TR199902934T2 - S-Omeprazolün yeni yapisi. - Google Patents

S-Omeprazolün yeni yapisi.

Info

Publication number
TR199902934T2
TR199902934T2 TR1999/02934T TR9902934T TR199902934T2 TR 199902934 T2 TR199902934 T2 TR 199902934T2 TR 1999/02934 T TR1999/02934 T TR 1999/02934T TR 9902934 T TR9902934 T TR 9902934T TR 199902934 T2 TR199902934 T2 TR 199902934T2
Authority
TR
Turkey
Prior art keywords
omeprazole
refers
new structure
enantiomer
methoxy
Prior art date
Application number
TR1999/02934T
Other languages
English (en)
Inventor
Cotton Hanna
Kronstr�m Anders
Mattson Anders
M�ller Eva
Original Assignee
Astra Aktiebolag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20407186&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TR199902934(T2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astra Aktiebolag filed Critical Astra Aktiebolag
Publication of TR199902934T2 publication Critical patent/TR199902934T2/tr

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Abstract

Bu bulus, 5-metoksi-2-[[(4-metoksi-3, 5-dimetil-2-pridinil)-metil]sülfinil]-1H-benzimidazol'ün (-) enantiomeri, yani S-omeprazol'ün yeni yapisina iliskindir. Daha özele inilirse, omeprazol trihidrat'in S-enantiomerinin magnezyum tuzunun yeni bir yapisina deginir. Bu bulus ayni zamanda, böyle bir yapiya sahip magnezyum tuzu ve bu tuzu içeren ilaç bilesimleri hazirlamak için kullanilan proseslere deginir. Bunun da ötesinde bulus, prosesteki ara ürünlere de deginir.
TR1999/02934T 1997-05-30 1998-05-25 S-Omeprazolün yeni yapisi. TR199902934T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE9702065A SE510650C2 (sv) 1997-05-30 1997-05-30 Ny förening

Publications (1)

Publication Number Publication Date
TR199902934T2 true TR199902934T2 (tr) 2000-04-21

Family

ID=20407186

Family Applications (1)

Application Number Title Priority Date Filing Date
TR1999/02934T TR199902934T2 (tr) 1997-05-30 1998-05-25 S-Omeprazolün yeni yapisi.

Country Status (44)

Country Link
US (6) US6369085B1 (tr)
EP (2) EP1273581B1 (tr)
JP (2) JP4002303B2 (tr)
KR (2) KR100540720B1 (tr)
CN (1) CN1161351C (tr)
AR (2) AR012717A1 (tr)
AT (2) ATE239011T1 (tr)
AU (1) AU722839B2 (tr)
BR (1) BR9809509A (tr)
CA (2) CA2290963C (tr)
CY (1) CY2012029I2 (tr)
CZ (1) CZ297585B6 (tr)
DE (3) DE69829511T2 (tr)
DK (2) DK0984957T3 (tr)
DZ (1) DZ2495A1 (tr)
EE (1) EE03875B1 (tr)
EG (1) EG24291A (tr)
ES (2) ES2236407T3 (tr)
HK (2) HK1025962A1 (tr)
HR (1) HRP980263B1 (tr)
HU (1) HU225987B1 (tr)
ID (1) ID29306A (tr)
IL (1) IL132947A0 (tr)
IS (2) IS2142B (tr)
LU (2) LU91871I2 (tr)
MA (1) MA26500A1 (tr)
ME (3) MEP24908A (tr)
MY (2) MY120745A (tr)
NO (3) NO317518B1 (tr)
NZ (1) NZ500991A (tr)
PL (1) PL193546B1 (tr)
PT (2) PT984957E (tr)
RS (2) RS50067B (tr)
RU (1) RU2184115C2 (tr)
SA (2) SA05260296B1 (tr)
SE (1) SE510650C2 (tr)
SI (2) SI1273581T1 (tr)
SK (2) SK285137B6 (tr)
TN (1) TNSN98074A1 (tr)
TR (1) TR199902934T2 (tr)
TW (1) TW538040B (tr)
UA (1) UA60334C2 (tr)
WO (1) WO1998054171A1 (tr)
ZA (1) ZA984179B (tr)

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KR102080023B1 (ko) 2018-01-29 2020-02-21 주식회사 종근당 에스오메프라졸 및 탄산수소나트륨을 포함하는 안정한 약제학적 조성물
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KR102432084B1 (ko) 2021-11-16 2022-08-12 알리코제약(주) S-오메프라졸을 함유하는 안정성이 개선되고 소형화된 정제
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AU695966B2 (en) 1994-07-08 1998-08-27 Astrazeneca Ab Multiple unit tableted dosage form I
FR2722191B1 (fr) 1994-07-08 1996-08-23 Rhone Poulenc Rorer Sa Procede de preparation du trihydrate du (2r,3s)-3-tertbutoxycarbonylamino-2-hydroxy-3-phenylpropionate de 4-acetoxy2alpha-benzoyloxy-5beta,20epoxy-1,7beta,10beta trihydroxy-9-oxo-tax-11-en-13alpha-yle
SE504459C2 (sv) 1994-07-15 1997-02-17 Astra Ab Förfarande för framställning av substituerade sulfoxider
DK0792879T3 (da) 1994-11-14 2001-03-26 Daiichi Seiyaku Co Fremgangsmåde til fremstilling af 3-[2-[4-(3-chlor-2-methylphenyl)-1-piperzinyl]ethyl]-5,6-dimethoxy-1-(4-imidazolylmethyl)
GB9423970D0 (en) 1994-11-28 1995-01-11 Astra Ab Oxidation
SE9500422D0 (sv) 1995-02-06 1995-02-06 Astra Ab New oral pharmaceutical dosage forms
CN1042423C (zh) 1995-05-25 1999-03-10 常州市第四制药厂 奥美拉唑盐水合物及其制备方法
SE9600070D0 (sv) 1996-01-08 1996-01-08 Astra Ab New oral pharmaceutical dosage forms
SE9600072D0 (sv) 1996-01-08 1996-01-08 Astra Ab New oral formulation of two active ingredients II
SE9600071D0 (sv) 1996-01-08 1996-01-08 Astra Ab New oral formulation of two active ingredients I
US6747155B2 (en) * 1997-05-30 2004-06-08 Astrazeneca Ab Process
SE510650C2 (sv) * 1997-05-30 1999-06-14 Astra Ab Ny förening
AR057181A1 (es) 2005-11-30 2007-11-21 Astra Ab Nueva forma de dosificacion de combinacion

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