SU1052158A3 - Способ получени производных пиримидилхиназолина или их солей (его варианты) - Google Patents

Способ получени производных пиримидилхиназолина или их солей (его варианты) Download PDF

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Publication number
SU1052158A3
SU1052158A3 SU813261941A SU3261941A SU1052158A3 SU 1052158 A3 SU1052158 A3 SU 1052158A3 SU 813261941 A SU813261941 A SU 813261941A SU 3261941 A SU3261941 A SU 3261941A SU 1052158 A3 SU1052158 A3 SU 1052158A3
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SU
USSR - Soviet Union
Prior art keywords
formula
alkyl
compound
amino
hydrogen
Prior art date
Application number
SU813261941A
Other languages
English (en)
Russian (ru)
Inventor
Бендер Хейнц
Рабе Томас
Бон Хельмут
Марторана Пьеро
Original Assignee
Касселла Аг (Фирма)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Касселла Аг (Фирма) filed Critical Касселла Аг (Фирма)
Application granted granted Critical
Publication of SU1052158A3 publication Critical patent/SU1052158A3/ru

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Hospice & Palliative Care (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Catching Or Destruction (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
SU813261941A 1980-03-27 1981-03-25 Способ получени производных пиримидилхиназолина или их солей (его варианты) SU1052158A3 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19803011809 DE3011809A1 (de) 1980-03-27 1980-03-27 Pyrimidyl-chinazoline, verfahren zu ihrer herstellung, sie enthaltende pharmazeutische praeparate und ihre verwendung

Publications (1)

Publication Number Publication Date
SU1052158A3 true SU1052158A3 (ru) 1983-10-30

Family

ID=6098481

Family Applications (1)

Application Number Title Priority Date Filing Date
SU813261941A SU1052158A3 (ru) 1980-03-27 1981-03-25 Способ получени производных пиримидилхиназолина или их солей (его варианты)

Country Status (18)

Country Link
EP (1) EP0037495A1 (enExample)
JP (1) JPS56150088A (enExample)
AR (1) AR227542A1 (enExample)
AU (1) AU6877481A (enExample)
CA (1) CA1156656A (enExample)
CS (1) CS219898B2 (enExample)
DD (1) DD157614A5 (enExample)
DE (1) DE3011809A1 (enExample)
DK (1) DK115581A (enExample)
ES (1) ES500738A0 (enExample)
FI (1) FI810778L (enExample)
GR (1) GR71870B (enExample)
IL (1) IL62495A0 (enExample)
NO (1) NO810870L (enExample)
PL (2) PL230320A1 (enExample)
PT (1) PT72724B (enExample)
SU (1) SU1052158A3 (enExample)
ZA (1) ZA812034B (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6267077A (ja) * 1985-09-18 1987-03-26 Mitsui Petrochem Ind Ltd キナゾリン誘導体及び医薬
JPS61140568A (ja) * 1984-12-14 1986-06-27 Mitsui Petrochem Ind Ltd キナゾリン誘導体及びそれを有効成分とする血圧降下剤
KR101071390B1 (ko) * 2004-03-15 2011-10-07 다케다 야쿠힌 고교 가부시키가이샤 디펩티딜 펩티다제 억제제
EP1778236B1 (en) * 2004-07-02 2010-07-14 Corcept Therapeutics, Inc. Modified pyrimidine glucocorticoid receptor modulators
MX347862B (es) 2011-03-18 2017-05-17 Corcept Therapeutics Inc Moduladores de receptores de glucocorticoides de pirimidina ciclohexilo.
CA3102099C (en) 2018-06-04 2023-09-26 Corcept Therapeutics Incorporated Pyrimidine cyclohexenyl glucocorticoid receptor modulators
MX2022006633A (es) 2019-12-11 2022-06-24 Corcept Therapeutics Inc Metodos de tratamiento del aumento de peso inducido por antipsicoticos con miricorilant.
WO2021226260A1 (en) 2020-05-06 2021-11-11 Corcept Therapeutics Incorporated Polymorphs of pyrimidine cyclohexyl glucocorticoid receptor modulators
CN115515569A (zh) 2020-05-06 2022-12-23 科赛普特治疗公司 嘧啶环己基糖皮质激素受体调节剂的制剂
CA3202353A1 (en) 2020-12-21 2022-06-30 Jeffrey Mark Dener Method of preparing pyrimidine cyclohexyl glucocorticoid receptor modulators

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2007656B (en) * 1977-11-05 1982-05-19 Pfizer Ltd Therapeutic agents

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
1. Бюлер К., Пирсон Д. Органические синтезы. М., Мир, 1973, ч. 1,с. 504. 2. Патент US №3511836, кл. 260-г25&.4, 1970. *

Also Published As

Publication number Publication date
DE3011809A1 (de) 1981-10-01
FI810778A7 (fi) 1981-09-28
AR227542A1 (es) 1982-11-15
GR71870B (enExample) 1983-07-08
NO810870L (no) 1981-09-28
DK115581A (da) 1981-09-28
PT72724A (de) 1981-04-01
PL233882A1 (enExample) 1982-05-10
ES8202000A1 (es) 1982-01-16
CA1156656A (en) 1983-11-08
IL62495A0 (en) 1981-05-20
CS219898B2 (en) 1983-03-25
AU6877481A (en) 1981-10-01
FI810778L (fi) 1981-09-28
ES500738A0 (es) 1982-01-16
PT72724B (de) 1982-03-24
ZA812034B (en) 1982-05-26
EP0037495A1 (de) 1981-10-14
JPS56150088A (en) 1981-11-20
PL230320A1 (enExample) 1982-03-29
DD157614A5 (de) 1982-11-24

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