SV2009002851A - Inhibidores de la pde y combinaciones de los mismos para el tratamiento de trastornos urologicos - Google Patents

Inhibidores de la pde y combinaciones de los mismos para el tratamiento de trastornos urologicos

Info

Publication number
SV2009002851A
SV2009002851A SV2008002851A SV2008002851A SV2009002851A SV 2009002851 A SV2009002851 A SV 2009002851A SV 2008002851 A SV2008002851 A SV 2008002851A SV 2008002851 A SV2008002851 A SV 2008002851A SV 2009002851 A SV2009002851 A SV 2009002851A
Authority
SV
El Salvador
Prior art keywords
pde
treatment
combinations
urological disorders
same
Prior art date
Application number
SV2008002851A
Other languages
English (en)
Inventor
Ernest Ulbrich
Peter Sandder
Hanna Tinel
Joachim Hutter
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=37831473&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SV2009002851(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of SV2009002851A publication Critical patent/SV2009002851A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12Q—MEASURING OR TESTING PROCESSES INVOLVING ENZYMES, NUCLEIC ACIDS OR MICROORGANISMS; COMPOSITIONS OR TEST PAPERS THEREFOR; PROCESSES OF PREPARING SUCH COMPOSITIONS; CONDITION-RESPONSIVE CONTROL IN MICROBIOLOGICAL OR ENZYMOLOGICAL PROCESSES
    • C12Q1/00—Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions
    • C12Q1/34—Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions involving hydrolase
    • C12Q1/44—Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions involving hydrolase involving esterase
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/10—Drugs for disorders of the urinary system of the bladder
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • G—PHYSICS
    • G01—MEASURING; TESTING
    • G01N—INVESTIGATING OR ANALYSING MATERIALS BY DETERMINING THEIR CHEMICAL OR PHYSICAL PROPERTIES
    • G01N2500/00—Screening for compounds of potential therapeutic value

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Wood Science & Technology (AREA)
  • Urology & Nephrology (AREA)
  • Biophysics (AREA)
  • Biotechnology (AREA)
  • Diabetes (AREA)
  • Microbiology (AREA)
  • Molecular Biology (AREA)
  • Endocrinology (AREA)
  • Analytical Chemistry (AREA)
  • Biochemistry (AREA)
  • General Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Physics & Mathematics (AREA)
  • Pain & Pain Management (AREA)
  • Reproductive Health (AREA)
  • Transplantation (AREA)
  • Gynecology & Obstetrics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Epidemiology (AREA)

Abstract

LA PRESENTE INVENICIÓN PROPORCIONA COMPOSICIONES FARMACOLÓGICAS QUE COMPRENDEN INHIBIDORES DE LA PDE-5 Y LA PDE-4, SÓLOS O EN COMBINACIÓN, PARA EL TRATAMIENTO DE TRASTORNOS UROLÓGICOS QUE COMPRENDEN HIPERPLASIA PROSTÁTICA BENIGNA (HPB), SÍNTOMAS DEL TRACTO UTINARIO INFERIOR (STUI) Y EN PARTÍCULAR SÍNTOMAS IRRITATIVOS CAUSADOS POR HPB INDUCIDA POR OBSTRUCCIÓN DEL TRACTO DE SALIDA DE LA VEJIGA (OSV). LA INVENCIÓN TAMBIÉN PROPORCIONA PROCEDIMIENTOS DE DETECCIÓN PARA DICHO INHIBIDORES DE LA PDE-5 Y LA PDE-4 PARA USO, SÓLOS O EN COMBINACIÓN, EN LA PREPARACIÓN DE MEDICAMENTOS PARA EL TRATAMIENTO DE DICHOS TRASTORNOS UROLÓGICOS
SV2008002851A 2005-09-29 2008-03-26 Inhibidores de la pde y combinaciones de los mismos para el tratamiento de trastornos urologicos SV2009002851A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP05021261 2005-09-29
EP06007776 2006-04-13

Publications (1)

Publication Number Publication Date
SV2009002851A true SV2009002851A (es) 2009-01-14

Family

ID=37831473

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2008002851A SV2009002851A (es) 2005-09-29 2008-03-26 Inhibidores de la pde y combinaciones de los mismos para el tratamiento de trastornos urologicos

Country Status (23)

Country Link
US (1) US20090186896A1 (es)
EP (1) EP1931797A2 (es)
JP (1) JP2009509984A (es)
KR (1) KR20080056250A (es)
AR (1) AR057867A1 (es)
AU (1) AU2006299232A1 (es)
BR (1) BRPI0616633A2 (es)
CA (1) CA2623657A1 (es)
CR (1) CR9840A (es)
DO (1) DOP2006000207A (es)
EC (1) ECSP088311A (es)
GT (1) GT200600442A (es)
IL (1) IL190201A0 (es)
MA (1) MA29880B1 (es)
NO (1) NO20081973L (es)
PE (1) PE20070587A1 (es)
RU (1) RU2435588C2 (es)
SG (1) SG166106A1 (es)
SV (1) SV2009002851A (es)
TN (1) TNSN08147A1 (es)
TW (1) TW200804603A (es)
UY (1) UY29816A1 (es)
WO (1) WO2007039075A2 (es)

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TW201625591A (zh) 2014-09-12 2016-07-16 美國禮來大藥廠 吖丁啶基氧苯基吡咯啶化合物
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Also Published As

Publication number Publication date
TNSN08147A1 (en) 2009-07-14
UY29816A1 (es) 2007-04-30
WO2007039075A3 (en) 2007-06-21
DOP2006000207A (es) 2007-07-15
TW200804603A (en) 2008-01-16
PE20070587A1 (es) 2007-08-17
AU2006299232A1 (en) 2007-04-12
KR20080056250A (ko) 2008-06-20
RU2008116547A (ru) 2009-11-10
JP2009509984A (ja) 2009-03-12
US20090186896A1 (en) 2009-07-23
IL190201A0 (en) 2008-11-03
CR9840A (es) 2008-10-31
BRPI0616633A2 (pt) 2011-06-28
NO20081973L (no) 2008-06-20
CA2623657A1 (en) 2007-04-12
SG166106A1 (en) 2010-11-29
GT200600442A (es) 2007-05-15
AR057867A1 (es) 2007-12-26
WO2007039075A2 (en) 2007-04-12
ECSP088311A (es) 2008-06-30
RU2435588C2 (ru) 2011-12-10
EP1931797A2 (en) 2008-06-18
MA29880B1 (fr) 2008-10-03

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