SK283367B6 - Endoparaziticídne prostriedky a ich použitie - Google Patents
Endoparaziticídne prostriedky a ich použitie Download PDFInfo
- Publication number
- SK283367B6 SK283367B6 SK31-95A SK3195A SK283367B6 SK 283367 B6 SK283367 B6 SK 283367B6 SK 3195 A SK3195 A SK 3195A SK 283367 B6 SK283367 B6 SK 283367B6
- Authority
- SK
- Slovakia
- Prior art keywords
- spp
- praziquantel
- group
- methyl
- epsiprantel
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/15—Depsipeptides; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/08—Peptides having 5 to 11 amino acids
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N33/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic nitrogen compounds
- A01N33/02—Amines; Quaternary ammonium compounds
- A01N33/04—Nitrogen directly attached to aliphatic or cycloaliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Immunology (AREA)
- Gastroenterology & Hepatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Plant Pathology (AREA)
- Agronomy & Crop Science (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Luminescent Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Peptides Or Proteins (AREA)
- Compositions Of Oxide Ceramics (AREA)
- Cosmetics (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Steroid Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
Description
Cčinná iátíca | -f. <tóvka íras*sl |
CyKÍo-Í.NíeLei-D-Lac-Mei.sti-O-PiLac-Miá.sd-D-Lsc-MíLÄi-D- (F.Uac)· pF I022J | 1 |
12<CytIohcQ'lfcarbdnyl)’12^6^lľo*h«xahy<iro^H^yraziiioí2,la.liío-quiaGUa-4-or. pnziqutQtel] | 0 |
2^Cy«iohar/lsarboByi)-2,3,6,7,8,!2Wiax3ŕiydro»pyraxífio[2,1 · a](2]b«iz-azspÍn-4(iH)-aa [Epsipniiis:] | 0 |
?hLac)- pF 1022] * 2-(Cytíoaíxyliarôonyl)’I2,3,5.7,llb-hecaíiydto-4H-tynxaop,I· Prsdqcantel] (1:1) | OJ |
Cy hlc -{MaLai-D-Lac •MeLÄ-D‘?hLac-MdrSC«D’Lac-M«L ss-DFhLac)- PF 1022]' 2-(Cyiíloiic^rlkaŕboayI)-2,3,ô,7?8,12b-íie»ihydro-pyti2Ínc[2,l· a](.2]besz-azepÍ3*4(lH)-oo [Sršpraotel] (1:1) | 0,5 |
D-0-Mctfhí.ac·) | OJ |
í Ľ-o-McrPaLac-) ŕ- 2~(Cyc|oiwxytííarbonyI)“14.3,6,7.1U*heX3hyära-4H<fyr3zb0(fcTl» a]iso-quinout-4-oG prsdícuafltói] (Ll) | 025 |
Cyílo(-^íei,íc-Ĺ?*Lac->íe£ed-D-Ľi-Moi?liLacT4cLsy-D-L3c-MeLsu- i D-p-MoďhUc·) * j 2<CvfclohexyleartJOttyL>23^,7,8,12Mi«c4Ítyá»-pyrízáwí2J· ä a](2]benz*az»?in.’4(iK)-«íi (Epíiprantei) (1:1) | 025 |
ôčisná látkŕ. | íť. Wlí?J |
Cyilo-(MeLs!:>D-L«:’J/íeLea-D-?hLac*MeLeii.D-Lac-Mei,«u-D?hLw-) pF 1022] | t |
a]Í3c-qui.n.oui-4-oa | 0 |
a](l}bea2-az8?ia«4(lH>oa | 0 |
PhLac)- [PF 1022] + 2^CyHoasxyIftarWyí>lX3,6,7,ÍIb4iexQhydro^H^yrsziao(2,l· íJiso-tfuiaalBj-é-oa prszjcujDtei] (1:1) | 0.5 |
Cyilo^J/íeLsti-D-LsC'MeLeU'C'PbliC-MeLsti-D’Lac-MíLeu-D?hlac> (PF 1022] * 2^CyJúoaexylbi«bcfiyl>2^,6,7,S1Ub-hexiÄyáx-5yfmnoľ2,l31[2]béS2-«za?a-KlK)-ča. pasisnottl) (1:1) | 0.5 |
D-o-MorFilac·) | C, 5 |
D“p-Mor?hL3c-) 4* 2-(Cytíeaexy Unrboay ‘,11^-ΐ«χώ.νώχ;-4Η·ργπζ:ηοΓ2,1- ip5G<uinolii-4-0Q [rrazisujats’.l (!:’) | OJÍ |
C7sio(’MeLM<0-L3e-MeLstt-D-p-MoďhLac«Me'.5tt’D-Lx-M«LffuD-a'Mur?hLac-) * 2-(Cyfclohc^UaréonyD-2,3,ó5,V2b^Mwyiro«pyT3Zino[2,!- [Fpipnauí] (VI) | o.a |
Claims (2)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE4400464A DE4400464A1 (de) | 1994-01-11 | 1994-01-11 | Endoparasitizide Mittel |
Publications (2)
Publication Number | Publication Date |
---|---|
SK3195A3 SK3195A3 (en) | 1995-08-09 |
SK283367B6 true SK283367B6 (sk) | 2003-06-03 |
Family
ID=6507651
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SK31-95A SK283367B6 (sk) | 1994-01-11 | 1995-01-10 | Endoparaziticídne prostriedky a ich použitie |
Country Status (27)
Country | Link |
---|---|
US (1) | US5589503A (sk) |
EP (1) | EP0662326B1 (sk) |
JP (2) | JP4033920B2 (sk) |
KR (1) | KR100359618B1 (sk) |
CN (1) | CN1165338C (sk) |
AT (1) | ATE209501T1 (sk) |
AU (1) | AU685535B2 (sk) |
CA (1) | CA2139725C (sk) |
CZ (1) | CZ290246B6 (sk) |
DE (3) | DE4400464A1 (sk) |
DK (1) | DK0662326T5 (sk) |
ES (1) | ES2168285T3 (sk) |
FI (1) | FI116885B (sk) |
FR (1) | FR06C0002I2 (sk) |
HU (1) | HU226207B1 (sk) |
IL (1) | IL112285A (sk) |
NL (1) | NL300218I2 (sk) |
NO (2) | NO307030B1 (sk) |
NZ (1) | NZ270300A (sk) |
PH (1) | PH31462A (sk) |
PL (1) | PL180019B1 (sk) |
PT (1) | PT662326E (sk) |
RU (1) | RU2124364C1 (sk) |
SK (1) | SK283367B6 (sk) |
TW (1) | TW364850B (sk) |
UA (1) | UA41327C2 (sk) |
ZA (1) | ZA95136B (sk) |
Families Citing this family (22)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE4317458A1 (de) * | 1992-06-11 | 1993-12-16 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung |
DE19520275A1 (de) * | 1995-06-02 | 1996-12-05 | Bayer Ag | Endoparasitizide Mittel |
BR9814090A (pt) * | 1997-10-20 | 2000-10-03 | Dainippon Pharmaceutical Co | Composição de drogas rapidamente solúvel |
DE19921887A1 (de) * | 1999-05-12 | 2000-11-16 | Bayer Ag | Endoparasitizide Mittel |
DE10008128A1 (de) * | 2000-02-22 | 2001-08-23 | Bayer Ag | Endoparasitizide Mittel |
KR100358084B1 (ko) * | 2000-10-04 | 2002-10-25 | 주식회사대성미생물연구소 | 프라지콴텔과 시메티딘 합제를 이용한 어류의아가미흡충증 치료방법 |
DE10104362A1 (de) * | 2001-02-01 | 2002-08-08 | Bayer Ag | Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit |
KR20040012990A (ko) * | 2001-06-28 | 2004-02-11 | 제온 코포레이션 | 시클로알킬 알킬 에테르 화합물을 함유하여 이루어지는용제 및 시클로알킬 알킬 에테르 화합물의 제조방법 |
BR0213124A (pt) * | 2001-10-05 | 2004-09-21 | Rubicon Scient Llc | Alimentos para animais incluindo ativos e métodos de uso dos mesmos |
DE10358525A1 (de) * | 2003-12-13 | 2005-07-07 | Bayer Healthcare Ag | Endoparasitizide Mittel zur topischen Applikation |
DE10359798A1 (de) * | 2003-12-19 | 2005-07-21 | Bayer Healthcare Ag | Cyclohexadepsipeptide zur Bekämpfung von Endoparasiten und ein Verfahren zu ihrer Herstellung |
DE102004055316A1 (de) * | 2004-11-16 | 2006-05-18 | Bayer Healthcare Ag | Verhinderung vertikaler Endoparasiten-Infektionen |
DE102005011779A1 (de) * | 2005-03-11 | 2006-09-14 | Bayer Healthcare Ag | Endoparasitizide Mittel |
RS52236B (en) * | 2008-08-28 | 2012-10-31 | Pfizer Inc. | DIOKASA-BICYCLE DERIVATIVES (3.2.1) OCTOBER-2,3,4-TRIOLA |
DE102009012423A1 (de) | 2009-03-10 | 2010-09-16 | Bayer Animal Health Gmbh | Zubereitung auf Ölbasis |
CN103415288B (zh) | 2011-03-02 | 2018-04-03 | 国立大学法人东京大学 | 体内寄生虫防除剂 |
HUE047738T2 (hu) * | 2011-11-25 | 2020-05-28 | Bayer Ip Gmbh | Aril- és hetaril-karboxamidok alkalmazása mint endoparaziticid szerek |
RS62130B1 (sr) * | 2015-05-20 | 2021-08-31 | Boehringer Ingelheim Animal Health Usa Inc | Antihelmintička depsipeptidna jedinjenja |
RU2715556C2 (ru) | 2015-12-28 | 2020-03-02 | Мериал, Инк. | Противогельминтные депсипептидные соединения |
WO2018093920A1 (en) | 2016-11-16 | 2018-05-24 | Merial, Inc. | Anthelmintic depsipeptide compounds |
US20220331314A1 (en) | 2019-08-14 | 2022-10-20 | Vetoquinol Sa | Compositions comprising tigolaner for controlling parasites |
CN113943350B (zh) * | 2021-11-02 | 2023-08-15 | 海南大学三亚南繁研究院 | 一种环肽化合物或其药学上可接受的盐及其制备方法和应用、药物及其应用 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NO176766C (no) * | 1989-02-07 | 1995-05-24 | Meiji Seika Kaisha | Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet |
GB9024924D0 (en) * | 1990-11-16 | 1991-01-02 | Beecham Group Plc | Novel compositions |
NZ247278A (en) * | 1991-02-12 | 1995-03-28 | Ancare Distributors | Veterinary anthelmintic drench comprising a suspension of praziquantel in a liquid carrier |
WO1993019053A1 (fr) * | 1992-03-17 | 1993-09-30 | Fujisawa Pharmaceutical Co., Ltd. | Derive de depsipeptide, production et utilisation |
DE4317458A1 (de) * | 1992-06-11 | 1993-12-16 | Bayer Ag | Verwendung von cyclischen Depsipeptiden mit 18 Ringatomen zur Bekämpfung von Endoparasiten, neue cyclische Depsipeptide mit 18 Ringatomen und Verfahren zu ihrer Herstellung |
NZ261630A (en) * | 1993-02-19 | 1998-05-27 | Meiji Seika Kaisha | Heteromacrocyclic compound and use as an assthelmintie |
DE4317432A1 (de) * | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
DE4317457A1 (de) * | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptide mit endoparasitizider Wirkung |
-
1994
- 1994-01-11 DE DE4400464A patent/DE4400464A1/de not_active Withdrawn
- 1994-12-16 TW TW083111751A patent/TW364850B/zh not_active IP Right Cessation
- 1994-12-20 AU AU81592/94A patent/AU685535B2/en not_active Expired
- 1994-12-27 DK DK94120772T patent/DK0662326T5/da active
- 1994-12-27 DE DE1994509977 patent/DE122006000001I2/de active Active
- 1994-12-27 DE DE59409977T patent/DE59409977D1/de not_active Expired - Lifetime
- 1994-12-27 ES ES94120772T patent/ES2168285T3/es not_active Expired - Lifetime
- 1994-12-27 PT PT94120772T patent/PT662326E/pt unknown
- 1994-12-27 EP EP94120772A patent/EP0662326B1/de not_active Expired - Lifetime
- 1994-12-27 AT AT94120772T patent/ATE209501T1/de active
-
1995
- 1995-01-04 US US08/368,515 patent/US5589503A/en not_active Expired - Lifetime
- 1995-01-06 CA CA002139725A patent/CA2139725C/en not_active Expired - Lifetime
- 1995-01-06 NZ NZ270300A patent/NZ270300A/en not_active IP Right Cessation
- 1995-01-09 FI FI950091A patent/FI116885B/fi not_active IP Right Cessation
- 1995-01-09 PL PL95306709A patent/PL180019B1/pl unknown
- 1995-01-09 PH PH49754A patent/PH31462A/en unknown
- 1995-01-09 KR KR1019950000274A patent/KR100359618B1/ko not_active IP Right Cessation
- 1995-01-09 IL IL11228595A patent/IL112285A/xx not_active IP Right Cessation
- 1995-01-09 JP JP01633595A patent/JP4033920B2/ja not_active Expired - Lifetime
- 1995-01-10 HU HU9500065A patent/HU226207B1/hu active Protection Beyond IP Right Term
- 1995-01-10 NO NO950093A patent/NO307030B1/no not_active IP Right Cessation
- 1995-01-10 CZ CZ199561A patent/CZ290246B6/cs not_active IP Right Cessation
- 1995-01-10 SK SK31-95A patent/SK283367B6/sk not_active IP Right Cessation
- 1995-01-10 ZA ZA95136A patent/ZA95136B/xx unknown
- 1995-01-10 UA UA95018024A patent/UA41327C2/uk unknown
- 1995-01-11 RU RU95100759/13A patent/RU2124364C1/ru active Protection Beyond IP Right Term
- 1995-01-11 CN CNB951011588A patent/CN1165338C/zh not_active Expired - Lifetime
-
2006
- 2006-01-26 FR FR06C0002C patent/FR06C0002I2/fr active Active
- 2006-01-26 NL NL300218C patent/NL300218I2/nl unknown
- 2006-01-27 NO NO2006001C patent/NO2006001I2/no unknown
-
2007
- 2007-09-04 JP JP2007228858A patent/JP2007314580A/ja active Pending
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC4A | Assignment and transfer of rights |
Owner name: BAYER INTELLECTUAL PROPERTY GMBH, MONHEIM AM R, DE Free format text: FORMER OWNER: BAYER ANIMAL HEALTH GMBH, LEVERKUSEN, DE Effective date: 20121011 |
|
SPCT | Transfer of rights of an spc |
Owner name: BAYER INTELLECTUAL PROPERTY GMBH Free format text: PRODUCT NAME: EMODEPSID A PRAZIQUANTEL; REGISTRATION NO/DATE: EU/2/05/054/001-014 20050727 Spc suppl protection certif: DO 42; 5001-2006 Filing date: 20060119 Extension date: 20200111 Effective date: 20130108 |
|
MK4A | Patent expired |
Expiry date: 20150110 |
|
SPCE | Expiry of an spc |
Free format text: PRODUCT NAME: EMODEPSID A PRAZIQUANTEL Spc suppl protection certif: 42, 5001-2006 Effective date: 20200111 |