TR201821285T4 - CCR3 antagonisti içeren farmasötik formülasyonlar. - Google Patents

CCR3 antagonisti içeren farmasötik formülasyonlar. Download PDF

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Publication number
TR201821285T4
TR201821285T4 TR2018/21285T TR201821285T TR201821285T4 TR 201821285 T4 TR201821285 T4 TR 201821285T4 TR 2018/21285 T TR2018/21285 T TR 2018/21285T TR 201821285 T TR201821285 T TR 201821285T TR 201821285 T4 TR201821285 T4 TR 201821285T4
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TR
Turkey
Prior art keywords
tablet
tablets
solvent
lubricant
premix
Prior art date
Application number
TR2018/21285T
Other languages
English (en)
Turkish (tr)
Inventor
Fetscher Alfred
Matthias Scher Jochen
Original Assignee
Alkahest Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49292482&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TR201821285(T4) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Alkahest Inc filed Critical Alkahest Inc
Publication of TR201821285T4 publication Critical patent/TR201821285T4/tr

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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4545Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring hetero atom, e.g. pipamperone, anabasine
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    • A61K9/0012Galenical forms characterised by the site of application
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    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605Excipients; Inactive ingredients
    • A61K9/1617Organic compounds, e.g. phospholipids, fats
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  • Transplantation (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TR2018/21285T 2012-04-04 2013-04-02 CCR3 antagonisti içeren farmasötik formülasyonlar. TR201821285T4 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP12163078 2012-04-04

Publications (1)

Publication Number Publication Date
TR201821285T4 true TR201821285T4 (tr) 2019-01-21

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Application Number Title Priority Date Filing Date
TR2018/21285T TR201821285T4 (tr) 2012-04-04 2013-04-02 CCR3 antagonisti içeren farmasötik formülasyonlar.

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Families Citing this family (12)

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US8278302B2 (en) 2009-04-08 2012-10-02 Boehringer Ingelheim International Gmbh Substituted piperidines as CCR3 antagonists
UA109290C2 (uk) 2010-10-07 2015-08-10 Спільні кристали і солі інгібіторів ccr3
US8680280B2 (en) 2012-04-02 2014-03-25 Boehringer Ingelheim International Gmbh Process for the manufacturing of CRR inhibitors
US20130261153A1 (en) * 2012-04-03 2013-10-03 Boehringer Ingelheim International Gmbh Use of ccr3-inhibitors
US10213421B2 (en) * 2012-04-04 2019-02-26 Alkahest, Inc. Pharmaceutical formulations comprising CCR3 antagonists
UA125658C2 (uk) 2017-04-05 2022-05-11 Алкахест Інк. Спосіб та композиція для лікування захворювання, пов'язаного з сітківкою ока, з використанням інгібітора ccr3
JP2020513005A (ja) * 2017-04-05 2020-04-30 アルカヘスト,インコーポレイテッド Ccr3阻害剤を用いて、加齢性機能障害を治療するための方法及び組成物
US20190111042A1 (en) * 2017-10-13 2019-04-18 Alkahest, Inc. Methods and Compositions for Treating Pruritus, Xerosis, and Associated Disease Using CCR-Inhibitors
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