TR200000805T2 - Antibakteriyel etki gösteren 3'-N degişimli 6-0 ikameli eritromisin ketolid türevleri. - Google Patents
Antibakteriyel etki gösteren 3'-N degişimli 6-0 ikameli eritromisin ketolid türevleri.Info
- Publication number
- TR200000805T2 TR200000805T2 TR2000/00805T TR200000805T TR200000805T2 TR 200000805 T2 TR200000805 T2 TR 200000805T2 TR 2000/00805 T TR2000/00805 T TR 2000/00805T TR 200000805 T TR200000805 T TR 200000805T TR 200000805 T2 TR200000805 T2 TR 200000805T2
- Authority
- TR
- Turkey
- Prior art keywords
- ketolid
- erythromycin
- derivatives
- change
- antibacterial effect
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Engineering & Computer Science (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
Bulus antibakteriyel aktiviteye sahip 3'-N, ile degisiklige ugratilmis yeni 6-0 ikameli eritromisin ketolid bilesikleri ve bunlarin farmasötik olarak kabul edilebilir tuzlari ve esterleriyle, böyle bir bilesigin terapötik olarak etkili bir miktarini ve bir farmasötik olarak kabul edilebilir tasiyici madde içeren farmasötik bilesimlerle ve memelilerde bakteriyel enfeksiyonlarin tedavisi için bir yöntemle ilgili olup bu yöntem söz konusu memeliye yukarida açiklanan bir bilesigin terapötik olarak etkili bir miktarinin uygulanmasini içermektedir.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US94087197A | 1997-09-30 | 1997-09-30 | |
US13312198A | 1998-08-12 | 1998-08-12 |
Publications (1)
Publication Number | Publication Date |
---|---|
TR200000805T2 true TR200000805T2 (tr) | 2000-10-23 |
Family
ID=26831064
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2000/00805T TR200000805T2 (tr) | 1997-09-30 | 1998-09-16 | Antibakteriyel etki gösteren 3'-N degişimli 6-0 ikameli eritromisin ketolid türevleri. |
Country Status (22)
Country | Link |
---|---|
EP (1) | EP1025114B1 (tr) |
JP (1) | JP2001518476A (tr) |
KR (1) | KR20010030807A (tr) |
CN (1) | CN1271363A (tr) |
AR (1) | AR015727A1 (tr) |
AT (1) | ATE260293T1 (tr) |
AU (1) | AU737310B2 (tr) |
BG (1) | BG104340A (tr) |
BR (1) | BR9812577A (tr) |
CA (1) | CA2303930A1 (tr) |
CO (1) | CO4990958A1 (tr) |
DE (1) | DE69821964T2 (tr) |
DK (1) | DK1025114T3 (tr) |
ES (1) | ES2217579T3 (tr) |
HU (1) | HUP0004579A3 (tr) |
IL (1) | IL134608A0 (tr) |
NO (1) | NO20001439L (tr) |
PL (1) | PL339575A1 (tr) |
PT (1) | PT1025114E (tr) |
SK (1) | SK4562000A3 (tr) |
TR (1) | TR200000805T2 (tr) |
WO (1) | WO1999016779A1 (tr) |
Families Citing this family (19)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP4573925B2 (ja) * | 1998-07-09 | 2010-11-04 | アベンティス・ファーマ・ソシエテ・アノニム | 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用 |
US6395710B1 (en) * | 1999-04-16 | 2002-05-28 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
US6355620B1 (en) * | 1999-05-14 | 2002-03-12 | Abbott Laboratories | C-2 modified erythromycin derivatives |
US6437106B1 (en) * | 1999-06-24 | 2002-08-20 | Abbott Laboratories | Process for preparing 6-o-substituted erythromycin derivatives |
CN1197870C (zh) * | 2000-08-14 | 2005-04-20 | 大正制药株式会社 | 一种红霉素衍生物的制备方法及其中间体 |
AU2002230386A1 (en) * | 2000-09-25 | 2002-04-29 | Kosan Biosciences, Inc. | Sixteen-membered macrolide compounds |
ITMI20021726A1 (it) | 2002-08-01 | 2004-02-02 | Zambon Spa | Macrolidi ad attivita' antiinfiammatoria. |
AR043050A1 (es) | 2002-09-26 | 2005-07-13 | Rib X Pharmaceuticals Inc | Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos |
CN108101948A (zh) * | 2004-02-27 | 2018-06-01 | 瑞伯-X医药品有限公司 | 大环化合物以及其制作和使用方法 |
EP2716647A3 (en) | 2004-02-27 | 2014-08-20 | Rib-X Pharmaceuticals, Inc. | Macrocyclic compounds and methods of making and using the same |
EP1794171A2 (en) * | 2004-07-28 | 2007-06-13 | Ranbaxy Laboratories, Ltd. | Ketolide derivatives as antibacterial agents |
WO2006046112A2 (en) * | 2004-10-25 | 2006-05-04 | Ranbaxy Laboratories Limited | Ketolide derivatives as antibacterial agents |
WO2006129257A2 (en) * | 2005-05-30 | 2006-12-07 | Ranbaxy Laboratories Limited | Ketolide derivatives as antibacterial agents |
EP1934237A2 (en) | 2005-08-24 | 2008-06-25 | Rib-X Pharmaceuticals, Inc. | Triazole compounds and methods of making and using the same |
JP5395432B2 (ja) * | 2005-08-24 | 2014-01-22 | リブ−エックス ファーマシューティカルズ,インコーポレイテッド | トリアゾール化合物ならびにこれを作製する方法および使用する方法 |
EP1957508A2 (en) * | 2005-11-23 | 2008-08-20 | Ranbaxy Laboratories Limited | Ketolide derivatives as antibacterial agents |
JP5126685B2 (ja) * | 2006-05-01 | 2013-01-23 | 大正製薬株式会社 | マクロライド誘導体 |
WO2008099368A1 (en) * | 2007-02-15 | 2008-08-21 | Ranbaxy Laboratories Limited | Macrolide derivatives as antibacterial agents |
WO2008111020A2 (en) * | 2007-03-14 | 2008-09-18 | Ranbaxy Laboratories Limited | Macrolide derivatives as antibacterial agents |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL99995A (en) * | 1990-11-21 | 1997-11-20 | Roussel Uclaf | Erythromycin derivatives, their preparation and pharmaceutical compositions containing them |
WO1997017356A1 (en) * | 1995-11-08 | 1997-05-15 | Abbott Laboratories | Tricyclic erythromycin derivatives |
-
1998
- 1998-09-16 SK SK456-2000A patent/SK4562000A3/sk unknown
- 1998-09-16 EP EP98946087A patent/EP1025114B1/en not_active Expired - Lifetime
- 1998-09-16 DE DE69821964T patent/DE69821964T2/de not_active Expired - Fee Related
- 1998-09-16 PL PL98339575A patent/PL339575A1/xx unknown
- 1998-09-16 HU HU0004579A patent/HUP0004579A3/hu unknown
- 1998-09-16 IL IL13460898A patent/IL134608A0/xx unknown
- 1998-09-16 ES ES98946087T patent/ES2217579T3/es not_active Expired - Lifetime
- 1998-09-16 PT PT98946087T patent/PT1025114E/pt unknown
- 1998-09-16 AT AT98946087T patent/ATE260293T1/de not_active IP Right Cessation
- 1998-09-16 CN CN98809567A patent/CN1271363A/zh active Pending
- 1998-09-16 AU AU93176/98A patent/AU737310B2/en not_active Ceased
- 1998-09-16 WO PCT/US1998/019311 patent/WO1999016779A1/en active IP Right Grant
- 1998-09-16 KR KR1020007003408A patent/KR20010030807A/ko not_active Application Discontinuation
- 1998-09-16 DK DK98946087T patent/DK1025114T3/da active
- 1998-09-16 BR BR9812577-0A patent/BR9812577A/pt not_active IP Right Cessation
- 1998-09-16 TR TR2000/00805T patent/TR200000805T2/tr unknown
- 1998-09-16 CA CA002303930A patent/CA2303930A1/en not_active Abandoned
- 1998-09-16 JP JP2000513861A patent/JP2001518476A/ja not_active Withdrawn
- 1998-09-28 CO CO98056259A patent/CO4990958A1/es unknown
- 1998-09-29 AR ARP980104856A patent/AR015727A1/es unknown
-
2000
- 2000-03-20 NO NO20001439A patent/NO20001439L/no not_active Application Discontinuation
- 2000-04-14 BG BG104340A patent/BG104340A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
NO20001439L (no) | 2000-05-29 |
CN1271363A (zh) | 2000-10-25 |
AU9317698A (en) | 1999-04-23 |
BR9812577A (pt) | 2000-10-17 |
NO20001439D0 (no) | 2000-03-20 |
HUP0004579A3 (en) | 2001-11-28 |
JP2001518476A (ja) | 2001-10-16 |
IL134608A0 (en) | 2001-04-30 |
ES2217579T3 (es) | 2004-11-01 |
ATE260293T1 (de) | 2004-03-15 |
CA2303930A1 (en) | 1999-04-08 |
SK4562000A3 (en) | 2000-09-12 |
EP1025114B1 (en) | 2004-02-25 |
EP1025114A1 (en) | 2000-08-09 |
KR20010030807A (ko) | 2001-04-16 |
HUP0004579A2 (hu) | 2001-05-28 |
AR015727A1 (es) | 2001-05-16 |
WO1999016779A1 (en) | 1999-04-08 |
CO4990958A1 (es) | 2000-12-26 |
BG104340A (en) | 2001-01-31 |
DE69821964T2 (de) | 2004-12-30 |
PT1025114E (pt) | 2004-07-30 |
PL339575A1 (en) | 2000-12-18 |
AU737310B2 (en) | 2001-08-16 |
DE69821964D1 (de) | 2004-04-01 |
DK1025114T3 (da) | 2004-07-05 |
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