO2006001I2 (no) 2008-02-04
CZ290246B6 (cs) 2002-06-12
ES2168285T3 (es) 2002-06-16
PT662326E (pt) 2002-05-31
DE122006000001I2 (de) 2007-05-24
NZ270300A (en) 1995-09-26
NO307030B1 (no) 2000-01-31
DK0662326T5 (da) 2008-11-03
NO950093D0 (no) 1995-01-10
CA2139725C (en) 2005-01-04
CA2139725A1 (en) 1995-07-12
NL300218I2 (nl) 2006-07-03
TW364850B (en) 1999-07-21
NL300218I1 (nl) 2006-04-03
EP0662326A3 (de) 1997-12-17
KR100359618B1 (ko) 2003-01-29
FI116885B (fi) 2006-03-31
IL112285A0 (en) 1995-03-30
FI950091A0 (fi) 1995-01-09
HU226207B1 (en) 2008-06-30
RU95100759A (ru) 1997-03-20
CN1165338C (zh) 2004-09-08
JPH07223951A (ja) 1995-08-22
PL180019B1 (pl) 2000-12-29
EP0662326B1 (de) 2001-11-28
US5589503A (en) 1996-12-31
SK3195A3 (en) 1995-08-09
AU685535B2 (en) 1998-01-22
IL112285A (en) 1999-06-20
SK283367B6 (sk) 2003-06-03
FI950091A (fi) 1995-07-12
DE122006000001I1 (de) 2006-05-04
HUT69180A (en) 1995-08-28
ATE209501T1 (de) 2001-12-15
PL306709A1 (en) 1995-07-24
KR950031104A (ko) 1995-12-18
ZA95136B (en) 1995-09-07
JP2007314580A (ja) 2007-12-06
DK0662326T3 (da) 2002-03-18
JP4033920B2 (ja) 2008-01-16
PH31462A (en) 1998-11-03
DE59409977D1 (de) 2002-01-10

Similar Documents

Publication Publication Date Title
UA41327C2 (uk) Ендопаразитицидний засіб
HUP9802866A3 (en) 2,4,5-trisubstituted phenylketo-enol-derivatives, intermediates, insecticide, acaricide and herbicide compositions containing these compounds as active ingredients, process for the preparation and use of the compounds and compositions
DE69632841D1 (de) Verfahren zur Herstellung von fluorinierten Nitrilen aus den entsprechenden Amiden
DE69801973T2 (de) Verfahren zur Herstellung von 1,1,1,3,3-Pentafluorpropan
PL315653A1 (en) Application of 4-chloro-5-(imidazolyn-2-ylamino)-6-methoxy-2-methylpyrimidine and i1 agonist as pharmaceutic agents and pharmaceutic agent as such
DE69509624T2 (de) Verfahren zur Herstellung von 1-(2'-Deoxy-2',2'-difluoro-D-ribofuranosyl)-4-amino-pyrimidin-2-on-hydrochlorid
ZA956276B (en) Insect viruses sequences insecticidal compositions and methods of use
DE59809260D1 (de) Verfahren zur Herstellung von niedermolekularen Homopolymerisaten des N-Vinylpyrrolidons
DE69608414D1 (de) Als insektizid aktive zusammensetzung
HUT75053A (en) Insecticidal n-(substituted arylmethyl)-4-[bis(substituted phenyl)methyl]piperidines, insecticid composition and use of it
HUP9900795A3 (en) Sinergetical fungicide composition containing fenazaquine and amide compound as active ingredients and use thereof
DE69524111T2 (de) Verfahren zur Herstellung von Poly-p-Phenylenterephtalamidpulpen
SI0688771T1 (en) Use of lactam compounds as pharmaceutical agents
EA199901113A1 (ru) Карбоксамиды в качестве агонистов 5-ht1f
CA2149969A1 (en) Suspension concentrate compositions of arylpyrrole insecticidal and acaricidal agents
DE59401009D1 (de) Verfahren zur Herstellung von 1,1,1,3,3-Pentafluorpropan
DE69511788D1 (de) Verfahren zur Herstellung von 1,1,1,3,3-Pentafluorpropan
DE59907526D1 (de) Verfahren zur Herstellung von 3-Cyano-3,5,5-trimethyl-cyclohexanon
CA2042673A1 (en) Acetyl-tri- and tetramethyl-octahydronaphthalenes and fragrance compositions containing the same
DE59407859D1 (de) Verfahren zur Herstellung von N-substituierten Pyrazolen
DE59105224D1 (de) Verfahren zur Herstellung von N-substituierten Pyrrolidonen.
AU8023498A (en) Cosmetic composition comprising an amide and novel amides
DE69610037T2 (de) Verfahren zur Herstellung von 2-(2'-Hydroxyphenol)-Benzotriazolverbindungen
DE69801180D1 (de) Verfahren zur Herstellung von 3,3-dichlor-1,1,1-trifluoraceton
GEP20032975B (en) Echinocandin Derivatives, Preparation Method and Pharmaceutical Composition