SV1999000009A - Derivados de 2-(purin-9-il)-tetrahidrofuran-3,4-diol ref. pg3388/sv - Google Patents

Derivados de 2-(purin-9-il)-tetrahidrofuran-3,4-diol ref. pg3388/sv

Info

Publication number
SV1999000009A
SV1999000009A SV1999000009A SV1999000009A SV1999000009A SV 1999000009 A SV1999000009 A SV 1999000009A SV 1999000009 A SV1999000009 A SV 1999000009A SV 1999000009 A SV1999000009 A SV 1999000009A SV 1999000009 A SV1999000009 A SV 1999000009A
Authority
SV
El Salvador
Prior art keywords
tetrahidrofuran
purin
ref
diol
derivatives
Prior art date
Application number
SV1999000009A
Other languages
English (en)
Inventor
Chuen Chan
Richard Peter Charles Cousins
Brian Cox
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9802066.2A external-priority patent/GB9802066D0/en
Priority claimed from GBGB9813528.8A external-priority patent/GB9813528D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of SV1999000009A publication Critical patent/SV1999000009A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/16—Purine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
    • A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Abstract

SE PROPORCIONA DE ACUERDO CON LA INVENCION, COMPUESTOS NOVEDOSOS DE LA FORMULA (I), VER FORMULAEN DONDE R1, R2 Y R3 SON COMO SE DESCRIBEN EN LA ESPECIFICACION, A LOS PROCESOS PARA PREPARLOS, A LAS FORMULACIONES QUE LOS CONTIENEN Y A SU USO EN TERAPIA PARA EL TRATAMIENTO DE ENFERMEDADES INFLAMATORIAS.
SV1999000009A 1998-01-31 1999-01-29 Derivados de 2-(purin-9-il)-tetrahidrofuran-3,4-diol ref. pg3388/sv SV1999000009A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB9802066.2A GB9802066D0 (en) 1998-01-31 1998-01-31 Chemical compounds
GBGB9813528.8A GB9813528D0 (en) 1998-06-23 1998-06-23 Chemical compounds

Publications (1)

Publication Number Publication Date
SV1999000009A true SV1999000009A (es) 2000-09-05

Family

ID=26313042

Family Applications (1)

Application Number Title Priority Date Filing Date
SV1999000009A SV1999000009A (es) 1998-01-31 1999-01-29 Derivados de 2-(purin-9-il)-tetrahidrofuran-3,4-diol ref. pg3388/sv

Country Status (39)

Country Link
US (1) US6762170B1 (es)
EP (1) EP1051425B1 (es)
JP (1) JP2002501928A (es)
KR (1) KR20010034473A (es)
CN (1) CN1289338A (es)
AP (1) AP2000001875A0 (es)
AR (1) AR014508A1 (es)
AT (1) ATE226957T1 (es)
AU (1) AU757183B2 (es)
BG (1) BG63783B1 (es)
BR (1) BR9907270A (es)
CA (1) CA2318278A1 (es)
CO (1) CO4980872A1 (es)
DE (1) DE69903708T2 (es)
DK (1) DK1051425T3 (es)
EA (1) EA003194B1 (es)
EE (1) EE200000441A (es)
ES (1) ES2186330T3 (es)
GE (1) GEP20022839B (es)
HK (1) HK1030611A1 (es)
HR (1) HRP20000511A2 (es)
HU (1) HUP0101305A3 (es)
ID (1) ID26326A (es)
IL (1) IL137042A0 (es)
IS (1) IS5550A (es)
MA (1) MA26601A1 (es)
NO (1) NO20003867D0 (es)
NZ (1) NZ505452A (es)
OA (1) OA11447A (es)
PE (1) PE20000280A1 (es)
PL (1) PL342670A1 (es)
PT (1) PT1051425E (es)
SI (1) SI1051425T1 (es)
SK (1) SK11192000A3 (es)
SV (1) SV1999000009A (es)
TR (1) TR200002218T2 (es)
TW (1) TW434250B (es)
WO (1) WO1999038877A2 (es)
YU (1) YU44900A (es)

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Also Published As

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EA200000723A1 (ru) 2001-04-23
EA003194B1 (ru) 2003-02-27
SK11192000A3 (sk) 2001-06-11
DK1051425T3 (da) 2003-03-03
ES2186330T3 (es) 2003-05-01
HRP20000511A2 (en) 2000-12-31
HUP0101305A3 (en) 2002-08-28
YU44900A (sh) 2003-01-31
CO4980872A1 (es) 2000-11-27
BG63783B1 (bg) 2002-12-29
MA26601A1 (fr) 2004-12-20
BG104729A (en) 2001-04-30
CN1289338A (zh) 2001-03-28
ID26326A (id) 2000-12-14
PL342670A1 (en) 2001-07-02
SI1051425T1 (en) 2003-04-30
AR014508A1 (es) 2001-02-28
NZ505452A (en) 2003-01-31
AU757183B2 (en) 2003-02-06
BR9907270A (pt) 2000-10-24
US6762170B1 (en) 2004-07-13
IS5550A (is) 2000-06-27
NO20003867L (no) 2000-07-28
KR20010034473A (ko) 2001-04-25
TW434250B (en) 2001-05-16
WO1999038877A2 (en) 1999-08-05
EE200000441A (et) 2001-12-17
PE20000280A1 (es) 2000-03-28
DE69903708D1 (de) 2002-12-05
PT1051425E (pt) 2003-03-31
ATE226957T1 (de) 2002-11-15
EP1051425A2 (en) 2000-11-15
NO20003867D0 (no) 2000-07-28
CA2318278A1 (en) 1999-08-05
GEP20022839B (en) 2002-11-25
OA11447A (en) 2004-04-29
HUP0101305A2 (hu) 2002-04-29
WO1999038877A3 (en) 1999-09-30
HK1030611A1 (en) 2001-05-11
EP1051425B1 (en) 2002-10-30
IL137042A0 (en) 2001-06-14
DE69903708T2 (de) 2003-07-03
TR200002218T2 (tr) 2000-12-21
AU2719799A (en) 1999-08-16
AP2000001875A0 (en) 2000-09-30
JP2002501928A (ja) 2002-01-22

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