SMP201000118B - Composto di ossimetilene arile e loro utilizzo - Google Patents

Composto di ossimetilene arile e loro utilizzo

Info

Publication number
SMP201000118B
SMP201000118B SM201000118T SM201000118T SMP201000118B SM P201000118 B SMP201000118 B SM P201000118B SM 201000118 T SM201000118 T SM 201000118T SM 201000118 T SM201000118 T SM 201000118T SM P201000118 B SMP201000118 B SM P201000118B
Authority
SM
San Marino
Prior art keywords
oxygenate
aryl compound
aryl
compound
oxygenate aryl
Prior art date
Application number
SM201000118T
Other languages
English (en)
Other versions
SMAP201000118A (it
Inventor
Maria E Wilson
Jeffrey Johnson
Edward L Clemens
Zuchun Zhao
Xin Chen
Original Assignee
Metabolex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40668739&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SMP201000118(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Metabolex Inc filed Critical Metabolex Inc
Publication of SMAP201000118A publication Critical patent/SMAP201000118A/it
Publication of SMP201000118B publication Critical patent/SMP201000118B/it

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/401—Proline; Derivatives thereof, e.g. captopril
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
SM201000118T 2008-03-31 2010-10-28 Composto di ossimetilene arile e loro utilizzo SMP201000118B (it)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US4119608P 2008-03-31 2008-03-31
PCT/US2009/038847 WO2009123992A1 (en) 2008-03-31 2009-03-30 Oxymethylene aryl compounds and uses thereof

Publications (2)

Publication Number Publication Date
SMAP201000118A SMAP201000118A (it) 2011-01-19
SMP201000118B true SMP201000118B (it) 2011-09-09

Family

ID=40668739

Family Applications (1)

Application Number Title Priority Date Filing Date
SM201000118T SMP201000118B (it) 2008-03-31 2010-10-28 Composto di ossimetilene arile e loro utilizzo

Country Status (19)

Country Link
US (1) US20090270404A1 (it)
EP (1) EP2280704B1 (it)
JP (1) JP5711655B2 (it)
KR (1) KR20100134659A (it)
CN (1) CN102026636B (it)
AR (1) AR072352A1 (it)
AU (1) AU2009231906A1 (it)
BR (1) BRPI0909469A2 (it)
CA (1) CA2719507C (it)
CL (1) CL2009000782A1 (it)
DK (1) DK2280704T3 (it)
ES (1) ES2543358T3 (it)
IL (1) IL208230A0 (it)
MX (1) MX2010010562A (it)
PL (1) PL2280704T3 (it)
SM (1) SMP201000118B (it)
TW (1) TW201002705A (it)
WO (1) WO2009123992A1 (it)
ZA (1) ZA201006687B (it)

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ZA201006687B (en) 2011-12-28
EP2280704B1 (en) 2015-05-13
BRPI0909469A2 (pt) 2015-12-29
SMAP201000118A (it) 2011-01-19
JP5711655B2 (ja) 2015-05-07
ES2543358T3 (es) 2015-08-18
CA2719507C (en) 2018-03-27
CA2719507A1 (en) 2009-10-08
EP2280704A1 (en) 2011-02-09
CN102026636A (zh) 2011-04-20
WO2009123992A1 (en) 2009-10-08
KR20100134659A (ko) 2010-12-23
TW201002705A (en) 2010-01-16
PL2280704T3 (pl) 2015-10-30
CL2009000782A1 (es) 2010-04-30
AR072352A1 (es) 2010-08-25
AU2009231906A1 (en) 2009-10-08
US20090270404A1 (en) 2009-10-29
MX2010010562A (es) 2010-12-07
HK1153946A1 (en) 2012-04-20
JP2011516428A (ja) 2011-05-26
CN102026636B (zh) 2014-07-16
DK2280704T3 (en) 2015-06-29

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