SK8132001A3 - Sulphonyloxazolamines as therapeutic active ingredients - Google Patents
Sulphonyloxazolamines as therapeutic active ingredients Download PDFInfo
- Publication number
- SK8132001A3 SK8132001A3 SK813-2001A SK8132001A SK8132001A3 SK 8132001 A3 SK8132001 A3 SK 8132001A3 SK 8132001 A SK8132001 A SK 8132001A SK 8132001 A3 SK8132001 A3 SK 8132001A3
- Authority
- SK
- Slovakia
- Prior art keywords
- formula
- oxazol
- compounds
- amine
- benzenesulfonyl
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/48—Nitrogen atoms not forming part of a nitro radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19858593A DE19858593A1 (de) | 1998-12-18 | 1998-12-18 | Sulfonyloxazolamine als therapeutische Wirkstoffe |
| PCT/EP1999/009335 WO2000037452A1 (de) | 1998-12-18 | 1999-12-01 | Sulfonyloxazolamine als therapeutische wirkstoffe |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SK8132001A3 true SK8132001A3 (en) | 2002-02-05 |
Family
ID=7891645
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SK813-2001A SK8132001A3 (en) | 1998-12-18 | 1999-12-01 | Sulphonyloxazolamines as therapeutic active ingredients |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US6441013B1 (ja) |
| EP (1) | EP1140875A1 (ja) |
| JP (1) | JP2002533332A (ja) |
| CN (1) | CN1146549C (ja) |
| AR (1) | AR021896A1 (ja) |
| AU (1) | AU763070B2 (ja) |
| BR (1) | BR9916310A (ja) |
| CA (1) | CA2356134A1 (ja) |
| CZ (1) | CZ20012144A3 (ja) |
| DE (1) | DE19858593A1 (ja) |
| HK (1) | HK1043125A1 (ja) |
| HU (1) | HUP0104834A3 (ja) |
| ID (1) | ID29966A (ja) |
| NO (1) | NO20012965D0 (ja) |
| PL (1) | PL349393A1 (ja) |
| RU (1) | RU2232757C2 (ja) |
| SK (1) | SK8132001A3 (ja) |
| WO (1) | WO2000037452A1 (ja) |
| ZA (1) | ZA200105881B (ja) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19956791A1 (de) * | 1999-11-25 | 2001-05-31 | Merck Patent Gmbh | Neue Sulfonyloxazolamine |
| DE10129940A1 (de) * | 2001-06-13 | 2002-12-19 | Merck Patent Gmbh | Sulfonyloxazolamine als therapeutische Wirkstoffe |
| US6875771B2 (en) * | 2002-07-26 | 2005-04-05 | Bristol-Myers Squibb Company | Pyridopyrimidine derivatives as 5-HT6 antagonists |
| FR2854632B1 (fr) * | 2003-05-07 | 2005-06-17 | Centre Nat Rech Scient | Synthese de composes heterocycliques substitues |
| PT1831159E (pt) * | 2004-12-21 | 2010-03-03 | Hoffmann La Roche | Derivados de tetralina e de indano e as suas utilizações |
| KR20080031038A (ko) * | 2005-07-29 | 2008-04-07 | 4에스체 악티엔게젤샤프트 | 신규의 헤테로환 ＮＦ-κＢ 억제제 |
| WO2008061248A2 (en) * | 2006-11-16 | 2008-05-22 | The Regents Of The University Of California | Phenylsulfoxyoxazole compound inhibitors of urea transporters |
| RU2473545C2 (ru) * | 2007-02-02 | 2013-01-27 | Ф.Хоффманн-Ля Рош Аг | Новые 2-аминооксазолины в качестве лигандов taar1 для заболеваний цнс |
| MX2009008465A (es) * | 2007-02-15 | 2009-08-20 | Hoffmann La Roche | Nuevas 2-aminooxazolinas como ligandos de taar1. |
| RU2443697C1 (ru) | 2010-12-21 | 2012-02-27 | Александр Васильевич Иващенко | Замещенные метил-амины, антагонисты серотониновых 5-ht6 рецепторов, способы получения и применения |
| CN109789129B (zh) * | 2016-07-12 | 2022-04-29 | 延世大学校产学协力团 | 自噬改良材料及其用途 |
| KR102533605B1 (ko) * | 2018-01-10 | 2023-05-17 | 주식회사 라이조테크 | 신규한 페닐설포닐 옥사졸 유도체 및 이의 용도 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG87052A1 (en) | 1996-02-20 | 2002-03-19 | Bristol Myers Squibb Co | Pinacol ester intermediates useful for the preparation of biphenyl isoxazole sulfonamides |
-
1998
- 1998-12-18 DE DE19858593A patent/DE19858593A1/de not_active Withdrawn
-
1999
- 1999-12-01 EP EP99962190A patent/EP1140875A1/de not_active Withdrawn
- 1999-12-01 WO PCT/EP1999/009335 patent/WO2000037452A1/de not_active Application Discontinuation
- 1999-12-01 US US09/868,097 patent/US6441013B1/en not_active Expired - Fee Related
- 1999-12-01 ID IDW00200101555A patent/ID29966A/id unknown
- 1999-12-01 CN CNB998147281A patent/CN1146549C/zh not_active Expired - Fee Related
- 1999-12-01 CA CA002356134A patent/CA2356134A1/en not_active Abandoned
- 1999-12-01 RU RU2001119273/04A patent/RU2232757C2/ru not_active IP Right Cessation
- 1999-12-01 SK SK813-2001A patent/SK8132001A3/sk unknown
- 1999-12-01 JP JP2000589524A patent/JP2002533332A/ja active Pending
- 1999-12-01 BR BR9916310-1A patent/BR9916310A/pt not_active IP Right Cessation
- 1999-12-01 AU AU18612/00A patent/AU763070B2/en not_active Ceased
- 1999-12-01 PL PL99349393A patent/PL349393A1/xx unknown
- 1999-12-01 HU HU0104834A patent/HUP0104834A3/hu unknown
- 1999-12-01 CZ CZ20012144A patent/CZ20012144A3/cs unknown
- 1999-12-17 AR ARP990106528A patent/AR021896A1/es not_active Application Discontinuation
-
2001
- 2001-06-15 NO NO20012965A patent/NO20012965D0/no not_active Application Discontinuation
- 2001-07-17 ZA ZA200105881A patent/ZA200105881B/en unknown
-
2002
- 2002-07-02 HK HK02104944.7A patent/HK1043125A1/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| PL349393A1 (en) | 2002-07-15 |
| AR021896A1 (es) | 2002-08-07 |
| HK1043125A1 (zh) | 2002-09-06 |
| CZ20012144A3 (cs) | 2002-01-16 |
| ZA200105881B (en) | 2002-10-17 |
| CN1331684A (zh) | 2002-01-16 |
| CN1146549C (zh) | 2004-04-21 |
| JP2002533332A (ja) | 2002-10-08 |
| AU1861200A (en) | 2000-07-12 |
| HUP0104834A3 (en) | 2005-06-28 |
| NO20012965L (no) | 2001-06-15 |
| US6441013B1 (en) | 2002-08-27 |
| DE19858593A1 (de) | 2000-06-21 |
| ID29966A (id) | 2001-10-25 |
| EP1140875A1 (de) | 2001-10-10 |
| RU2232757C2 (ru) | 2004-07-20 |
| AU763070B2 (en) | 2003-07-10 |
| NO20012965D0 (no) | 2001-06-15 |
| BR9916310A (pt) | 2001-11-06 |
| HUP0104834A2 (hu) | 2002-07-29 |
| WO2000037452A1 (de) | 2000-06-29 |
| CA2356134A1 (en) | 2000-06-29 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| Turner et al. | Antihypertensive thiadiazoles. 2. Vasodilator activity of some 2-aryl-5-guanidino-1, 3, 4-thiadiazoles | |
| SK8132001A3 (en) | Sulphonyloxazolamines as therapeutic active ingredients | |
| HU213113B (en) | Process for producing 2-aminobenzoxazole and 2-amino-benzothiazole derivatives and pharmaceutical compositions containing them | |
| SK122099A3 (en) | Substituted 4-arylmethylene-2-imino-2,3-dihydrothiazoles and derivatives and their pharmaceutical use | |
| SK281457B6 (sk) | 3-[4-(4-(4-kyánfenyl)-1-piperazinyl)butyl]-5-kyánindol, spôsob jeho prípravy, jeho použitie a farmaceutický prostriedok, ktorý ho obsahuje | |
| KR100417506B1 (ko) | 항우울 치료를 위한 5ｈｔ1 길항제 | |
| CZ20011551A3 (cs) | Derivát benzoylpyridazinu, způsob jeho přípravy a farmaceutický prostředek, který ho obsahuje | |
| FI89915B (fi) | Foerfarande foer framstaellning av psykotropiska acykliska amidderivat | |
| SK112799A3 (en) | Oxazolidinones, preparation method and use thereof, pharmaceutical compositions | |
| US20230406853A1 (en) | Covalent cdk2-binding compounds for therapeutic purposes | |
| US6737426B1 (en) | Sulfonyloxazoleamines | |
| WO2002100842A1 (en) | Sulfonyloxazolamines and their use as 5-ht6 ligands | |
| KR20010086457A (ko) | 치료 활성 화합물로서의 술포닐옥사졸아민류 | |
| CZ20033194A3 (cs) | Deriváty 6H-oxazolo[4,5-e]indolu jako ligandy nikotinacetyl-cholinového receptoru a/nebo serotonergické ligandy, způsob jejich přípravy a jejich použití | |
| CZ291446B6 (cs) | Derivát piperidinylmethyloxazolidinonu a farmaceutický prostředek, který ho obsahuje | |
| SK2192002A3 (en) | Piperidine alcohol derivative, process for the preparation and use thereof and pharmaceutical composition comprising same | |
| EP0405905B1 (en) | Use of Isoxazolin-3-one Derivatives as antidepressants | |
| US4105795A (en) | Antispasmodic substituted sulphoximides | |
| MXPA01006230A (en) | Sulphonyloxazolamines as therapeutic active ingredients | |
| GB2031427A (en) | N-substituted cyclic amines their preparation and pharmaceutical compositions containing them | |
| BG60318B2 (bg) | Метод за получаване на триазолил тиоамидни производни | |
| CZ9903260A3 (cs) | Terapeutická činidla |