SK286981B6 - Prášok na použitie v inhalátore na suché prášky, nosič na tento prášok a spôsob výroby prášku - Google Patents
Prášok na použitie v inhalátore na suché prášky, nosič na tento prášok a spôsob výroby prášku Download PDFInfo
- Publication number
- SK286981B6 SK286981B6 SK1248-2001A SK12482001A SK286981B6 SK 286981 B6 SK286981 B6 SK 286981B6 SK 12482001 A SK12482001 A SK 12482001A SK 286981 B6 SK286981 B6 SK 286981B6
- Authority
- SK
- Slovakia
- Prior art keywords
- carrier
- powder
- magnesium stearate
- particles
- carrier particles
- Prior art date
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- HQKMJHAJHXVSDF-UHFFFAOYSA-L magnesium stearate Chemical compound [Mg+2].CCCCCCCCCCCCCCCCCC([O-])=O.CCCCCCCCCCCCCCCCCC([O-])=O HQKMJHAJHXVSDF-UHFFFAOYSA-L 0.000 claims abstract description 119
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- NDAUXUAQIAJITI-UHFFFAOYSA-N albuterol Chemical compound CC(C)(C)NCC(O)C1=CC=C(O)C(CO)=C1 NDAUXUAQIAJITI-UHFFFAOYSA-N 0.000 claims description 8
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- MIXMJCQRHVAJIO-TZHJZOAOSA-N qk4dys664x Chemical compound O.C1([C@@H](F)C2)=CC(=O)C=C[C@]1(C)[C@@H]1[C@@H]2[C@@H]2C[C@H]3OC(C)(C)O[C@@]3(C(=O)CO)[C@@]2(C)C[C@@H]1O.C1([C@@H](F)C2)=CC(=O)C=C[C@]1(C)[C@@H]1[C@@H]2[C@@H]2C[C@H]3OC(C)(C)O[C@@]3(C(=O)CO)[C@@]2(C)C[C@@H]1O MIXMJCQRHVAJIO-TZHJZOAOSA-N 0.000 claims description 2
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- QIQXTHQIDYTFRH-UHFFFAOYSA-N octadecanoic acid Chemical compound CCCCCCCCCCCCCCCCCC(O)=O QIQXTHQIDYTFRH-UHFFFAOYSA-N 0.000 description 3
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- 229910002016 Aerosil® 200 Inorganic materials 0.000 description 1
- GUBGYTABKSRVRQ-XLOQQCSPSA-N Alpha-Lactose Chemical compound O[C@@H]1[C@@H](O)[C@@H](O)[C@@H](CO)O[C@H]1O[C@@H]1[C@@H](CO)O[C@H](O)[C@H](O)[C@H]1O GUBGYTABKSRVRQ-XLOQQCSPSA-N 0.000 description 1
- 101100386627 Arabidopsis thaliana SAMDC4 gene Proteins 0.000 description 1
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- DBMJMQXJHONAFJ-UHFFFAOYSA-M Sodium laurylsulphate Chemical compound [Na+].CCCCCCCCCCCCOS([O-])(=O)=O DBMJMQXJHONAFJ-UHFFFAOYSA-M 0.000 description 1
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Classifications
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- A61P37/08—Antiallergic agents
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/27—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation
- C07C45/29—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups
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- C—CHEMISTRY; METALLURGY
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/27—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation
- C07C45/29—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups
- C07C45/298—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups with manganese derivatives
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
- C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
- C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
- C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
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- C—CHEMISTRY; METALLURGY
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- C07C47/00—Compounds having —CHO groups
- C07C47/38—Unsaturated compounds having —CHO groups bound to carbon atoms of rings other than six—membered aromatic rings
- C07C47/47—Unsaturated compounds having —CHO groups bound to carbon atoms of rings other than six—membered aromatic rings containing ether groups, groups, groups, or groups
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/58—Unsaturated compounds containing ether groups, groups, groups, or groups
- C07C59/64—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings
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- C—CHEMISTRY; METALLURGY
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
- C07C59/40—Unsaturated compounds
- C07C59/58—Unsaturated compounds containing ether groups, groups, groups, or groups
- C07C59/72—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings and other rings
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/66—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety
- C07C69/73—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of unsaturated acids
- C07C69/734—Ethers
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Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/EP1999/001449 WO2000053157A1 (fr) | 1999-03-05 | 1999-03-05 | Compositions pharmaceutiques en poudre ameliorees pour inhalation |
Publications (2)
Publication Number | Publication Date |
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SK12482001A3 SK12482001A3 (sk) | 2002-01-07 |
SK286981B6 true SK286981B6 (sk) | 2009-08-06 |
Family
ID=8167234
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SK1248-2001A SK286981B6 (sk) | 1999-03-05 | 1999-03-05 | Prášok na použitie v inhalátore na suché prášky, nosič na tento prášok a spôsob výroby prášku |
Country Status (17)
Country | Link |
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US (3) | US6528096B1 (fr) |
EP (1) | EP1158958B1 (fr) |
AT (1) | ATE363892T1 (fr) |
AU (1) | AU3409399A (fr) |
BR (1) | BR9917246A (fr) |
CY (1) | CY1106817T1 (fr) |
CZ (1) | CZ298489B6 (fr) |
DE (1) | DE69936268T2 (fr) |
DK (1) | DK1158958T3 (fr) |
ES (1) | ES2286881T3 (fr) |
HU (1) | HUP0200185A3 (fr) |
PL (1) | PL196951B1 (fr) |
PT (1) | PT1158958E (fr) |
SI (1) | SI1158958T1 (fr) |
SK (1) | SK286981B6 (fr) |
TR (1) | TR200102567T2 (fr) |
WO (1) | WO2000053157A1 (fr) |
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CN105412049B (zh) * | 2014-09-16 | 2020-01-07 | 四川海思科制药有限公司 | 一种干粉吸入剂用药物组合物及其制备方法 |
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1999
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- 1999-03-05 PT PT99915547T patent/PT1158958E/pt unknown
- 1999-03-05 CZ CZ20013185A patent/CZ298489B6/cs not_active IP Right Cessation
- 1999-03-05 ES ES99915547T patent/ES2286881T3/es not_active Expired - Lifetime
- 1999-03-05 AU AU34093/99A patent/AU3409399A/en not_active Abandoned
- 1999-03-05 SK SK1248-2001A patent/SK286981B6/sk not_active IP Right Cessation
- 1999-03-05 EP EP99915547A patent/EP1158958B1/fr not_active Revoked
- 1999-03-05 HU HU0200185A patent/HUP0200185A3/hu unknown
- 1999-03-05 AT AT99915547T patent/ATE363892T1/de active
- 1999-03-05 PL PL354841A patent/PL196951B1/pl unknown
- 1999-03-05 WO PCT/EP1999/001449 patent/WO2000053157A1/fr active IP Right Grant
- 1999-03-05 TR TR2001/02567T patent/TR200102567T2/xx unknown
- 1999-03-05 BR BR9917246-1A patent/BR9917246A/pt active Search and Examination
- 1999-03-05 DK DK99915547T patent/DK1158958T3/da active
- 1999-03-05 DE DE69936268T patent/DE69936268T2/de not_active Expired - Lifetime
-
2000
- 2000-06-26 US US09/603,620 patent/US6528096B1/en not_active Expired - Lifetime
-
2003
- 2003-02-05 US US10/358,174 patent/US20030133880A1/en not_active Abandoned
-
2006
- 2006-07-25 US US11/492,105 patent/US20060257330A1/en not_active Abandoned
-
2007
- 2007-08-13 CY CY20071101082T patent/CY1106817T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
SI1158958T1 (sl) | 2007-10-31 |
WO2000053157A1 (fr) | 2000-09-14 |
EP1158958A1 (fr) | 2001-12-05 |
EP1158958B1 (fr) | 2007-06-06 |
ES2286881T3 (es) | 2007-12-01 |
ATE363892T1 (de) | 2007-06-15 |
CZ20013185A3 (cs) | 2002-01-16 |
TR200102567T2 (tr) | 2002-01-21 |
US6528096B1 (en) | 2003-03-04 |
DE69936268D1 (de) | 2007-07-19 |
PL354841A1 (en) | 2004-02-23 |
CY1106817T1 (el) | 2012-05-23 |
AU3409399A (en) | 2000-09-28 |
HUP0200185A2 (en) | 2002-06-29 |
DE69936268T2 (de) | 2008-02-14 |
CZ298489B6 (cs) | 2007-10-17 |
US20060257330A1 (en) | 2006-11-16 |
PT1158958E (pt) | 2007-08-13 |
US20030133880A1 (en) | 2003-07-17 |
HUP0200185A3 (en) | 2006-07-28 |
PL196951B1 (pl) | 2008-02-29 |
SK12482001A3 (sk) | 2002-01-07 |
DK1158958T3 (da) | 2007-10-08 |
BR9917246A (pt) | 2002-03-26 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Patent lapsed due to non-payment of maintenance fees |
Effective date: 20170305 |