SI2364302T1 - Tirazinski analogi in njihova uporaba kot terapevtska sredstva in diagnostične sonde - Google Patents
Tirazinski analogi in njihova uporaba kot terapevtska sredstva in diagnostične sondeInfo
- Publication number
- SI2364302T1 SI2364302T1 SI200931578A SI200931578A SI2364302T1 SI 2364302 T1 SI2364302 T1 SI 2364302T1 SI 200931578 A SI200931578 A SI 200931578A SI 200931578 A SI200931578 A SI 200931578A SI 2364302 T1 SI2364302 T1 SI 2364302T1
- Authority
- SI
- Slovenia
- Prior art keywords
- therapeutic agents
- diagnostic probes
- triazine analogs
- triazine
- analogs
- Prior art date
Links
- 239000003814 drug Substances 0.000 title 1
- 239000000523 sample Substances 0.000 title 1
- 229940124597 therapeutic agent Drugs 0.000 title 1
- 150000003918 triazines Chemical class 0.000 title 1
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- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/444—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
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- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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PCT/IB2009/007404 WO2010052569A2 (en) | 2008-11-10 | 2009-11-10 | Triazine, pyrimidine and pyridine analogs and their use as therapeutic agents and diagnostic probes |
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EP2532667A1 (en) * | 2005-09-30 | 2012-12-12 | Vertex Pharmaceuticals Incorporated | Deazapurines useful as inhibitors of janus kinases |
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AU2007243457B2 (en) | 2006-04-26 | 2012-02-23 | F. Hoffmann-La Roche Ag | Pharmaceutical compounds |
PT2050749T (pt) * | 2006-08-08 | 2018-01-02 | Chugai Pharmaceutical Co Ltd | Derivado de pirimidina como inibidador de pi3k e sua utilização |
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EP2118087B1 (en) * | 2007-02-06 | 2012-03-28 | Novartis AG | Pi 3-kinase inhibitors and methods of their use |
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DE202008001253U1 (de) * | 2008-01-28 | 2008-04-10 | Mirror Image Ag | Bildanzeigegerät |
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GB2465405A (en) * | 2008-11-10 | 2010-05-19 | Univ Basel | Triazine, pyrimidine and pyridine analogues and their use in therapy |
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2008
- 2008-11-10 GB GB0821219A patent/GB2465405A/en not_active Withdrawn
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2009
- 2009-11-10 NZ NZ592617A patent/NZ592617A/en active IP Right Revival
- 2009-11-10 US US13/128,436 patent/US8921361B2/en active Active
- 2009-11-10 MX MX2011004889A patent/MX2011004889A/es active IP Right Grant
- 2009-11-10 BR BRPI0921709-6A patent/BRPI0921709B1/pt active IP Right Grant
- 2009-11-10 KR KR1020117013081A patent/KR101749192B1/ko active IP Right Grant
- 2009-11-10 JP JP2011535182A patent/JP5738768B2/ja active Active
- 2009-11-10 LT LTEP09764032.0T patent/LT2364302T/lt unknown
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- 2009-11-10 DK DK09764032.0T patent/DK2364302T3/en active
- 2009-11-10 ES ES09764032.0T patent/ES2609296T3/es active Active
- 2009-11-10 CN CN200980144674.6A patent/CN102209714B/zh active Active
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- 2009-11-10 RU RU2011114559/04A patent/RU2537945C2/ru active
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