SK282902B6 - Azolové zlúčeniny s antimykotickou aktivitou na použitie v humánnej medicíne, vo veterinárnej medicíne a farmaceutický prostriedok s ich obsahom - Google Patents

Azolové zlúčeniny s antimykotickou aktivitou na použitie v humánnej medicíne, vo veterinárnej medicíne a farmaceutický prostriedok s ich obsahom Download PDF

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Publication number
SK282902B6
SK282902B6 SK1351-97A SK135197A SK282902B6 SK 282902 B6 SK282902 B6 SK 282902B6 SK 135197 A SK135197 A SK 135197A SK 282902 B6 SK282902 B6 SK 282902B6
Authority
SK
Slovakia
Prior art keywords
methyl
triazolyl
hydroxy
hydrogen
compounds
Prior art date
Application number
SK1351-97A
Other languages
English (en)
Slovak (sk)
Other versions
SK135197A3 (en
Inventor
Enrico Albini
Giovanna Schioppacassi
Original Assignee
Zambon Group S. P. A.
Isagro S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Group S. P. A., Isagro S.P.A. filed Critical Zambon Group S. P. A.
Publication of SK135197A3 publication Critical patent/SK135197A3/sk
Publication of SK282902B6 publication Critical patent/SK282902B6/sk

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C07D233/60Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by oxygen or sulfur atoms, attached to ring nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Treatments For Attaching Organic Compounds To Fibrous Goods (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SK1351-97A 1995-04-07 1996-04-02 Azolové zlúčeniny s antimykotickou aktivitou na použitie v humánnej medicíne, vo veterinárnej medicíne a farmaceutický prostriedok s ich obsahom SK282902B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ITMI950707A IT1273509B (it) 1995-04-07 1995-04-07 Composti azolici ad attivita' antimicotica per uso umano e veterinario
PCT/EP1996/001443 WO1996031490A1 (en) 1995-04-07 1996-04-02 Azole compounds with antimycotic activity for human and veterinary use

Publications (2)

Publication Number Publication Date
SK135197A3 SK135197A3 (en) 1998-02-04
SK282902B6 true SK282902B6 (sk) 2003-01-09

Family

ID=11371242

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1351-97A SK282902B6 (sk) 1995-04-07 1996-04-02 Azolové zlúčeniny s antimykotickou aktivitou na použitie v humánnej medicíne, vo veterinárnej medicíne a farmaceutický prostriedok s ich obsahom

Country Status (23)

Country Link
EP (1) EP0819124B1 (de)
JP (1) JPH11503141A (de)
KR (1) KR100418128B1 (de)
AP (1) AP875A (de)
AT (1) ATE207909T1 (de)
AU (1) AU704289B2 (de)
CA (1) CA2217695A1 (de)
CZ (1) CZ289586B6 (de)
DE (1) DE69616531T2 (de)
DK (1) DK0819124T3 (de)
EA (1) EA002142B1 (de)
ES (1) ES2164882T3 (de)
HU (1) HUP9801596A3 (de)
IT (1) IT1273509B (de)
MX (1) MX9707672A (de)
NO (1) NO974609L (de)
NZ (1) NZ306439A (de)
OA (1) OA10522A (de)
PL (1) PL186247B1 (de)
PT (1) PT819124E (de)
SK (1) SK282902B6 (de)
UA (1) UA49830C2 (de)
WO (1) WO1996031490A1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1283038B1 (it) * 1996-02-28 1998-04-07 Zambon Spa Composti azolici ad attivita' antimicotica per uso umano e veterinario
IT1296925B1 (it) 1997-12-05 1999-08-03 Zambon Spa Procedimento per la preparazione di composti ad attivita' antimicotica

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5998073A (ja) * 1982-11-02 1984-06-06 フアイザ−・コ−ポレ−シヨン トリアゾ−ル系抗真菌剤
IT1204773B (it) * 1986-01-23 1989-03-10 Montedison Spa Azolilderivati fungicidi
IT1198240B (it) * 1986-12-23 1988-12-21 Agrimont Spa Azolilderivati fungicidi
DE3644615A1 (de) * 1986-12-29 1988-07-07 Lentia Gmbh Imidazol- und triazolderivate zur verwendung als antimykotische mittel
IT1232943B (it) * 1987-11-09 1992-03-10 Mini Ricerca Scient Tecnolog Azolilderivati fungicidi.
JPH0770087A (ja) * 1993-08-26 1995-03-14 Taisho Pharmaceut Co Ltd 新規なトリアゾール誘導体およびその塩

Also Published As

Publication number Publication date
CZ289586B6 (cs) 2002-02-13
CA2217695A1 (en) 1996-10-10
OA10522A (en) 2002-04-29
AP9701100A0 (en) 1997-10-31
NZ306439A (en) 1999-02-25
AU704289B2 (en) 1999-04-15
NO974609D0 (no) 1997-10-06
DK0819124T3 (da) 2002-02-18
NO974609L (no) 1997-12-04
HUP9801596A1 (hu) 1998-11-30
EA199700299A1 (ru) 1998-04-30
WO1996031490A1 (en) 1996-10-10
PL186247B1 (pl) 2003-12-31
DE69616531D1 (de) 2001-12-06
AP875A (en) 2000-09-27
ES2164882T3 (es) 2002-03-01
AU5499496A (en) 1996-10-23
KR19980703669A (ko) 1998-12-05
EA002142B1 (ru) 2001-12-24
EP0819124A1 (de) 1998-01-21
ATE207909T1 (de) 2001-11-15
PT819124E (pt) 2002-04-29
UA49830C2 (uk) 2002-10-15
MX9707672A (es) 1997-11-29
HUP9801596A3 (en) 2000-07-28
SK135197A3 (en) 1998-02-04
PL322612A1 (en) 1998-02-02
JPH11503141A (ja) 1999-03-23
KR100418128B1 (ko) 2004-04-28
DE69616531T2 (de) 2002-07-11
ITMI950707A1 (it) 1996-10-07
ITMI950707A0 (it) 1995-04-07
EP0819124B1 (de) 2001-10-31
IT1273509B (it) 1997-07-08
CZ316997A3 (cs) 1998-03-18

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