TW200602058A - Fused pyrazolo pyrimidine and pyrazolo pyrimidinone derivatives - Google Patents
Fused pyrazolo pyrimidine and pyrazolo pyrimidinone derivativesInfo
- Publication number
- TW200602058A TW200602058A TW094105812A TW94105812A TW200602058A TW 200602058 A TW200602058 A TW 200602058A TW 094105812 A TW094105812 A TW 094105812A TW 94105812 A TW94105812 A TW 94105812A TW 200602058 A TW200602058 A TW 200602058A
- Authority
- TW
- Taiwan
- Prior art keywords
- pyrazolo
- fused
- pyrimidine
- pyrimidinone derivatives
- compounds
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
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- A61P11/16—Central respiratory analeptics
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- A—HUMAN NECESSITIES
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- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Virology (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Oncology (AREA)
- Pulmonology (AREA)
- Communicable Diseases (AREA)
- Diabetes (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Neurosurgery (AREA)
- Dermatology (AREA)
- Molecular Biology (AREA)
- Ophthalmology & Optometry (AREA)
- Cardiology (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Endocrinology (AREA)
- Hematology (AREA)
- Hospice & Palliative Care (AREA)
- Toxicology (AREA)
- Emergency Medicine (AREA)
- Psychiatry (AREA)
- Obesity (AREA)
- AIDS & HIV (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US54858304P | 2004-02-27 | 2004-02-27 |
Publications (1)
Publication Number | Publication Date |
---|---|
TW200602058A true TW200602058A (en) | 2006-01-16 |
Family
ID=34919377
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TW094105812A TW200602058A (en) | 2004-02-27 | 2005-02-25 | Fused pyrazolo pyrimidine and pyrazolo pyrimidinone derivatives |
Country Status (16)
Country | Link |
---|---|
US (1) | US7435731B2 (zh) |
EP (1) | EP1737865A1 (zh) |
JP (1) | JP2007523938A (zh) |
KR (1) | KR100843526B1 (zh) |
CN (1) | CN1926139A (zh) |
AR (1) | AR048302A1 (zh) |
AU (1) | AU2005219525B2 (zh) |
BR (1) | BRPI0508036A (zh) |
CA (1) | CA2557575A1 (zh) |
CO (1) | CO5721008A2 (zh) |
IL (1) | IL177569A (zh) |
NO (1) | NO20064015L (zh) |
RU (1) | RU2006134020A (zh) |
TW (1) | TW200602058A (zh) |
WO (1) | WO2005085249A1 (zh) |
ZA (1) | ZA200606921B (zh) |
Families Citing this family (101)
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US8076338B2 (en) * | 2004-04-23 | 2011-12-13 | Exelixis, Inc. | Kinase modulators and methods of use |
AU2005271669A1 (en) * | 2004-08-03 | 2006-02-16 | Merck & Co., Inc. | 1,3-disubstituted heteroaryl NMDA/NR2B antagonists |
WO2006068760A2 (en) | 2004-11-19 | 2006-06-29 | The Regents Of The University Of California | Anti-inflammatory pyrazolopyrimidines |
US20060122185A1 (en) | 2004-11-22 | 2006-06-08 | Jeremy Green | Bicyclic inhibitors of Rho kinase |
GB0427604D0 (en) * | 2004-12-16 | 2005-01-19 | Novartis Ag | Organic compounds |
WO2006071819A1 (en) * | 2004-12-28 | 2006-07-06 | Exelixis, Inc. | [1h-pyrazolo[3, 4-d]pyrimidin-4-yl]-piperidine or -piperazine compounds as serine-theoronine kinase modulators (p70s6k, atk1 and atk2) for the treatment of immunological, inflammatory and proliferative diseases |
AR057455A1 (es) * | 2005-07-22 | 2007-12-05 | Merck & Co Inc | Inhibidores de la transcriptasa reversa de vih y composicion farmaceutica |
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BRPI0615272A2 (pt) * | 2005-08-25 | 2009-08-04 | Hoffmann La Roche | inibidores de p38 map kinase e métodos para uso dos mesmos |
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US7585868B2 (en) | 2006-04-04 | 2009-09-08 | The Regents Of The University Of California | Substituted pyrazolo[3,4-D]pyrimidines as kinase antagonists |
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TW200831085A (en) * | 2006-12-13 | 2008-08-01 | Merck & Co Inc | Non-nucleoside reverse transcriptase inhibitors |
WO2008074676A1 (en) * | 2006-12-19 | 2008-06-26 | F. Hoffmann-La Roche Ag | Pyrazolo [3, 4 -d] pyrimidine p38 map kinase inhibitors |
WO2008081928A1 (ja) | 2006-12-28 | 2008-07-10 | Taisho Pharmaceutical Co., Ltd. | ピラゾロピリミジン化合物 |
US8309138B2 (en) | 2007-02-16 | 2012-11-13 | Aska Pharmaceutical Co., Ltd. | Pharmaceutical composition comprising microparticle oily suspension |
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US20110160232A1 (en) | 2007-10-04 | 2011-06-30 | Pingda Ren | Certain chemical entities and therapeutic uses thereof |
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- 2005-02-24 EP EP05707608A patent/EP1737865A1/en not_active Withdrawn
- 2005-02-24 BR BRPI0508036-3A patent/BRPI0508036A/pt not_active IP Right Cessation
- 2005-02-24 RU RU2006134020/04A patent/RU2006134020A/ru not_active Application Discontinuation
- 2005-02-24 CA CA002557575A patent/CA2557575A1/en not_active Abandoned
- 2005-02-24 KR KR1020067017111A patent/KR100843526B1/ko not_active IP Right Cessation
- 2005-02-24 CN CNA2005800063442A patent/CN1926139A/zh active Pending
- 2005-02-24 JP JP2007500149A patent/JP2007523938A/ja active Pending
- 2005-02-24 WO PCT/EP2005/001936 patent/WO2005085249A1/en active Application Filing
- 2005-02-25 TW TW094105812A patent/TW200602058A/zh unknown
- 2005-02-25 US US11/067,336 patent/US7435731B2/en not_active Expired - Fee Related
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CA2557575A1 (en) | 2005-09-15 |
KR20060114019A (ko) | 2006-11-03 |
AR048302A1 (es) | 2006-04-19 |
BRPI0508036A (pt) | 2007-07-17 |
AU2005219525A1 (en) | 2005-09-15 |
AU2005219525B2 (en) | 2011-08-18 |
IL177569A (en) | 2012-08-30 |
CO5721008A2 (es) | 2007-01-31 |
US20050197340A1 (en) | 2005-09-08 |
US7435731B2 (en) | 2008-10-14 |
NO20064015L (no) | 2006-11-23 |
WO2005085249A1 (en) | 2005-09-15 |
ZA200606921B (en) | 2008-08-27 |
IL177569A0 (en) | 2006-12-10 |
JP2007523938A (ja) | 2007-08-23 |
KR100843526B1 (ko) | 2008-07-03 |
EP1737865A1 (en) | 2007-01-03 |
RU2006134020A (ru) | 2008-04-10 |
CN1926139A (zh) | 2007-03-07 |
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