SK8132001A3 - Sulphonyloxazolamines as therapeutic active ingredients - Google Patents

Sulphonyloxazolamines as therapeutic active ingredients Download PDF

Info

Publication number
SK8132001A3
SK8132001A3 SK813-2001A SK8132001A SK8132001A3 SK 8132001 A3 SK8132001 A3 SK 8132001A3 SK 8132001 A SK8132001 A SK 8132001A SK 8132001 A3 SK8132001 A3 SK 8132001A3
Authority
SK
Slovakia
Prior art keywords
formula
oxazol
compounds
amine
benzenesulfonyl
Prior art date
Application number
SK813-2001A
Other languages
English (en)
Slovak (sk)
Inventor
Hartmut Greiner
Gerd Bartoszyk
Henning Bottcher
Gerhard Barnickel
Bertram Cezanne
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of SK8132001A3 publication Critical patent/SK8132001A3/sk

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/48Nitrogen atoms not forming part of a nitro radical
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
SK813-2001A 1998-12-18 1999-12-01 Sulphonyloxazolamines as therapeutic active ingredients SK8132001A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19858593A DE19858593A1 (de) 1998-12-18 1998-12-18 Sulfonyloxazolamine als therapeutische Wirkstoffe
PCT/EP1999/009335 WO2000037452A1 (de) 1998-12-18 1999-12-01 Sulfonyloxazolamine als therapeutische wirkstoffe

Publications (1)

Publication Number Publication Date
SK8132001A3 true SK8132001A3 (en) 2002-02-05

Family

ID=7891645

Family Applications (1)

Application Number Title Priority Date Filing Date
SK813-2001A SK8132001A3 (en) 1998-12-18 1999-12-01 Sulphonyloxazolamines as therapeutic active ingredients

Country Status (19)

Country Link
US (1) US6441013B1 (ja)
EP (1) EP1140875A1 (ja)
JP (1) JP2002533332A (ja)
CN (1) CN1146549C (ja)
AR (1) AR021896A1 (ja)
AU (1) AU763070B2 (ja)
BR (1) BR9916310A (ja)
CA (1) CA2356134A1 (ja)
CZ (1) CZ20012144A3 (ja)
DE (1) DE19858593A1 (ja)
HK (1) HK1043125A1 (ja)
HU (1) HUP0104834A3 (ja)
ID (1) ID29966A (ja)
NO (1) NO20012965D0 (ja)
PL (1) PL349393A1 (ja)
RU (1) RU2232757C2 (ja)
SK (1) SK8132001A3 (ja)
WO (1) WO2000037452A1 (ja)
ZA (1) ZA200105881B (ja)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE19956791A1 (de) * 1999-11-25 2001-05-31 Merck Patent Gmbh Neue Sulfonyloxazolamine
DE10129940A1 (de) * 2001-06-13 2002-12-19 Merck Patent Gmbh Sulfonyloxazolamine als therapeutische Wirkstoffe
US6875771B2 (en) * 2002-07-26 2005-04-05 Bristol-Myers Squibb Company Pyridopyrimidine derivatives as 5-HT6 antagonists
FR2854632B1 (fr) * 2003-05-07 2005-06-17 Centre Nat Rech Scient Synthese de composes heterocycliques substitues
PT1831159E (pt) * 2004-12-21 2010-03-03 Hoffmann La Roche Derivados de tetralina e de indano e as suas utilizações
KR20080031038A (ko) * 2005-07-29 2008-04-07 4에스체 악티엔게젤샤프트 신규의 헤테로환 NF-κB 억제제
WO2008061248A2 (en) * 2006-11-16 2008-05-22 The Regents Of The University Of California Phenylsulfoxyoxazole compound inhibitors of urea transporters
RU2473545C2 (ru) * 2007-02-02 2013-01-27 Ф.Хоффманн-Ля Рош Аг Новые 2-аминооксазолины в качестве лигандов taar1 для заболеваний цнс
MX2009008465A (es) * 2007-02-15 2009-08-20 Hoffmann La Roche Nuevas 2-aminooxazolinas como ligandos de taar1.
RU2443697C1 (ru) 2010-12-21 2012-02-27 Александр Васильевич Иващенко Замещенные метил-амины, антагонисты серотониновых 5-ht6 рецепторов, способы получения и применения
CN109789129B (zh) * 2016-07-12 2022-04-29 延世大学校产学协力团 自噬改良材料及其用途
KR102533605B1 (ko) * 2018-01-10 2023-05-17 주식회사 라이조테크 신규한 페닐설포닐 옥사졸 유도체 및 이의 용도

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG87052A1 (en) 1996-02-20 2002-03-19 Bristol Myers Squibb Co Pinacol ester intermediates useful for the preparation of biphenyl isoxazole sulfonamides

Also Published As

Publication number Publication date
PL349393A1 (en) 2002-07-15
AR021896A1 (es) 2002-08-07
HK1043125A1 (zh) 2002-09-06
CZ20012144A3 (cs) 2002-01-16
ZA200105881B (en) 2002-10-17
CN1331684A (zh) 2002-01-16
CN1146549C (zh) 2004-04-21
JP2002533332A (ja) 2002-10-08
AU1861200A (en) 2000-07-12
HUP0104834A3 (en) 2005-06-28
NO20012965L (no) 2001-06-15
US6441013B1 (en) 2002-08-27
DE19858593A1 (de) 2000-06-21
ID29966A (id) 2001-10-25
EP1140875A1 (de) 2001-10-10
RU2232757C2 (ru) 2004-07-20
AU763070B2 (en) 2003-07-10
NO20012965D0 (no) 2001-06-15
BR9916310A (pt) 2001-11-06
HUP0104834A2 (hu) 2002-07-29
WO2000037452A1 (de) 2000-06-29
CA2356134A1 (en) 2000-06-29

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