SV1996000109A - Nueva variante cristalina del cdch, procedimiento para su produccion y preparados farmaceuticos que la contienen ref. lea 31308-sv - Google Patents

Nueva variante cristalina del cdch, procedimiento para su produccion y preparados farmaceuticos que la contienen ref. lea 31308-sv

Info

Publication number
SV1996000109A
SV1996000109A SV1996000109A SV1996000109A SV1996000109A SV 1996000109 A SV1996000109 A SV 1996000109A SV 1996000109 A SV1996000109 A SV 1996000109A SV 1996000109 A SV1996000109 A SV 1996000109A SV 1996000109 A SV1996000109 A SV 1996000109A
Authority
SV
El Salvador
Prior art keywords
cdch
procedure
production
ref
read
Prior art date
Application number
SV1996000109A
Other languages
English (en)
Spanish (es)
Inventor
Patrick Bosche
Alfons Grunenberg
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7779831&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SV1996000109(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of SV1996000109A publication Critical patent/SV1996000109A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SV1996000109A 1995-12-12 1996-12-12 Nueva variante cristalina del cdch, procedimiento para su produccion y preparados farmaceuticos que la contienen ref. lea 31308-sv SV1996000109A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19546249A DE19546249A1 (de) 1995-12-12 1995-12-12 Neue Kristallmodifikation des 1-Cyclopropyl-7-([S,S]-2,8-diazabicyclo[4,3,0]non-8-yl)-6-fluor-1,4-dihydro-8-methoxy-4-oxo-3-chinolincarbonsäure Hydrochlorid (CDCH), Verfahren zu dessen Herstellung und diese enthaltende pharmazeutische Zubereitungen

Publications (1)

Publication Number Publication Date
SV1996000109A true SV1996000109A (es) 1997-10-23

Family

ID=7779831

Family Applications (1)

Application Number Title Priority Date Filing Date
SV1996000109A SV1996000109A (es) 1995-12-12 1996-12-12 Nueva variante cristalina del cdch, procedimiento para su produccion y preparados farmaceuticos que la contienen ref. lea 31308-sv

Country Status (42)

Country Link
US (1) US5849752A (forum.php)
EP (1) EP0780390B1 (forum.php)
JP (1) JP4104687B2 (forum.php)
KR (1) KR100525146B1 (forum.php)
CN (1) CN1061348C (forum.php)
AR (1) AR005009A1 (forum.php)
AT (1) ATE221531T1 (forum.php)
AU (1) AU708006B2 (forum.php)
BG (1) BG62258B1 (forum.php)
BR (1) BR9605968A (forum.php)
CA (1) CA2192418C (forum.php)
CO (1) CO4480105A1 (forum.php)
CU (1) CU22774A3 (forum.php)
CZ (1) CZ288657B6 (forum.php)
DE (2) DE19546249A1 (forum.php)
DK (1) DK0780390T3 (forum.php)
EE (1) EE03474B1 (forum.php)
ES (1) ES2179910T3 (forum.php)
HR (1) HRP960558B1 (forum.php)
HU (1) HU226521B1 (forum.php)
ID (1) ID22625A (forum.php)
IL (1) IL119795A (forum.php)
IN (1) IN185805B (forum.php)
MA (1) MA24342A1 (forum.php)
MY (1) MY117492A (forum.php)
NL (1) NL300109I1 (forum.php)
NO (1) NO306725B1 (forum.php)
NZ (1) NZ299905A (forum.php)
PL (1) PL184885B1 (forum.php)
PT (1) PT780390E (forum.php)
RO (1) RO119782B1 (forum.php)
RU (1) RU2162468C2 (forum.php)
SA (1) SA96170492B1 (forum.php)
SG (1) SG47201A1 (forum.php)
SI (1) SI0780390T1 (forum.php)
SK (1) SK282805B6 (forum.php)
SV (1) SV1996000109A (forum.php)
TR (1) TR199600970A2 (forum.php)
TW (1) TW411340B (forum.php)
UA (1) UA35638C2 (forum.php)
YU (1) YU49485B (forum.php)
ZA (1) ZA9610405B (forum.php)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1895233A (zh) * 1997-09-25 2007-01-17 拜尔公司 控释活性化合物的药物制剂
DE19751948A1 (de) * 1997-11-24 1999-05-27 Bayer Ag Verfahren zur Herstellung von 8-Methoxy-Chinoloncarbonsäuren
US6716830B2 (en) 1998-09-30 2004-04-06 Alcon, Inc. Ophthalmic antibiotic compositions containing moxifloxacin
US6395746B1 (en) 1998-09-30 2002-05-28 Alcon Manufacturing, Ltd. Methods of treating ophthalmic, otic and nasal infections and attendant inflammation
US6509327B1 (en) 1998-09-30 2003-01-21 Alcon Manufacturing, Ltd. Compositions and methods for treating otic, ophthalmic and nasal infections
KR100650489B1 (ko) * 1998-11-10 2006-11-28 바이엘 헬스케어 아게 목시플록사신 제약 제제
DE19854357A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Semi-Hydrochlorid von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo/4.3.0/ -nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854356A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation A von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo-/4.3.0/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19854355A1 (de) * 1998-11-25 2000-05-31 Bayer Ag Kristallmodifikation B von 8-Cyan-1-cyclopropyl-7-(1S, 6S-2,8-diazabicyclo-/4.3.O/nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE19908449A1 (de) * 1999-02-26 2000-08-31 Bayer Ag Kristallmodifikation C von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicylo-[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chino/incarbonsäure
EP1562942A1 (en) * 2002-10-31 2005-08-17 Ranbaxy Laboratories, Ltd. Amorphous moxifloxacin hydrochloride
DE602004022646D1 (de) * 2003-04-09 2009-10-01 Reddys Lab Ltd Dr Kristalline form iii von wasserfreiem moxifloxacin-hydrochlorid und ein verfahren zu seiner herstellung
WO2005012285A1 (en) * 2003-08-05 2005-02-10 Matrix Laboratories Ltd An improved process for the preparation of moxifloxacin hydrochloride
EP1685130B1 (en) * 2003-11-20 2008-12-10 CHEMI S.p.A. Polymorphs of 1-cyclopropyl-7-([s,s] - 2,8-diazadicyclo [4.3.0] non-8-yl) -6-fluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinoline carboxylic acid hydrochloride and methods for the preparation thereof
ITMI20032259A1 (it) 2003-11-20 2005-05-21 Chemi Spa Nuovo polimorfo dell'acido 1-ciclopropil-7-(s,s-2,8-diazabciclo-4.3.0-non-8-il)-6-fluoro-1,4-diidro-8-metossi-4-oxo-chinolin carbossilico cloridrato e metodi per la sua preparazione
US7491725B2 (en) 2004-02-06 2009-02-17 Bristol-Myers Squibb Company Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
DE102004015981A1 (de) * 2004-04-01 2005-10-20 Bayer Healthcare Ag Neue kirstalline Form von 8-Cyan-1-cyclopropyl-7-(1S,6S-2,8-diazabicyclo[4.3.0]nonan-8-yl)-6-fluor-1,4-dihydro-4-oxo-3-chinolincarbonsäure
DE102004063347A1 (de) * 2004-12-23 2006-07-13 Stada Arzneimittel Ag Gebrauchsfertige Gemcitabinlösungen und Gemcitabinlösungskonzentrate
WO2007033515A1 (fr) * 2005-09-21 2007-03-29 Shenzhen Tys R & D Co., Ltd. Formulation orale contenant de la moxifloxacine et son procédé de préparation
GB0612422D0 (en) * 2006-06-23 2006-08-02 Generics Uk Ltd Novel hydrate form
RU2461542C2 (ru) 2006-06-27 2012-09-20 Сандоз Аг Новый способ получения соли
ES2303768B1 (es) * 2006-09-08 2009-06-05 Quimica Sintetica, S.A. Nueva forma cristalina de moxifloxacino clorhidrato.
EP2089388B1 (en) * 2006-11-13 2014-01-29 Cipla Limited Process for the synthesis of moxifloxacin hydrochloride
EP1992626A1 (en) * 2007-05-10 2008-11-19 Sandoz AG Process for the preparation of moxifloxacin hydrochloride
EP2083010A1 (en) * 2008-01-08 2009-07-29 Chemo Ibérica, S.A. Polymorphic Forms of Moxifloxacin hydrochloride and processes for preparation thereof
EP2154137A1 (en) 2008-08-04 2010-02-17 Chemo Ibérica, S.A. Crystalline form of moxifloxacin base
EP2349220B1 (en) * 2008-10-09 2012-07-25 Abdi Ibrahim Ilac Sanayi ve Ticaret Anonim Sirketi Using of organic solvents in wet granulation of moxifloxacin
EP2342204A1 (en) * 2008-11-06 2011-07-13 Hetero Research Foundation Novel polymorph of moxifloxacin hydrochloride
EP2735307A1 (de) 2008-12-08 2014-05-28 Ratiopharm GmbH Kompaktiertes Moxifloxacin
BRPI1010981A2 (pt) 2009-05-15 2018-12-04 Redx Pharma Ltd "derivados de fármaco redox"
WO2011121596A2 (en) * 2010-04-01 2011-10-06 Neuland Laboratories Ltd. Crystal modification of moxifloxacin hydrochloride
BRPI1106900A2 (pt) 2011-12-26 2013-11-05 Ems Sa Composição farmacêutica sólida compreendendo antibótico da familia das quinolonas e processo de sua obtenção
FR2992218B1 (fr) 2012-06-22 2015-01-23 Rivopharm Sa Composition pharmaceutique de chlorhydrate de moxifloxacine et procede de preparation
CN102924449B (zh) * 2012-10-30 2015-08-12 重庆福安药业集团庆余堂制药有限公司 盐酸莫西沙星h晶型及其制备方法和药物组合物
EP2928892B1 (en) 2012-12-04 2018-03-21 Mankind Pharma Ltd. An improved process for the preparation of moxifloxacin hydrochloride
RU2561037C2 (ru) * 2013-02-07 2015-08-20 Открытое акционерное общество "Химико-фармацевтический комбинат "АКРИХИН" (ОАО "АКРИХИН") Антибактериальная фармацевтическая композиция и способ ее получения
EP2969004A4 (en) 2013-03-15 2016-09-21 Melinta Therapeutics Inc METHOD FOR THE TREATMENT OF INFECTIONS IN OVERWEIGHT AND ADIPOSIVE PATIENTS USING ANTIBIOTICS

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3601567A1 (de) * 1986-01-21 1987-07-23 Bayer Ag 7-(azabicycloalkyl)-chinoloncarbonsaeure- und -naphthyridon-carbonsaeure-derivate
EP0241206A3 (en) * 1986-03-31 1989-05-10 Sankyo Company Limited Quinoline-3-carboxylic acid derivatives, their preparation and use
AU609974B2 (en) * 1988-05-18 1991-05-09 Warner-Lambert Company Improved process for the preparation of 5-amino-7- (substituted amino)-quinoline-3-carboxylic acids
DE3910663A1 (de) * 1989-04-03 1990-10-04 Bayer Ag 5-alkylchinoloncarbonsaeuren
RO108347B1 (ro) * 1989-10-30 1994-04-28 Bellon Labor Sa Roger DERIVATI DE BENZO-(b)-NAFTIRIDIN-1,8 SI PROCEDEU DE PREPARARE A ACESTORA
TW209865B (forum.php) 1992-01-10 1993-07-21 Bayer Ag
WO1993015070A1 (en) * 1992-01-31 1993-08-05 Chugai Seiyaku Kabushiki Kaisha Crystal of quinolonecarboxylic acid derivative hydrate
DE4234078A1 (de) * 1992-10-09 1994-04-14 Bayer Ag Chinoloncarbonsäuren
JP3268098B2 (ja) * 1992-12-25 2002-03-25 第一製薬株式会社 二環性環状アミン誘導体
ZA946853B (en) * 1993-09-10 1995-04-24 Daiichi Seiyaku Co Crystals of antimicrobial compound.
ES2121293T3 (es) * 1994-04-07 1998-11-16 Pfizer Uso de trovafloxacina o derivados de la misma para la fabricacion de un medicamento para el tratamiento de infecciones por h. pylori.

Also Published As

Publication number Publication date
EE03474B1 (et) 2001-08-15
MY117492A (en) 2004-07-31
CU22774A3 (es) 2002-07-24
CN1160052A (zh) 1997-09-24
SA96170492B1 (ar) 2006-05-23
NO965298D0 (no) 1996-12-11
AR005009A1 (es) 1999-04-07
MA24342A1 (fr) 1998-07-01
BG101043A (en) 1998-04-30
MX9606325A (es) 1997-10-31
HU9603428D0 (en) 1997-01-28
SK159196A3 (en) 1997-10-08
HUP9603428A2 (en) 1997-08-28
EP0780390B1 (de) 2002-07-31
JPH09169757A (ja) 1997-06-30
PL317415A1 (en) 1997-06-23
US5849752A (en) 1998-12-15
KR970042550A (ko) 1997-07-24
ZA9610405B (en) 1997-06-23
RU2162468C2 (ru) 2001-01-27
NO306725B1 (no) 1999-12-13
RO119782B1 (ro) 2005-03-30
IL119795A0 (en) 1997-03-18
EP0780390A1 (de) 1997-06-25
NO965298L (no) 1997-06-13
HUP9603428A3 (en) 1997-10-28
HU226521B1 (en) 2009-03-30
AU7421696A (en) 1997-06-19
ATE221531T1 (de) 2002-08-15
YU65096A (sh) 1998-12-23
ES2179910T3 (es) 2003-02-01
BR9605968A (pt) 1998-08-18
NZ299905A (en) 1998-09-24
DE19546249A1 (de) 1997-06-19
JP4104687B2 (ja) 2008-06-18
DE59609501D1 (de) 2002-09-05
HRP960558B1 (en) 2002-04-30
CZ288657B6 (cs) 2001-08-15
YU49485B (sh) 2006-08-17
IN185805B (forum.php) 2001-05-05
PT780390E (pt) 2002-11-29
DK0780390T3 (da) 2002-11-11
HRP960558A2 (en) 1998-02-28
BG62258B1 (bg) 1999-06-30
AU708006B2 (en) 1999-07-29
CA2192418C (en) 2001-06-12
CZ364696A3 (en) 1997-07-16
ID22625A (id) 1999-12-02
EE9600201A (et) 1997-06-16
SK282805B6 (sk) 2002-12-03
CN1061348C (zh) 2001-01-31
SI0780390T1 (en) 2002-10-31
TW411340B (en) 2000-11-11
IL119795A (en) 1998-12-27
UA35638C2 (uk) 2001-04-16
SG47201A1 (en) 1998-03-20
NL300109I1 (nl) 2003-02-03
CA2192418A1 (en) 1997-06-13
CO4480105A1 (es) 1997-07-09
PL184885B1 (pl) 2003-01-31
KR100525146B1 (ko) 2006-01-27
TR199600970A2 (tr) 1997-06-21

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