TW350845B - New substituted oxazolidinones - Google Patents
New substituted oxazolidinonesInfo
- Publication number
- TW350845B TW350845B TW086101259A TW86101259A TW350845B TW 350845 B TW350845 B TW 350845B TW 086101259 A TW086101259 A TW 086101259A TW 86101259 A TW86101259 A TW 86101259A TW 350845 B TW350845 B TW 350845B
- Authority
- TW
- Taiwan
- Prior art keywords
- branched chain
- straight
- carbon atoms
- chain alkyl
- substituted
- Prior art date
Links
- IZXIZTKNFFYFOF-UHFFFAOYSA-N 2-Oxazolidone Chemical class O=C1NCCO1 IZXIZTKNFFYFOF-UHFFFAOYSA-N 0.000 title abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 12
- 125000004432 carbon atom Chemical group C* 0.000 abstract 9
- 229910052739 hydrogen Inorganic materials 0.000 abstract 9
- 239000001257 hydrogen Substances 0.000 abstract 9
- 229910052799 carbon Inorganic materials 0.000 abstract 6
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 5
- 150000003254 radicals Chemical group 0.000 abstract 4
- 150000002431 hydrogen Chemical group 0.000 abstract 3
- 229910052757 nitrogen Inorganic materials 0.000 abstract 3
- 229910052717 sulfur Inorganic materials 0.000 abstract 3
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 2
- 125000003342 alkenyl group Chemical group 0.000 abstract 2
- 125000004414 alkyl thio group Chemical group 0.000 abstract 2
- 125000003118 aryl group Chemical group 0.000 abstract 2
- 125000001797 benzyl group Chemical group [H]C1=C([H])C([H])=C(C([H])=C1[H])C([H])([H])* 0.000 abstract 2
- 150000001721 carbon Chemical group 0.000 abstract 2
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 2
- 125000005842 heteroatom Chemical group 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 229920006395 saturated elastomer Polymers 0.000 abstract 2
- UHOVQNZJYSORNB-UHFFFAOYSA-N Benzene Chemical group C1=CC=CC=C1 UHOVQNZJYSORNB-UHFFFAOYSA-N 0.000 abstract 1
- 150000005840 aryl radicals Chemical group 0.000 abstract 1
- 125000000524 functional group Chemical group 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 229910052760 oxygen Inorganic materials 0.000 abstract 1
- 125000004076 pyridyl group Chemical group 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6564—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms
- C07F9/6581—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and nitrogen atoms with or without oxygen or sulfur atoms, as ring hetero atoms
- C07F9/6584—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and nitrogen atoms with or without oxygen or sulfur atoms, as ring hetero atoms having one phosphorus atom as ring hetero atom
- C07F9/65842—Cyclic amide derivatives of acids of phosphorus, in which one nitrogen atom belongs to the ring
- C07F9/65844—Cyclic amide derivatives of acids of phosphorus, in which one nitrogen atom belongs to the ring the phosphorus atom being part of a five-membered ring which may be condensed with another ring system
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19604223A DE19604223A1 (de) | 1996-02-06 | 1996-02-06 | Neue substituierte Oxazolidinone |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW350845B true TW350845B (en) | 1999-01-21 |
Family
ID=7784633
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW086101259A TW350845B (en) | 1996-02-06 | 1997-02-04 | New substituted oxazolidinones |
Country Status (36)
| Country | Link |
|---|---|
| US (1) | US5792765A (fr) |
| EP (1) | EP0789025B1 (fr) |
| JP (1) | JPH09316073A (fr) |
| KR (1) | KR970061888A (fr) |
| CN (1) | CN1160051A (fr) |
| AR (1) | AR005703A1 (fr) |
| AT (1) | ATE200285T1 (fr) |
| AU (1) | AU1251697A (fr) |
| BG (1) | BG101193A (fr) |
| BR (1) | BR9700885A (fr) |
| CA (1) | CA2196862A1 (fr) |
| CO (1) | CO4560411A1 (fr) |
| CZ (1) | CZ34097A3 (fr) |
| DE (2) | DE19604223A1 (fr) |
| DK (1) | DK0789025T3 (fr) |
| EE (1) | EE9700043A (fr) |
| ES (1) | ES2157027T3 (fr) |
| GR (1) | GR3036015T3 (fr) |
| HR (1) | HRP970048A2 (fr) |
| HU (1) | HUP9700358A3 (fr) |
| ID (1) | ID15881A (fr) |
| IL (1) | IL120125A0 (fr) |
| MX (1) | MX9700886A (fr) |
| NO (1) | NO970511L (fr) |
| NZ (1) | NZ314179A (fr) |
| PL (1) | PL318277A1 (fr) |
| PT (1) | PT789025E (fr) |
| SG (1) | SG50791A1 (fr) |
| SI (1) | SI0789025T1 (fr) |
| SK (1) | SK15897A3 (fr) |
| SV (1) | SV1997000009A (fr) |
| TN (1) | TNSN97032A1 (fr) |
| TR (1) | TR199700092A2 (fr) |
| TW (1) | TW350845B (fr) |
| YU (1) | YU4397A (fr) |
| ZA (1) | ZA97927B (fr) |
Families Citing this family (67)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9601666D0 (en) * | 1996-01-27 | 1996-03-27 | Zeneca Ltd | Chemical compounds |
| WO1998054161A1 (fr) * | 1997-05-30 | 1998-12-03 | Pharmacia & Upjohn Company | Agents antibacteriens oxazolidinone ayant une fonctionnalite thiocarbonyle |
| US6255304B1 (en) | 1997-05-30 | 2001-07-03 | Pharmacia & Upjohn Company | Oxazolidinone antibacterial agents having a thiocarbonyl functionality |
| AU9001598A (en) * | 1997-09-11 | 1999-03-29 | Hokuriku Seiyaku Co. Ltd | Thiourea derivatives |
| CZ20001613A3 (cs) * | 1997-11-07 | 2001-12-12 | Pharmacia & Upjohn Company | Způsob výroby oxazolidinonů |
| DE19802239A1 (de) * | 1998-01-22 | 1999-07-29 | Bayer Ag | Neue mit Bicyclen substituierte Oxazolidinone |
| AU764184B2 (en) | 1998-01-23 | 2003-08-14 | Pharmacia & Upjohn Company | Oxazolidinone combinatorial libraries, compositions and methods of preparation |
| CN1311787A (zh) * | 1998-06-05 | 2001-09-05 | 阿斯特拉曾尼卡有限公司 | 噁唑烷酮衍生物、其制备方法以及含有它们的药物组合物 |
| GB9821938D0 (en) | 1998-10-09 | 1998-12-02 | Zeneca Ltd | Chemical compounds |
| JP2000204084A (ja) * | 1998-11-11 | 2000-07-25 | Hokuriku Seiyaku Co Ltd | チオカルバミド酸誘導体 |
| WO2000029409A1 (fr) * | 1998-11-17 | 2000-05-25 | Bayer Aktiengesellschaft | Nouveaux derives d'oxazolidone substitues par un heterocyclyle |
| WO2000029396A1 (fr) * | 1998-11-17 | 2000-05-25 | Bayer Aktiengesellschaft | Nouveaux derives de phenyloxazolidone substitues |
| EP1008590B1 (fr) | 1998-12-07 | 2006-10-11 | Takasago International Corporation | Procédé pour la préparation de derivés d'oxazolidinone optiquement actifs |
| ATE246189T1 (de) * | 1999-05-27 | 2003-08-15 | Upjohn Co | Bizyklische oxazolidinone als antibakterielle mittel |
| IL147503A0 (en) | 1999-07-28 | 2002-08-14 | Upjohn Co | Oxazolidinone compounds and methods of preparation and use thereof |
| US6413981B1 (en) | 1999-08-12 | 2002-07-02 | Ortho-Mcneil Pharamceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| US6608081B2 (en) * | 1999-08-12 | 2003-08-19 | Ortho-Mcneil Pharmaceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
| US6297242B1 (en) | 1999-08-12 | 2001-10-02 | Ortho-Mcneil Pharmaceutical, Inc. | N-substituted amidine and guanidine oxazolidinone antibacterials and methods of use thereof |
| GB9928568D0 (en) | 1999-12-03 | 2000-02-02 | Zeneca Ltd | Chemical compounds |
| US6518285B2 (en) | 1999-12-21 | 2003-02-11 | Ortho Mcneil Pharmaceutical, Inc. | Piperidinyloxy and pyrrolidinyloxy oxazolidinone antibacterials |
| DE29923691U1 (de) | 1999-12-23 | 2001-01-18 | Wilfer, Hans-Peter, 08258 Markneukirchen | Behältnis für Musikinstrumente, insbesondere für Gitarren |
| DE19962924A1 (de) | 1999-12-24 | 2001-07-05 | Bayer Ag | Substituierte Oxazolidinone und ihre Verwendung |
| KR100355345B1 (ko) * | 2000-01-21 | 2002-10-12 | 한국과학기술연구원 | 티오펜환을 함유한 신규한 옥사졸리디논 유도체, 그의 제조방법 및 조성물 |
| MY127336A (en) * | 2000-03-22 | 2006-11-30 | Upjohn Co | Container for linezolid iv solution |
| US6514529B2 (en) | 2000-03-22 | 2003-02-04 | Pharmacia & Upjohn Company | Oxazolidinone tablet formulation |
| PE20011124A1 (es) | 2000-03-31 | 2001-10-28 | Upjohn Co | Nuevos agentes antibacterianos de benzosultam oxazolidinona |
| GB0009803D0 (en) * | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
| WO2002002095A2 (fr) | 2000-06-30 | 2002-01-10 | Pharmacia & Upjohn Company | Composition et techniques de traitement d'infections bacteriennes |
| PE20030044A1 (es) * | 2000-11-17 | 2003-02-09 | Upjohn Co | Isoxazolinonas biciclicas de formula i |
| US6951863B2 (en) * | 2001-02-07 | 2005-10-04 | Ortho-Mcneil Pharmaceutical, Inc. | Pyridoarylphenly oxazolidinone antibacterials, and related compositions and methods |
| DE10129725A1 (de) | 2001-06-20 | 2003-01-02 | Bayer Ag | Kombinationstherapie substituierter Oxazolidinone |
| TW200302095A (en) * | 2002-01-25 | 2003-08-01 | Upjohn Co | Oxazolidinone cotherapy |
| AR038536A1 (es) * | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
| US7141588B2 (en) * | 2002-02-25 | 2006-11-28 | Pfizer, Inc. | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
| BR0308806A (pt) * | 2002-03-29 | 2005-01-04 | Upjohn Co | Uso de oxazolidinonas para tratar infecções do tipo pé diabético |
| ES2258234T3 (es) * | 2002-08-12 | 2006-08-16 | PHARMACIA & UPJOHN COMPANY LLC | N-aril-2-oxazolidinonas y sus derivados. |
| WO2004026848A1 (fr) * | 2002-09-20 | 2004-04-01 | Lupin Limited | Derives d'oxazolidinone, leur procede de preparation et leur utilisation comme agents antimycobacterients |
| US7091196B2 (en) * | 2002-09-26 | 2006-08-15 | Rib-X Pharmaceuticals, Inc. | Bifunctional heterocyclic compounds and methods of making and using same |
| US7141570B2 (en) * | 2002-11-21 | 2006-11-28 | Pharmacia & Upjohn Company | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
| DE10300111A1 (de) | 2003-01-07 | 2004-07-15 | Bayer Healthcare Ag | Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid |
| BRPI0407252A (pt) * | 2003-02-07 | 2006-01-31 | Warner Lambert Co | Agentes antibacterianos. |
| MXPA05007937A (es) * | 2003-02-07 | 2005-09-30 | Warner Lambert Co | Agentes antibacterianos. |
| US7012088B2 (en) * | 2003-02-24 | 2006-03-14 | Pharmacia & Upjohn Company | Indolone oxazolidinones and derivatives thereof |
| US20040204463A1 (en) * | 2003-04-01 | 2004-10-14 | Harris Christina Renee | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
| CA2536480A1 (fr) * | 2003-08-25 | 2005-03-03 | Warner-Lambert Company Llc | Nouveaux composes d'aryloxazolidinone antimicrobiens |
| US7304050B2 (en) * | 2003-09-16 | 2007-12-04 | Pfizer Inc. | Antibacterial agents |
| DE10355461A1 (de) | 2003-11-27 | 2005-06-23 | Bayer Healthcare Ag | Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung |
| WO2005082900A2 (fr) * | 2004-01-28 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Amidoxines d'oxazolidinone utilisees en tant qu'agents antibacteriens |
| WO2005082897A1 (fr) * | 2004-01-28 | 2005-09-09 | Pharmacia & Upjohn Company Llc | Agents antibacteriens oxazolidinone |
| JP5383037B2 (ja) | 2004-02-27 | 2014-01-08 | リブ−エックス ファーマシューティカルズ，インコーポレイテッド | 大環状化合物およびそれらを製造し使用する方法 |
| DE102004062475A1 (de) * | 2004-12-24 | 2006-07-06 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung |
| EP1685841A1 (fr) | 2005-01-31 | 2006-08-02 | Bayer Health Care Aktiengesellschaft | Prevention et traitement de troubles thromboemboliques |
| AU2006231919A1 (en) | 2005-04-06 | 2006-10-12 | Pharmacia & Upjohn Company Llc | 7-fluoro-1,3-dihydro-indol-2-one oxazolidinones as antibacterial agents |
| WO2007025098A2 (fr) * | 2005-08-24 | 2007-03-01 | Rib-X Pharmaceuticals, Inc. | Composes de triazole et preparation et utilisation de ces composes |
| US8470985B2 (en) * | 2005-08-24 | 2013-06-25 | Rib-X Pharmaceuticals, Inc. | Triazole compounds and methods of making and using the same |
| DE102005045518A1 (de) | 2005-09-23 | 2007-03-29 | Bayer Healthcare Ag | 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung |
| DE102005047558A1 (de) * | 2005-10-04 | 2008-02-07 | Bayer Healthcare Ag | Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen |
| SG166126A1 (en) | 2005-10-04 | 2010-11-29 | Bayer Schering Pharma Ag | Novel polymorphous form and the amorphous form of 5-chloro-n-({(5s)-2-oxo- 3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidine-5-yl}-methyl)-2-thiophene carboxamide |
| DE102005047561A1 (de) | 2005-10-04 | 2007-04-05 | Bayer Healthcare Ag | Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung |
| US7652018B2 (en) * | 2006-08-15 | 2010-01-26 | Wyeth Llc | Imidazolidin-2-one derivatives useful as PR modulators |
| US7538107B2 (en) | 2006-08-15 | 2009-05-26 | Wyeth | Oxazinan-2-one derivatives useful as PR modulators |
| US7649007B2 (en) * | 2006-08-15 | 2010-01-19 | Wyeth Llc | Oxazolidine derivatives as PR modulators |
| TW200815428A (en) | 2006-08-15 | 2008-04-01 | Wyeth Corp | Oxazolidone derivatives as PR modulators |
| DE102006051625A1 (de) * | 2006-11-02 | 2008-05-08 | Bayer Materialscience Ag | Kombinationstherapie substituierter Oxazolidinone |
| WO2008143649A2 (fr) * | 2006-12-04 | 2008-11-27 | Dr. Reddy's Laboratories Limited | Nouveaux composés oxazolidinones comme agents anti-infectieux |
| JP5404652B2 (ja) * | 2008-02-22 | 2014-02-05 | アクテリオン ファーマシューティカルズ リミテッド | オキサゾリジノン誘導体 |
| WO2018170664A1 (fr) * | 2017-03-20 | 2018-09-27 | Merck Sharp & Dohme Corp. | Composés d'oxazolidinone et leurs procédés d'utilisation en tant qu'agents antibactériens |
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| DE4425613A1 (de) | 1994-07-20 | 1996-01-25 | Bayer Ag | 5-gliedrige Heteroaryl-oxazolidinone |
| DE19514313A1 (de) * | 1994-08-03 | 1996-02-08 | Bayer Ag | Benzoxazolyl- und Benzothiazolyloxazolidinone |
| HRP960159A2 (en) | 1995-04-21 | 1997-08-31 | Bayer Ag | Benzocyclopentane oxazolidinones containing heteroatoms |
-
1996
- 1996-02-06 DE DE19604223A patent/DE19604223A1/de not_active Withdrawn
-
1997
- 1997-01-27 HR HR19604223.2A patent/HRP970048A2/hr not_active Application Discontinuation
- 1997-01-31 EP EP97101509A patent/EP0789025B1/fr not_active Expired - Lifetime
- 1997-01-31 DK DK97101509T patent/DK0789025T3/da active
- 1997-01-31 ES ES97101509T patent/ES2157027T3/es not_active Expired - Lifetime
- 1997-01-31 SI SI9730110T patent/SI0789025T1/xx unknown
- 1997-01-31 DE DE59703261T patent/DE59703261D1/de not_active Expired - Fee Related
- 1997-01-31 AT AT97101509T patent/ATE200285T1/de not_active IP Right Cessation
- 1997-01-31 PT PT97101509T patent/PT789025E/pt unknown
- 1997-02-03 US US08/794,034 patent/US5792765A/en not_active Expired - Fee Related
- 1997-02-03 IL IL12012597A patent/IL120125A0/xx unknown
- 1997-02-03 NZ NZ314179A patent/NZ314179A/xx unknown
- 1997-02-04 ID IDP970341A patent/ID15881A/id unknown
- 1997-02-04 MX MX9700886A patent/MX9700886A/es unknown
- 1997-02-04 TW TW086101259A patent/TW350845B/zh active
- 1997-02-04 BG BG101193A patent/BG101193A/xx unknown
- 1997-02-04 AR ARP970100439A patent/AR005703A1/es unknown
- 1997-02-04 TN TNTNSN97032A patent/TNSN97032A1/fr unknown
- 1997-02-04 AU AU12516/97A patent/AU1251697A/en not_active Abandoned
- 1997-02-04 PL PL97318277A patent/PL318277A1/xx unknown
- 1997-02-05 NO NO970511A patent/NO970511L/no unknown
- 1997-02-05 SG SG1997000259A patent/SG50791A1/en unknown
- 1997-02-05 CA CA002196862A patent/CA2196862A1/fr not_active Abandoned
- 1997-02-05 CZ CZ97340A patent/CZ34097A3/cs unknown
- 1997-02-05 HU HU9700358A patent/HUP9700358A3/hu unknown
- 1997-02-05 ZA ZA9700927A patent/ZA97927B/xx unknown
- 1997-02-05 TR TR97/00092A patent/TR199700092A2/xx unknown
- 1997-02-05 SK SK158-97A patent/SK15897A3/sk unknown
- 1997-02-05 EE EE9700043A patent/EE9700043A/xx unknown
- 1997-02-05 KR KR1019970003610A patent/KR970061888A/ko not_active Application Discontinuation
- 1997-02-05 YU YU4397A patent/YU4397A/sh unknown
- 1997-02-05 BR BR9700885A patent/BR9700885A/pt not_active Application Discontinuation
- 1997-02-06 CN CN97101879A patent/CN1160051A/zh active Pending
- 1997-02-06 CO CO97006151A patent/CO4560411A1/es unknown
- 1997-02-06 JP JP9036908A patent/JPH09316073A/ja active Pending
- 1997-02-06 SV SV1997000009A patent/SV1997000009A/es unknown
-
2001
- 2001-06-08 GR GR20010400867T patent/GR3036015T3/el not_active IP Right Cessation
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