SI2571506T1 - Postopki za pripravo makrolidov in ketolidov ter njihovih intermediatov - Google Patents
Postopki za pripravo makrolidov in ketolidov ter njihovih intermediatovInfo
- Publication number
- SI2571506T1 SI2571506T1 SI201131256T SI201131256T SI2571506T1 SI 2571506 T1 SI2571506 T1 SI 2571506T1 SI 201131256 T SI201131256 T SI 201131256T SI 201131256 T SI201131256 T SI 201131256T SI 2571506 T1 SI2571506 T1 SI 2571506T1
- Authority
- SI
- Slovenia
- Prior art keywords
- ketolides
- processes
- intermediates therefor
- macrolides
- preparing
- Prior art date
Links
- 239000000543 intermediate Substances 0.000 title 1
- 239000003835 ketolide antibiotic agent Substances 0.000 title 1
- 239000003120 macrolide antibiotic agent Substances 0.000 title 1
- 229940041033 macrolides Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H1/00—Processes for the preparation of sugar derivatives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- General Chemical & Material Sciences (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US34666410P | 2010-05-20 | 2010-05-20 | |
| PCT/US2011/037330 WO2011146829A1 (en) | 2010-05-20 | 2011-05-20 | Processes for preparing macrolides and ketolides and intermediates therefor |
| EP11784318.5A EP2571506B1 (en) | 2010-05-20 | 2011-05-20 | Processes for preparing macrolides and ketolides and intermediates therefor |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SI2571506T1 true SI2571506T1 (sl) | 2017-12-29 |
Family
ID=44992076
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SI201131256T SI2571506T1 (sl) | 2010-05-20 | 2011-05-20 | Postopki za pripravo makrolidov in ketolidov ter njihovih intermediatov |
Country Status (15)
| Country | Link |
|---|---|
| US (4) | US9051346B2 (cg-RX-API-DMAC7.html) |
| EP (1) | EP2571506B1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP6184319B2 (cg-RX-API-DMAC7.html) |
| KR (1) | KR101945324B1 (cg-RX-API-DMAC7.html) |
| CN (2) | CN105198944B (cg-RX-API-DMAC7.html) |
| AU (1) | AU2011255464C1 (cg-RX-API-DMAC7.html) |
| BR (1) | BR112012029586A2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA2799937A1 (cg-RX-API-DMAC7.html) |
| DK (1) | DK2571506T3 (cg-RX-API-DMAC7.html) |
| ES (1) | ES2636948T3 (cg-RX-API-DMAC7.html) |
| IL (1) | IL223161A0 (cg-RX-API-DMAC7.html) |
| PL (1) | PL2571506T3 (cg-RX-API-DMAC7.html) |
| RU (1) | RU2608390C2 (cg-RX-API-DMAC7.html) |
| SI (1) | SI2571506T1 (cg-RX-API-DMAC7.html) |
| WO (1) | WO2011146829A1 (cg-RX-API-DMAC7.html) |
Families Citing this family (22)
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| CA2801100A1 (en) | 2003-03-10 | 2004-09-23 | Optimer Pharmaceuticals, Inc. | Macrolides and processes for their preparation |
| US8563573B2 (en) | 2007-11-02 | 2013-10-22 | Vertex Pharmaceuticals Incorporated | Azaindole derivatives as CFTR modulators |
| CA2703475A1 (en) | 2007-10-25 | 2009-04-30 | Cempra Pharmaceuticals, Inc. | Process for the preparation of macrolide antibacterial agents |
| CN102223794B (zh) | 2008-10-24 | 2017-12-22 | 森普拉制药公司 | 使用含三唑的大环内酯治疗抗性疾病的方法 |
| US9937194B1 (en) | 2009-06-12 | 2018-04-10 | Cempra Pharmaceuticals, Inc. | Compounds and methods for treating inflammatory diseases |
| CN108310000A (zh) | 2009-09-10 | 2018-07-24 | 森普拉制药公司 | 治疗疟疾、结核病和mac疾病的方法 |
| US8802868B2 (en) | 2010-03-25 | 2014-08-12 | Vertex Pharmaceuticals Incorporated | Solid forms of (R)-1(2,2-difluorobenzo[D][1,3]dioxo1-5-yl)-N-(1-(2,3-dihydroxypropyl-6-fluoro-2-(1-hydroxy-2-methylpropan2-yl)-1H-Indol-5-yl)-Cyclopropanecarboxamide |
| MX353408B (es) | 2010-04-22 | 2018-01-11 | Vertex Pharma | Proceso para producir compuestos de cicloalquilcarboxamido-indol. |
| CN105198944B (zh) * | 2010-05-20 | 2018-06-01 | 森普拉制药公司 | 制备大环内酯和酮内酯及其中间体的方法 |
| EP2613630A4 (en) | 2010-09-10 | 2014-01-15 | Cempra Pharmaceuticals Inc | HYDROGEN BOND FOR THE PREPARATION OF FLUOROCHETOLIDES FOR THE TREATMENT OF DISEASES |
| NZ700182A (en) | 2012-03-27 | 2017-02-24 | Cempra Pharmaceuticals Inc | Parenteral formulations for administering macrolide antibiotics |
| CN103897002A (zh) * | 2012-12-31 | 2014-07-02 | 菏泽市方明制药有限公司 | 一种粗品硫氰酸红霉素制备红霉素a9-肟的方法 |
| WO2014152326A1 (en) | 2013-03-14 | 2014-09-25 | Cempra Pharmaceuticals, Inc. | Methods for treating respiratory diseases and formulations therefor |
| WO2014145210A1 (en) * | 2013-03-15 | 2014-09-18 | Cempra Pharmaceuticals, Inc. | Convergent processes for preparing macrolide antibacterial agents |
| CN105246334A (zh) | 2013-04-04 | 2016-01-13 | 哈佛大学的校长及成员们 | 大环内酯及其制备和使用方法 |
| MX387720B (es) | 2014-04-15 | 2025-03-12 | Vertex Pharma | Composiciones farmacéuticas para el tratamiento de enfermedades mediadas por el regulador de conductancia de transmembrana de fibrosis quística. |
| CN104151382B (zh) * | 2014-08-08 | 2016-09-14 | 广东东阳光药业有限公司 | 一种固态大环内酯的晶型 |
| CN104311611B (zh) * | 2014-08-13 | 2017-01-18 | 广东东阳光药业有限公司 | 一种制备固态大环内酯的方法 |
| JP2017531663A (ja) | 2014-10-08 | 2017-10-26 | プレジデント アンド フェローズ オブ ハーバード カレッジ | 14員ケトライドならびにそれらの調製および使用の方法 |
| CA2980315A1 (en) | 2015-03-25 | 2016-09-29 | President And Fellows Of Harvard College | Macrolides with modified desosamine sugars and uses thereof |
| CN106554381A (zh) * | 2015-09-25 | 2017-04-05 | 苏州鹏旭医药科技有限公司 | 酮内酯类抗生素中间体及其制备方法和应用 |
| TW201811811A (zh) * | 2016-09-02 | 2018-04-01 | 森普拉製藥公司 | 製備氟酮內酯之方法 |
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2011
- 2011-05-20 CN CN201510604701.0A patent/CN105198944B/zh not_active Expired - Fee Related
- 2011-05-20 PL PL11784318T patent/PL2571506T3/pl unknown
- 2011-05-20 KR KR1020127032834A patent/KR101945324B1/ko not_active Expired - Fee Related
- 2011-05-20 EP EP11784318.5A patent/EP2571506B1/en not_active Not-in-force
- 2011-05-20 AU AU2011255464A patent/AU2011255464C1/en not_active Ceased
- 2011-05-20 RU RU2012150753A patent/RU2608390C2/ru not_active IP Right Cessation
- 2011-05-20 CN CN201180026739.4A patent/CN102917708B/zh not_active Expired - Fee Related
- 2011-05-20 BR BR112012029586A patent/BR112012029586A2/pt not_active IP Right Cessation
- 2011-05-20 WO PCT/US2011/037330 patent/WO2011146829A1/en not_active Ceased
- 2011-05-20 DK DK11784318.5T patent/DK2571506T3/en active
- 2011-05-20 JP JP2013511385A patent/JP6184319B2/ja active Active
- 2011-05-20 CA CA 2799937 patent/CA2799937A1/en not_active Abandoned
- 2011-05-20 SI SI201131256T patent/SI2571506T1/sl unknown
- 2011-05-20 US US13/699,020 patent/US9051346B2/en not_active Expired - Fee Related
- 2011-05-20 ES ES11784318.5T patent/ES2636948T3/es active Active
-
2012
- 2012-11-20 IL IL223161A patent/IL223161A0/en unknown
-
2015
- 2015-05-01 US US14/702,004 patent/US20150232500A1/en not_active Abandoned
-
2018
- 2018-03-06 US US15/913,650 patent/US20190048035A1/en not_active Abandoned
-
2019
- 2019-11-25 US US16/693,978 patent/US20200087335A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011146829A1 (en) | 2011-11-24 |
| RU2012150753A (ru) | 2014-06-27 |
| KR20130120374A (ko) | 2013-11-04 |
| EP2571506B1 (en) | 2017-05-10 |
| AU2011255464B2 (en) | 2016-06-16 |
| CN105198944B (zh) | 2018-06-01 |
| US20130066056A1 (en) | 2013-03-14 |
| JP6184319B2 (ja) | 2017-08-23 |
| ES2636948T3 (es) | 2017-10-10 |
| CN102917708A (zh) | 2013-02-06 |
| KR101945324B1 (ko) | 2019-02-07 |
| AU2011255464C1 (en) | 2017-02-23 |
| CN105198944A (zh) | 2015-12-30 |
| HK1181672A1 (zh) | 2013-11-15 |
| EP2571506A4 (en) | 2014-04-02 |
| BR112012029586A2 (pt) | 2016-08-02 |
| CN102917708B (zh) | 2015-11-25 |
| PL2571506T3 (pl) | 2017-10-31 |
| US20200087335A1 (en) | 2020-03-19 |
| CA2799937A1 (en) | 2011-11-24 |
| RU2608390C2 (ru) | 2017-01-18 |
| AU2011255464A1 (en) | 2012-12-13 |
| EP2571506A1 (en) | 2013-03-27 |
| US20150232500A1 (en) | 2015-08-20 |
| US9051346B2 (en) | 2015-06-09 |
| DK2571506T3 (en) | 2017-08-28 |
| JP2013527187A (ja) | 2013-06-27 |
| US20190048035A1 (en) | 2019-02-14 |
| IL223161A0 (en) | 2013-02-03 |
| HK1218919A1 (zh) | 2017-03-17 |
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