SK13282002A3 - Sulfónamidové substituované difenylmočovinové zlúčeniny, farmaceutický prostriedok s ich obsahom a ich použitie - Google Patents
Sulfónamidové substituované difenylmočovinové zlúčeniny, farmaceutický prostriedok s ich obsahom a ich použitie Download PDFInfo
- Publication number
- SK13282002A3 SK13282002A3 SK1328-2002A SK13282002A SK13282002A3 SK 13282002 A3 SK13282002 A3 SK 13282002A3 SK 13282002 A SK13282002 A SK 13282002A SK 13282002 A3 SK13282002 A3 SK 13282002A3
- Authority
- SK
- Slovakia
- Prior art keywords
- alkyl
- chloro
- aryl
- hydroxy
- heteroaryl
- Prior art date
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Classifications
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- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/04—Systems containing only non-condensed rings with a four-membered ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
- C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2603/00—Systems containing at least three condensed rings
- C07C2603/56—Ring systems containing bridged rings
- C07C2603/58—Ring systems containing bridged rings containing three rings
- C07C2603/70—Ring systems containing bridged rings containing three rings containing only six-membered rings
- C07C2603/74—Adamantanes
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Virology (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pulmonology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Neurology (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Tropical Medicine & Parasitology (AREA)
- Biotechnology (AREA)
- Molecular Biology (AREA)
- Diabetes (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Psychiatry (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Transplantation (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US18984800P | 2000-03-16 | 2000-03-16 | |
PCT/US2001/008672 WO2001068084A1 (en) | 2000-03-16 | 2001-03-16 | Il-8 receptor antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
SK13282002A3 true SK13282002A3 (sk) | 2003-02-04 |
Family
ID=22699008
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SK1328-2002A SK13282002A3 (sk) | 2000-03-16 | 2001-03-16 | Sulfónamidové substituované difenylmočovinové zlúčeniny, farmaceutický prostriedok s ich obsahom a ich použitie |
Country Status (23)
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR030689A1 (es) * | 2000-03-14 | 2003-09-03 | Smithkline Beecham Corp | Compuestos de 3-aminosulfonil-2-hidroxifenil urea, composiciones farmaceuticas que los comprenden, y uso de dichos compuestos en la manufactura de medicamentos para tratar enfermedades mediadas por quimioquinas |
US7326729B2 (en) | 2004-05-12 | 2008-02-05 | Schering Corporation | CXCR1 and CXCR2 chemokine antagonists |
AU2007240364A1 (en) * | 2006-04-21 | 2007-11-01 | Smithkline Beecham Corporation | IL-8 receptor antagonists |
BRPI0710232B8 (pt) * | 2006-04-21 | 2021-05-25 | Glaxosmithkline Llc | composto antagonista do receptor de il-8, composição farmacêutica que compreende o dito composto e uso do mesmo para o tratamento de uma doença mediada por quimiocina |
CR20160557A (es) * | 2014-05-29 | 2017-01-20 | Glaxosmithkline Ip Dev Ltd | Compuestos derivados de 1-(ciclopent-2-en-1-il)-3-(2-hidroxi-3-(arilsulfonil)fenil)urea como inhibidores cxcr2 |
BR112017002060A2 (pt) * | 2014-07-31 | 2017-12-26 | Glaxosmithkline Ip Dev Ltd | novo uso |
JP7223764B2 (ja) * | 2018-01-11 | 2023-02-16 | シェンチェン オプティマム バイオロジカル テクノロジー カンパニー,リミティド | Cxcr2アンタゴニスト |
CN114286819B (zh) * | 2019-07-11 | 2024-03-05 | 深圳嘉科生物科技有限公司 | 一种cxcr2拮抗剂的晶型及其应用 |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH11503110A (ja) * | 1995-02-17 | 1999-03-23 | スミスクライン・ビーチャム・コーポレイション | Il−8受容体拮抗剤 |
CA2258850A1 (en) * | 1996-06-27 | 1997-12-31 | Smithkline Beecham Corporation | Il-8 receptor antagonists |
WO1998007418A1 (en) * | 1996-08-21 | 1998-02-26 | Smithkline Beecham Corporation | Il-8 receptor antagonists |
PT1115701E (pt) * | 1998-09-23 | 2003-09-30 | Tularik Inc | Ureias de arilsulfonanilida |
UY25842A1 (es) * | 1998-12-16 | 2001-04-30 | Smithkline Beecham Corp | Antagonistas de receptores de il-8 |
-
2001
- 2001-03-14 CO CO01020681A patent/CO5280089A1/es not_active Application Discontinuation
- 2001-03-14 AR ARP010101183A patent/AR031098A1/es unknown
- 2001-03-16 WO PCT/US2001/008672 patent/WO2001068084A1/en not_active Application Discontinuation
- 2001-03-16 AU AU2001250873A patent/AU2001250873A1/en not_active Abandoned
- 2001-03-16 OA OA1200200289A patent/OA12231A/en unknown
- 2001-03-16 HU HU0300470A patent/HUP0300470A3/hu unknown
- 2001-03-16 KR KR1020027012102A patent/KR20020091130A/ko not_active Withdrawn
- 2001-03-16 MX MXPA02009094A patent/MXPA02009094A/es active IP Right Grant
- 2001-03-16 EA EA200200981A patent/EA200200981A1/ru unknown
- 2001-03-16 DZ DZ013317A patent/DZ3317A1/fr active
- 2001-03-16 BR BR0108749-5A patent/BR0108749A/pt not_active Application Discontinuation
- 2001-03-16 EP EP01924195A patent/EP1263427A4/en not_active Withdrawn
- 2001-03-16 CA CA002403062A patent/CA2403062A1/en not_active Abandoned
- 2001-03-16 CN CN01806605A patent/CN1424910A/zh active Pending
- 2001-03-16 SK SK1328-2002A patent/SK13282002A3/sk unknown
- 2001-03-16 AP APAP/P/2002/002606A patent/AP2002002606A0/en unknown
- 2001-03-16 JP JP2001566648A patent/JP2003526664A/ja not_active Withdrawn
- 2001-03-16 CZ CZ20023075A patent/CZ20023075A3/cs unknown
- 2001-03-16 PL PL01366034A patent/PL366034A1/xx not_active Application Discontinuation
-
2002
- 2002-08-20 BG BG107013A patent/BG107013A/bg unknown
- 2002-09-12 MA MA26815A patent/MA25659A1/fr unknown
- 2002-09-12 ZA ZA200207325A patent/ZA200207325B/en unknown
- 2002-09-12 NO NO20024367A patent/NO20024367L/no unknown
Also Published As
Publication number | Publication date |
---|---|
DZ3317A1 (enrdf_load_stackoverflow) | 2001-09-20 |
OA12231A (en) | 2003-11-07 |
MXPA02009094A (es) | 2003-03-12 |
EP1263427A1 (en) | 2002-12-11 |
NO20024367L (no) | 2002-10-22 |
KR20020091130A (ko) | 2002-12-05 |
WO2001068084A1 (en) | 2001-09-20 |
BG107013A (bg) | 2003-05-30 |
NO20024367D0 (no) | 2002-09-12 |
AP2002002606A0 (en) | 2002-09-30 |
CA2403062A1 (en) | 2001-09-20 |
PL366034A1 (en) | 2005-01-24 |
AR031098A1 (es) | 2003-09-10 |
HUP0300470A3 (en) | 2005-05-30 |
JP2003526664A (ja) | 2003-09-09 |
CN1424910A (zh) | 2003-06-18 |
BR0108749A (pt) | 2004-06-29 |
EP1263427A4 (en) | 2005-08-24 |
ZA200207325B (en) | 2003-10-17 |
CZ20023075A3 (cs) | 2003-05-14 |
MA25659A1 (fr) | 2002-12-31 |
HUP0300470A2 (hu) | 2003-06-28 |
AU2001250873A1 (en) | 2001-09-24 |
EA200200981A1 (ru) | 2003-02-27 |
CO5280089A1 (es) | 2003-05-30 |
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