SK391091A3 - Crystalline paroxetine hydrochloride hemihydrate, pharmacuetical composition containing the same and its use - Google Patents

Crystalline paroxetine hydrochloride hemihydrate, pharmacuetical composition containing the same and its use Download PDF

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Publication number
SK391091A3
SK391091A3 SK3910-91A SK391091A SK391091A3 SK 391091 A3 SK391091 A3 SK 391091A3 SK 391091 A SK391091 A SK 391091A SK 391091 A3 SK391091 A3 SK 391091A3
Authority
SK
Slovakia
Prior art keywords
solution
paroxetine
paroxetine hydrochloride
hemihydrate
hydrochloride
Prior art date
Application number
SK3910-91A
Other languages
English (en)
Slovak (sk)
Inventor
Roger D Barnes
Marian W Wood-Kaczmar
Alan David Curzons
Ian R Lynch
John E Richardson
Philip C Buxton
Original Assignee
Beecham Group Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26289934&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SK391091(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB858526408A external-priority patent/GB8526408D0/en
Priority claimed from GB858526407A external-priority patent/GB8526407D0/en
Application filed by Beecham Group Plc filed Critical Beecham Group Plc
Publication of SK391091A3 publication Critical patent/SK391091A3/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Psychiatry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
SK3910-91A 1985-10-25 1991-12-19 Crystalline paroxetine hydrochloride hemihydrate, pharmacuetical composition containing the same and its use SK391091A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB858526408A GB8526408D0 (en) 1985-10-25 1985-10-25 Chemical process
GB858526407A GB8526407D0 (en) 1985-10-25 1985-10-25 Compounds

Publications (1)

Publication Number Publication Date
SK391091A3 true SK391091A3 (en) 2000-10-09

Family

ID=26289934

Family Applications (1)

Application Number Title Priority Date Filing Date
SK3910-91A SK391091A3 (en) 1985-10-25 1991-12-19 Crystalline paroxetine hydrochloride hemihydrate, pharmacuetical composition containing the same and its use

Country Status (18)

Country Link
US (1) US4721723A (no)
EP (1) EP0223403B1 (no)
JP (1) JPH0647587B2 (no)
AU (1) AU593295B2 (no)
BG (1) BG61323B2 (no)
CA (1) CA1287060C (no)
CY (1) CY1743A (no)
CZ (1) CZ391091A3 (no)
DE (1) DE3688827T2 (no)
DK (1) DK171694B1 (no)
ES (1) ES2058061T3 (no)
FI (1) FI87785C (no)
HK (1) HK125993A (no)
IE (1) IE59901B1 (no)
NO (1) NO171453C (no)
NZ (1) NZ218047A (no)
PT (1) PT83608B (no)
SK (1) SK391091A3 (no)

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* Cited by examiner, † Cited by third party
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DE3688827D1 (de) 1993-09-09
FI864320A (fi) 1987-04-26
NO864237D0 (no) 1986-10-23
BG61323B2 (bg) 1997-05-30
EP0223403A2 (en) 1987-05-27
JPS62129280A (ja) 1987-06-11
CY1743A (en) 1995-02-17
IE862802L (en) 1987-04-25
CA1287060C (en) 1991-07-30
EP0223403A3 (en) 1989-09-06
US4721723A (en) 1988-01-26
HK125993A (en) 1993-11-19
ES2058061T3 (es) 1994-11-01
NO171453C (no) 1993-03-17
DK508786D0 (da) 1986-10-23
IE59901B1 (en) 1994-04-20
JPH0647587B2 (ja) 1994-06-22
AU593295B2 (en) 1990-02-08
DE3688827T2 (de) 1994-03-31
PT83608B (pt) 1989-05-31
PT83608A (en) 1986-11-01
NO864237L (no) 1987-04-27
FI87785C (fi) 1993-02-25
AU6433286A (en) 1987-04-30
NO171453B (no) 1992-12-07
EP0223403B1 (en) 1993-08-04
FI87785B (fi) 1992-11-13
CZ391091A3 (en) 1994-01-19
DK508786A (da) 1987-04-26
NZ218047A (en) 1989-03-29
FI864320A0 (fi) 1986-10-24
DK171694B1 (da) 1997-03-17

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