UA109414C2 - Арильовані камфени та фармацевтична композиція на їх основі - Google Patents

Арильовані камфени та фармацевтична композиція на їх основі

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Publication number
UA109414C2
UA109414C2 UAA201203785A UAA201203785A UA109414C2 UA 109414 C2 UA109414 C2 UA 109414C2 UA A201203785 A UAA201203785 A UA A201203785A UA A201203785 A UAA201203785 A UA A201203785A UA 109414 C2 UA109414 C2 UA 109414C2
Authority
UA
Ukraine
Prior art keywords
pharmaceutical formulation
camphenes
arylated
arylated camphenes
benefiting
Prior art date
Application number
UAA201203785A
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English (en)
Russian (ru)
Inventor
Рафаель МЕЧУЛАМ
Літаль Магід
Естер Шохамі
Ітаі Баб
Original Assignee
Їсум Ресьорч Девелопмент Компані Оф Зе Хебрю Юніверсіті Оф Єрусалім, Лтд.
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43875675&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA109414(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Їсум Ресьорч Девелопмент Компані Оф Зе Хебрю Юніверсіті Оф Єрусалім, Лтд. filed Critical Їсум Ресьорч Девелопмент Компані Оф Зе Хебрю Юніверсіті Оф Єрусалім, Лтд.
Publication of UA109414C2 publication Critical patent/UA109414C2/uk

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C43/00—Ethers; Compounds having groups, groups or groups
    • C07C43/02—Ethers
    • C07C43/20—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring
    • C07C43/23—Ethers having an ether-oxygen atom bound to a carbon atom of a six-membered aromatic ring containing hydroxy or O-metal groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D311/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/94—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems condensed with rings other than six-membered or with ring systems containing such rings
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/075—Ethers or acetals
    • A61K31/085—Ethers or acetals having an ether linkage to aromatic ring nuclear carbon
    • A61K31/09—Ethers or acetals having an ether linkage to aromatic ring nuclear carbon having two or more such linkages
    • A—HUMAN NECESSITIES
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A—HUMAN NECESSITIES
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    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
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    • C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
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  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Neurosurgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Hospice & Palliative Care (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
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  • Reproductive Health (AREA)
  • Vascular Medicine (AREA)
  • Otolaryngology (AREA)
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Abstract

Даний винахід стосується арильованих камфенів, способів їхнього отримання та їхніх застосувань для отримання лікарських засобів для лікування захворювань, розладів або станів, які пов'язані зі стимуляцією рецепторів СВ2 або на які сприятливо впливає стимуляція рецепторів СВ2.
UAA201203785A 2009-11-19 2010-11-18 Арильовані камфени та фармацевтична композиція на їх основі UA109414C2 (uk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US26267709P 2009-11-19 2009-11-19
PCT/IL2010/000970 WO2011061744A2 (en) 2009-11-19 2010-11-18 Novel arylated camphenes, processes for their preparation and uses thereof

Publications (1)

Publication Number Publication Date
UA109414C2 true UA109414C2 (uk) 2015-08-25

Family

ID=43875675

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201203785A UA109414C2 (uk) 2009-11-19 2010-11-18 Арильовані камфени та фармацевтична композиція на їх основі

Country Status (24)

Country Link
US (2) US8722938B2 (uk)
EP (1) EP2501669B1 (uk)
JP (1) JP5960058B2 (uk)
KR (1) KR20120091196A (uk)
CN (1) CN102648174B (uk)
AU (1) AU2010320467B2 (uk)
BR (1) BR112012010518A2 (uk)
CA (1) CA2774868C (uk)
CL (1) CL2012001290A1 (uk)
CO (1) CO6481008A2 (uk)
CR (1) CR20120247A (uk)
EC (1) ECSP12011864A (uk)
ES (1) ES2665519T3 (uk)
IL (1) IL218216A (uk)
MA (1) MA33753B1 (uk)
MX (2) MX2012005634A (uk)
MY (1) MY184647A (uk)
NZ (1) NZ599106A (uk)
PE (1) PE20121187A1 (uk)
RU (1) RU2578715C2 (uk)
SG (2) SG10201407706VA (uk)
UA (1) UA109414C2 (uk)
WO (1) WO2011061744A2 (uk)
ZA (1) ZA201200752B (uk)

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MX2012005634A (es) * 2009-11-19 2012-09-07 Yissum Res Dev Co Canfenos arilados novedosos, procesos para su preparacion y usos.
JP6637034B2 (ja) 2014-10-27 2020-01-29 エフ．ホフマン−ラ ロシュ アーゲーＦ． Ｈｏｆｆｍａｎｎ−Ｌａ Ｒｏｃｈｅ Ａｋｔｉｅｎｇｅｓｅｌｌｓｃｈａｆｔ 放射標識カンナビノイド受容体２リガンド
US9585867B2 (en) 2015-08-06 2017-03-07 Charles Everett Ankner Cannabinod formulation for the sedation of a human or animal
KR20180094856A (ko) * 2015-10-16 2018-08-24 스키티안 바이오사이언시즈 아이엔씨. 외상성 뇌손상 치료를 위한 방법 및 조성물
WO2018087767A1 (en) 2016-11-13 2018-05-17 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. Process for the preparation of hu-910 and crystalline structure thereof
RU2651754C1 (ru) * 2016-11-25 2018-04-23 Федеральное государственное бюджетное учреждение науки Новосибирский институт органической химии им. Н.Н. Ворожцова Сибирского отделения Российской академии наук (НИОХ СО РАН) ПРИМЕНЕНИЕ АЛИФАТИЧЕСКИХ ИМИНОПРОИЗВОДНЫХ КАМФОРЫ В КАЧЕСТВЕ ЭФФЕКТИВНЫХ ИНГИБИТОРОВ РЕПРОДУКЦИИ ВИРУСА ГРИППА штамм A/California/07/09 (H1N1) pdm09 и A/Puerto Rico/8/34 (H1N1)
KR102063962B1 (ko) * 2017-10-25 2020-01-08 대구대학교 산학협력단 캄펜을 유효성분으로 함유하는 골다공증의 예방 또는 치료용 약학적 조성물
CA3110195A1 (en) * 2018-08-20 2020-02-27 Bessor Pharma, Llc Process for the production of cannabinoids
WO2023058033A1 (en) * 2021-10-10 2023-04-13 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. Arylated fenchone derivatives, compositions comprising them, processes for their preparation and uses thereof

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BR112012010518A2 (pt) 2016-03-15
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CN102648174B (zh) 2016-04-27
SG179203A1 (en) 2012-04-27
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KR20120091196A (ko) 2012-08-17
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