SK283904B6 - Heterocyklické zlúčeniny na inhibíciu sekrécie žalúdočnej kyseliny, spôsoby ich prípravy a farmaceutické kompozície, ktoré ich obsahujú - Google Patents

Heterocyklické zlúčeniny na inhibíciu sekrécie žalúdočnej kyseliny, spôsoby ich prípravy a farmaceutické kompozície, ktoré ich obsahujú Download PDF

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Publication number
SK283904B6
SK283904B6 SK674-2000A SK6742000A SK283904B6 SK 283904 B6 SK283904 B6 SK 283904B6 SK 6742000 A SK6742000 A SK 6742000A SK 283904 B6 SK283904 B6 SK 283904B6
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SK
Slovakia
Prior art keywords
compound
pharmaceutically acceptable
acceptable salt
compound according
alkyl
Prior art date
Application number
SK674-2000A
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English (en)
Slovak (sk)
Other versions
SK6742000A3 (en
Inventor
Kosrat Amin
Mikael Dahlstrm
Peter Nordberg
Ingemar Starke
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of SK6742000A3 publication Critical patent/SK6742000A3/sk
Publication of SK283904B6 publication Critical patent/SK283904B6/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
SK674-2000A 1997-11-28 1998-11-18 Heterocyklické zlúčeniny na inhibíciu sekrécie žalúdočnej kyseliny, spôsoby ich prípravy a farmaceutické kompozície, ktoré ich obsahujú SK283904B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9704404A SE9704404D0 (sv) 1997-11-28 1997-11-28 New compounds
PCT/SE1998/002091 WO1999028322A1 (en) 1997-11-28 1998-11-18 Heterocyclic compounds for inhibition of gastric acid secretion, processes for their preparation and pharmaceutical compositions thereof

Publications (2)

Publication Number Publication Date
SK6742000A3 SK6742000A3 (en) 2001-03-12
SK283904B6 true SK283904B6 (sk) 2004-04-06

Family

ID=20409181

Family Applications (1)

Application Number Title Priority Date Filing Date
SK674-2000A SK283904B6 (sk) 1997-11-28 1998-11-18 Heterocyklické zlúčeniny na inhibíciu sekrécie žalúdočnej kyseliny, spôsoby ich prípravy a farmaceutické kompozície, ktoré ich obsahujú

Country Status (33)

Country Link
US (1) US6518270B1 (sv)
EP (1) EP1042324B1 (sv)
JP (1) JP2001525322A (sv)
KR (1) KR20010032559A (sv)
CN (1) CN1142933C (sv)
AR (1) AR016972A1 (sv)
AT (1) ATE233263T1 (sv)
AU (1) AU752187C (sv)
BR (1) BR9814755A (sv)
CA (1) CA2311798A1 (sv)
CZ (1) CZ292349B6 (sv)
DE (1) DE69811735T2 (sv)
DK (1) DK1042324T3 (sv)
EE (1) EE04060B1 (sv)
ES (1) ES2191356T3 (sv)
HK (1) HK1030216A1 (sv)
HU (1) HUP0100601A3 (sv)
ID (1) ID24730A (sv)
IL (1) IL136145A0 (sv)
IS (1) IS5486A (sv)
MY (1) MY121032A (sv)
NO (1) NO315704B1 (sv)
NZ (1) NZ504355A (sv)
PL (1) PL340920A1 (sv)
PT (1) PT1042324E (sv)
RU (1) RU2241000C2 (sv)
SE (1) SE9704404D0 (sv)
SK (1) SK283904B6 (sv)
TR (1) TR200001530T2 (sv)
TW (1) TW515798B (sv)
UA (1) UA70932C2 (sv)
WO (1) WO1999028322A1 (sv)
ZA (1) ZA9810468B (sv)

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DE602004016831D1 (de) * 2003-03-17 2008-11-13 Affinium Pharm Inc Pharmazeutische zusammensetzungen inhibitoren von fab i und weitere antibiotika enthaltend
WO2005014599A1 (en) 2003-06-04 2005-02-17 Cellular Genomics, Inc. Imidazo[1,2-a]pyrazin-8-ylamines and method of inhibition of bruton’s tyrosine kinase by such compounds
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AU2004285394B2 (en) 2003-11-03 2009-01-08 Astrazeneca Ab Imidazo (1,2-A) pyridine derivatives for the treatment of silent gastro-esophageal reflux
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US20070293532A1 (en) * 2004-07-28 2007-12-20 Takeda Pharmaceutical Compan6Y Limited Pyrrolo [2,3-C] Pyridine Compound, Process for Producing the Same, and Use
JP2008508347A (ja) * 2004-08-02 2008-03-21 ニコメッド ゲゼルシャフト ミット ベシュレンクテル ハフツング ５置換された１Ｈ−ピロロ［３，２−ｂ］ピリジン
MX2007002219A (es) * 2004-09-03 2007-05-04 Yuhan Corp Derivados de pirrolo [3,2-b ] piridina y procesos para su preparacion.
DK1784402T3 (da) * 2004-09-03 2011-11-14 Yuhan Corp Pyrrolo[3,2-c]pyridinderivater samt fremgangsmåder til deres fremstilling
CN101018789B (zh) 2004-09-03 2010-09-08 株式会社柳韩洋行 吡咯并[2,3-c]吡啶衍生物及其制备方法
JP4989477B2 (ja) * 2004-09-03 2012-08-01 ユーハン・コーポレイション ピロロ［３，２−ｃ］ピリジン誘導体及びその製造方法
US7777040B2 (en) 2005-05-03 2010-08-17 Cgi Pharmaceuticals, Inc. Certain substituted ureas, as modulators of kinase activity
CA2620223A1 (en) 2005-09-02 2007-03-08 Abbott Laboratories Novel imidazo based heterocycles
US20090156578A1 (en) * 2005-12-05 2009-06-18 PAULS Henry 3-Heterocyclylacrylamide Compounds as Fab I Inhibitors and Antibacterial Agents
US7557104B2 (en) 2006-06-06 2009-07-07 Schering Corporation Imidazopyrazines as protein kinase inhibitors
EP2687533B1 (en) 2006-07-20 2017-07-19 Debiopharm International SA Acrylamide derivatives as FAB I inhibitors
EP2125802A4 (en) 2007-02-16 2014-08-20 Debiopharm Int Sa SALTS, PRODRUGS AND POLYMORPHES OF FAB I INHIBITORS
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CA2745871C (en) 2008-12-08 2018-02-20 Gilead Connecticut, Inc. Imidazopyrazine syk inhibitors
US9562056B2 (en) 2010-03-11 2017-02-07 Gilead Connecticut, Inc. Imidazopyridines Syk inhibitors
PL2861608T3 (pl) 2012-06-19 2019-09-30 Debiopharm International Sa Pochodne prolekowe (e)-n-metylo-n-((3-metylobenzofuran-2-ylo)metylo)-3-(7-okso-5,6,7,8-tetrahydro-1,8-naftyrydyn-3-ylo)akryloamidu
MD4684B1 (ro) 2013-07-30 2020-03-31 Gilead Connecticut INc. Formulări pe bază de imidazopirazine în calitate de inhibitori SYK
US9657023B2 (en) 2013-07-30 2017-05-23 Gilead Connecticut, Inc. Polymorph of Syk inhibitors
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Also Published As

Publication number Publication date
IS5486A (is) 2000-05-10
KR20010032559A (ko) 2001-04-25
WO1999028322A1 (en) 1999-06-10
BR9814755A (pt) 2000-10-03
RU2241000C2 (ru) 2004-11-27
DE69811735T2 (de) 2003-12-18
UA70932C2 (uk) 2004-11-15
ATE233263T1 (de) 2003-03-15
CN1142933C (zh) 2004-03-24
DE69811735D1 (de) 2003-04-03
AU752187C (en) 2003-09-18
EP1042324B1 (en) 2003-02-26
EE200000315A (et) 2001-10-15
CZ20001947A3 (cs) 2000-11-15
EE04060B1 (et) 2003-06-16
TW515798B (en) 2003-01-01
SE9704404D0 (sv) 1997-11-28
PL340920A1 (en) 2001-03-12
AU1356599A (en) 1999-06-16
CN1284078A (zh) 2001-02-14
IL136145A0 (en) 2001-05-20
DK1042324T3 (da) 2003-05-05
EP1042324A1 (en) 2000-10-11
ES2191356T3 (es) 2003-09-01
SK6742000A3 (en) 2001-03-12
ID24730A (id) 2000-08-03
CZ292349B6 (cs) 2003-09-17
HK1030216A1 (en) 2001-04-27
AU752187B2 (en) 2002-09-12
PT1042324E (pt) 2003-06-30
NO20002721L (no) 2000-07-28
TR200001530T2 (tr) 2000-11-21
ZA9810468B (en) 1999-05-21
NO315704B1 (no) 2003-10-13
NO20002721D0 (no) 2000-05-26
JP2001525322A (ja) 2001-12-11
MY121032A (en) 2005-12-30
HUP0100601A2 (hu) 2001-09-28
HUP0100601A3 (en) 2002-10-28
AR016972A1 (es) 2001-08-01
NZ504355A (en) 2001-12-21
US6518270B1 (en) 2003-02-11
CA2311798A1 (en) 1999-06-10

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