HK1181672A1 - 製備大環內酯和酮內酯及其中間體的方法 - Google Patents

製備大環內酯和酮內酯及其中間體的方法

Info

Publication number
HK1181672A1
HK1181672A1 HK13109063.8A HK13109063A HK1181672A1 HK 1181672 A1 HK1181672 A1 HK 1181672A1 HK 13109063 A HK13109063 A HK 13109063A HK 1181672 A1 HK1181672 A1 HK 1181672A1
Authority
HK
Hong Kong
Prior art keywords
ketolides
processes
intermediates therefor
macrolides
preparing
Prior art date
Application number
HK13109063.8A
Other languages
English (en)
Inventor
．佩雷拉
Original Assignee
森普拉制藥公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 森普拉制藥公司 filed Critical 森普拉制藥公司
Publication of HK1181672A1 publication Critical patent/HK1181672A1/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HK13109063.8A 2010-05-20 2013-08-02 製備大環內酯和酮內酯及其中間體的方法 HK1181672A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US34666410P 2010-05-20 2010-05-20
PCT/US2011/037330 WO2011146829A1 (en) 2010-05-20 2011-05-20 Processes for preparing macrolides and ketolides and intermediates therefor

Publications (1)

Publication Number Publication Date
HK1181672A1 true HK1181672A1 (zh) 2013-11-15

Family

ID=44992076

Family Applications (2)

Application Number Title Priority Date Filing Date
HK13109063.8A HK1181672A1 (zh) 2010-05-20 2013-08-02 製備大環內酯和酮內酯及其中間體的方法
HK16106890.0A HK1218919A1 (zh) 2010-05-20 2016-06-15 製備大環內酯和酮內酯及其中間體的方法

Family Applications After (1)

Application Number Title Priority Date Filing Date
HK16106890.0A HK1218919A1 (zh) 2010-05-20 2016-06-15 製備大環內酯和酮內酯及其中間體的方法

Country Status (16)

Country Link
US (4) US9051346B2 (zh)
EP (1) EP2571506B1 (zh)
JP (1) JP6184319B2 (zh)
KR (1) KR101945324B1 (zh)
CN (2) CN102917708B (zh)
AU (1) AU2011255464C1 (zh)
BR (1) BR112012029586A2 (zh)
CA (1) CA2799937A1 (zh)
DK (1) DK2571506T3 (zh)
ES (1) ES2636948T3 (zh)
HK (2) HK1181672A1 (zh)
IL (1) IL223161A0 (zh)
PL (1) PL2571506T3 (zh)
RU (1) RU2608390C2 (zh)
SI (1) SI2571506T1 (zh)
WO (1) WO2011146829A1 (zh)

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AU2011255464A1 (en) 2012-12-13
CA2799937A1 (en) 2011-11-24
EP2571506A4 (en) 2014-04-02
US20130066056A1 (en) 2013-03-14
AU2011255464B2 (en) 2016-06-16
SI2571506T1 (sl) 2017-12-29
KR101945324B1 (ko) 2019-02-07
IL223161A0 (en) 2013-02-03
US20150232500A1 (en) 2015-08-20
BR112012029586A2 (pt) 2016-08-02
EP2571506B1 (en) 2017-05-10
DK2571506T3 (en) 2017-08-28
RU2012150753A (ru) 2014-06-27
JP2013527187A (ja) 2013-06-27
CN105198944B (zh) 2018-06-01
ES2636948T3 (es) 2017-10-10
US20190048035A1 (en) 2019-02-14
HK1218919A1 (zh) 2017-03-17
PL2571506T3 (pl) 2017-10-31
WO2011146829A1 (en) 2011-11-24
RU2608390C2 (ru) 2017-01-18
CN102917708A (zh) 2013-02-06
US20200087335A1 (en) 2020-03-19
US9051346B2 (en) 2015-06-09
CN102917708B (zh) 2015-11-25
AU2011255464C1 (en) 2017-02-23
JP6184319B2 (ja) 2017-08-23
CN105198944A (zh) 2015-12-30
KR20130120374A (ko) 2013-11-04
EP2571506A1 (en) 2013-03-27

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