TWI791423B - C3腎絲球病變之治療方法 - Google Patents

C3腎絲球病變之治療方法 Download PDF

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Publication number
TWI791423B
TWI791423B TW106100938A TW106100938A TWI791423B TW I791423 B TWI791423 B TW I791423B TW 106100938 A TW106100938 A TW 106100938A TW 106100938 A TW106100938 A TW 106100938A TW I791423 B TWI791423 B TW I791423B
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TW106100938A
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TW201726134A (zh
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佩脫拉斯 貝克
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美商卡默森屈有限公司
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/451—Non condensed piperidines, e.g. piperocaine having a carbocyclic group directly attached to the heterocyclic ring, e.g. glutethimide, meperidine, loperamide, phencyclidine, piminodine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Urology & Nephrology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicines Containing Plant Substances (AREA)
TW106100938A 2016-01-14 2017-01-12 C3腎絲球病變之治療方法 TWI791423B (zh)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
US201662278788P 2016-01-14 2016-01-14
US62/278,788 2016-01-14
US201662280346P 2016-01-19 2016-01-19
US62/280,346 2016-01-19
US201662347450P 2016-06-08 2016-06-08
US62/347,450 2016-06-08
US201662397527P 2016-09-21 2016-09-21
US62/397,527 2016-09-21

Publications (2)

Publication Number Publication Date
TW201726134A TW201726134A (zh) 2017-08-01
TWI791423B true TWI791423B (zh) 2023-02-11

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TW106100938A TWI791423B (zh) 2016-01-14 2017-01-12 C3腎絲球病變之治療方法

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US (3) US20170202821A1 (enExample)
EP (1) EP3402486B1 (enExample)
JP (4) JP7339733B2 (enExample)
KR (1) KR102767008B1 (enExample)
CN (1) CN108601790B (enExample)
AU (1) AU2017207359C1 (enExample)
BR (2) BR112018014222A2 (enExample)
CA (1) CA3010735C (enExample)
ES (1) ES3026359T3 (enExample)
IL (1) IL260539B (enExample)
MA (1) MA43872A (enExample)
MX (2) MX2022006069A (enExample)
NZ (1) NZ744083A (enExample)
RU (1) RU2742888C2 (enExample)
SG (1) SG11201805828YA (enExample)
TW (1) TWI791423B (enExample)
WO (1) WO2017123716A1 (enExample)
ZA (1) ZA201804513B (enExample)

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CN116322683A (zh) * 2020-08-07 2023-06-23 科越医药(苏州)有限公司 作为c5ar抑制剂的化合物
CN116635075A (zh) * 2020-12-21 2023-08-22 坎莫森特里克斯公司 使用c5a抑制剂治疗c3肾小球病
CN115192563B (zh) * 2022-05-09 2023-10-13 北京大学第一医院 C3a/C3aR通路拮抗剂治疗原发性膜性肾病的用途

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US8845515B2 (en) * 2011-01-17 2014-09-30 Coloplast A/S Penile implant with dilatant liquid

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BR112018014222A2 (pt) 2018-12-11
US11779576B2 (en) 2023-10-10
JP2024110998A (ja) 2024-08-16
US20170202821A1 (en) 2017-07-20
JP2021183625A (ja) 2021-12-02
CN108601790B (zh) 2026-01-27
JP7339733B2 (ja) 2023-09-06
EP3402486B1 (en) 2025-03-19
US11285138B2 (en) 2022-03-29
US20220354837A1 (en) 2022-11-10
TW201726134A (zh) 2017-08-01
AU2017207359C1 (en) 2022-09-01
BR122024002810A2 (pt) 2024-03-12
MX2022006069A (es) 2023-01-12
WO2017123716A1 (en) 2017-07-20
AU2017207359B2 (en) 2022-04-14
ES3026359T3 (en) 2025-06-11
KR20180102642A (ko) 2018-09-17
MA43872A (fr) 2021-05-19
MX2018008624A (es) 2018-12-10
US20190201388A1 (en) 2019-07-04
RU2018129378A3 (enExample) 2020-05-20
JP2019501935A (ja) 2019-01-24
CA3010735A1 (en) 2017-07-20
RU2018129378A (ru) 2020-02-14
IL260539B (en) 2021-05-31
SG11201805828YA (en) 2018-08-30
KR102767008B1 (ko) 2025-02-11
EP3402486C0 (en) 2025-03-19
JP7788814B2 (ja) 2025-12-19
NZ744083A (en) 2022-07-01
CA3010735C (en) 2023-06-13
ZA201804513B (en) 2024-01-31
EP3402486A4 (en) 2019-08-28
CN108601790A (zh) 2018-09-28
AU2017207359A1 (en) 2018-07-26
JP2023126235A (ja) 2023-09-07
RU2742888C2 (ru) 2021-02-11
EP3402486A1 (en) 2018-11-21

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